Structure–Activity Relationship Studies of Acetazolamide-Based Carbonic Anhydrase Inhibitors with Activity against Neisseria gonorrhoeae CS Hewitt, NS Abutaleb, AEM Elhassanny, A Nocentini, X Cao, DP Amos, ... ACS infectious diseases 7 (7), 1969-1984, 2021 | 66 | 2021 |
Identification, biochemical and structural evaluation of species-specific inhibitors against type I methionine aminopeptidases C Kishor, T Arya, R Reddi, X Chen, V Saddanapu, AK Marapaka, ... Journal of medicinal chemistry 56 (13), 5295-5305, 2013 | 34 | 2013 |
Single pot green synthesis, characterization, antitumor antibacterial, antioxidant activity of bimetallic silver and copper nanoparticles using fruit pulp of palmyra fruit KL Chitturi, S Garimella, AK Marapaka, KR Kudle, R Merugu Journal of Bionanoscience 12 (2), 284-289, 2018 | 31 | 2018 |
Highly functionalized tetrahydropyridines are cytotoxic and selective inhibitors of human puromycin sensitive aminopeptidase R Aeluri, RJ Ganji, AK Marapaka, V Pillalamarri, M Alla, A Addlagatta European Journal of Medicinal Chemistry 106, 26-33, 2015 | 20 | 2015 |
Structural basis for the inhibition of M1 family aminopeptidases by the natural product actinonin: Crystal structure in complex with E. coli aminopeptidase N RJ Ganji, R Reddi, R Gumpena, AK Marapaka, T Arya, P Sankoju, ... Protein Science 24 (5), 823-831, 2015 | 20 | 2015 |
Structural Characterization of Thiadiazolesulfonamide Inhibitors Bound to Neisseria gonorrhoeae α-Carbonic Anhydrase AK Marapaka, A Nocentini, MS Youse, W An, KJ Holly, C Das, R Yadav, ... ACS Medicinal Chemistry Letters 14 (1), 103-109, 2022 | 16 | 2022 |
Aminobenzosuberone scaffold as a modular chemical tool for the inhibition of therapeutically relevant M1 aminopeptidases E Salomon, M Schmitt, AK Marapaka, A Stamogiannos, G Revelant, ... Molecules 23 (10), 2607, 2018 | 13 | 2018 |
Discovery of natural product ovalicin sensitive type 1 methionine aminopeptidases: molecular and structural basis V Pillalamarri, T Arya, N Haque, SC Bala, AK Marapaka, A Addlagatta Biochemical Journal 476 (6), 991-1003, 2019 | 12 | 2019 |
Discovery of a new class of type 1 methionine aminopeptidases that have relaxed substrate specificity SC Bala, N Haque, V Pillalamarri, R Reddi, R Kashyap, AK Marapaka, ... International journal of biological macromolecules 129, 523-529, 2019 | 11 | 2019 |
Development of peptidomimetic hydroxamates as PfA-M1 and PfA-M17 dual inhibitors: Biological evaluation and structural characterization by cocrystallization AK Marapaka, P Sankoju, G Zhang, Y Ding, C Ma, V Pillalamarri, ... Chinese Chemical Letters 33 (5), 2550-2554, 2022 | 8 | 2022 |
Inhibition of pathogenic bacterial carbonic anhydrases by monothiocarbamates S Giovannuzzi, AK Marapaka, NS Abutaleb, F Carta, HW Liang, ... Journal of Enzyme Inhibition and Medicinal Chemistry 38 (1), 2284119, 2023 | 7 | 2023 |
Puromycin, a selective inhibitor of PSA acts as a substrate for other M1 family aminopeptidases: Biochemical and structural basis R Reddi, RJ Ganji, AK Marapaka, SC Bala, NV Yerra, N Haque, ... International Journal of Biological Macromolecules 165, 1373-1381, 2020 | 7 | 2020 |
Discovery, structural and biochemical studies of a rare Glu/Asp specific M1 class aminopeptidase from Legionella pneumophila AK Marapaka, V Pillalamarri, R Gumpena, N Haque, SC Bala, A Jangam, ... International journal of biological macromolecules 120, 1111-1118, 2018 | 6 | 2018 |
Development of selective inhibitors against malarial M1 family aminopeptidase A Addlagatta, AK Marapaka ACTA CRYSTALLOGRAPHICA A-FOUNDATION AND ADVANCES 73, C237-C237, 2017 | 1 | 2017 |
Study of quinoxaline-based new compounds against aminopeptidase N, and Plasmodium falciparum malarial parasite A Addlagatta, R Gumpena, A Marapaka, AD Allanki, JH Jun, PS Sijwali, ... ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 247, 2014 | 1 | 2014 |
Synthesis, Characterization and in vitro Studies of Metal Complexes Derived from Isoxazole Schiff base RMPMR Karunakar Dasa1*, Bhaskar Saggella2, Anil Kumar Marapaka3, Karunakar ... Journal of Applicable Chemistry 8 (4), 1568-1577, 2019 | | 2019 |
Understanding the Structural Differences Among M1-class Aminopeptidases and Development of Novel Inhibitors AK MARAPAKA CSIR-Indian Institute of Chemical Technology, Hyderabad, 2018 | | 2018 |
Understanding the structural basis of legionella pneumophila aminopeptidase N AK Marapaka, A Addlagatta ACTA CRYSTALLOGRAPHICA A-FOUNDATION AND ADVANCES 73, C158-C158, 2017 | | 2017 |
MS001. P05 AK Marapaka, A Addlagatta Acta Cryst 70, C158, 2017 | | 2017 |
MS009. P13 A Addlagatta, AK Marapaka Acta Cryst 70, C237, 2017 | | 2017 |