Design, synthesis, and docking studies of new 1, 3, 4-thiadiazole-2-thione derivatives with carbonic anhydrase inhibitory activity MK Abdel-Hamid, AA Abdel-Hafez, NA El-Koussi, NM Mahfouz, ... Bioorganic & medicinal chemistry 15 (22), 6975-6984, 2007 | 106 | 2007 |
HIV protease inhibitors: peptidomimetic drugs and future perspectives HM Abdel-Rahman, GS Al-karamany, NA El-Koussi, AF Youssef, Y Kiso Current medicinal chemistry 9 (21), 1905-1922, 2002 | 84 | 2002 |
Synthesis of 5‐Phenyl‐1‐(3‐pyridyl)‐1H‐1,2,4‐triazole‐3‐carboxylic Acid Derivatives of Potential Anti‐inflammatory Activity SM Rabea, NA El‐Koussi, HY Hassan, T Aboul‐Fadl Archiv der Pharmazie: An International Journal Pharmaceutical and Medicinal …, 2006 | 72 | 2006 |
Design, synthesis, and biological evaluation of new pyrimidine-5-carbonitrile derivatives bearing 1, 3-thiazole moiety as novel anti-inflammatory EGFR inhibitors with cardiac … SA Abdel-Aziz, ES Taher, P Lan, GF Asaad, HAM Gomaa, NA El-Koussi, ... Bioorganic Chemistry 111, 104890, 2021 | 49 | 2021 |
Fluorinated 1,2,4‐Triazolo[1,5‐a]pyrimidine‐6‐carboxylic Acid Derivatives as Antimycobacterial Agents HM Abdel‐Rahman, NA El‐Koussi, HY Hassan Archiv der Pharmazie: An International Journal Pharmaceutical and Medicinal …, 2009 | 48 | 2009 |
Synthesis and antimicrobial activity of pyridines bearing thiazoline and thiazolidinone moieties HY Hassan, NA El-Koussi, ZS Farghaly Chemical and pharmaceutical bulletin 46 (5), 863-866, 1998 | 47 | 1998 |
Design, synthesis, and antibacterial evaluation of new quinoline-1, 3, 4-oxadiazole and quinoline-1, 2, 4-triazole hybrids as potential inhibitors of DNA gyrase and … HA Hofny, MFA Mohamed, HAM Gomaa, SA Abdel-Aziz, BGM Youssif, ... Bioorganic Chemistry 112, 104920, 2021 | 45 | 2021 |
Brain delivery of HIV protease inhibitors MM Sheha, NA El‐Koussi, HH Farag Archiv der Pharmazie: An International Journal Pharmaceutical and Medicinal …, 2003 | 30 | 2003 |
Cu (I) catalyzed alkyne-azide 1, 3-dipolar cycloaddition (CuAAC): Synthesis of 17α-[1-(substituted phenyl)-1, 2, 3-triazol-4-yl]-19-nor-testosterone-17β-yl acetates targeting … ZH Mohamed, NA El-Koussi, NM Mahfouz, AF Youssef, GAA Jaleel, ... European Journal of Medicinal Chemistry 97, 75-82, 2015 | 16 | 2015 |
Design and synthesis of'some new 1H-1, 2, 4-triazoles of potential anti-inflammatory and analgesic activities HY Hassan, ANA El-Shorbagi, NA El-Koussi, AO Abdel-Zaher Bulletin of Pharmaceutical Sciences Assiut University 17 (1), 27-39, 1994 | 15 | 1994 |
New pyrimidine/thiazole hybrids endowed with analgesic, anti‐inflammatory, and lower cardiotoxic activities: Design, synthesis, and COX‐2/sEH dual inhibition SA Abdel‐Aziz, ES Taher, P Lan, NA El‐Koussi, OIA Salem, HAM Gomaa, ... Archiv der Pharmazie 355 (7), 2200024, 2022 | 11 | 2022 |
Synthesis and Antibacterial Screening Of Some 2, 5, 7triaryl-1, 2, 4-Triazolo [1, 5-a] PYRIMIDINES NA El-Koussi, FA Omar, SA Abdel-Aziz, MF Radwan Bulletin of Pharmaceutical Sciences Assiut University 27 (1), 144-154, 2004 | 11 | 2004 |
SYNTHESIS AND INVESTIGATION OF CERTAIN 3 (5)-SUBSTITUFED-1, 2, 4-TRIAZOLE-5 (3)-CARBOXYLIC ACID DERIVATIVES AA Abd-Elhafez, HM Mohamed, HY Hassan, GS El-Karamany, ... Bulletin of Pharmaceutical Sciences Assiut University 20 (1), 47-61, 1997 | 10 | 1997 |
Quantitative structure–activity relationship (QSAR) studies on a series of 1, 3, 4-thiadiazole-2-thione derivatives as tumor-associated carbonic anhydrase IX inhibitors MK Abdel-Hamid, AA Abdel-Hafez, NA El-Koussi, NM Mahfouz Journal of Enzyme Inhibition and Medicinal Chemistry 24 (3), 722-729, 2009 | 9 | 2009 |
Conjugate reduction-initiated tandem cyclization of a chiral α, β, χ, ψ–unsaturated bisphosphine oxide Y Nagaoka, N El-Koussi, S Uesato, K Tomioka Tetrahedron letters 43 (24), 4355-4359, 2002 | 9 | 2002 |
Synthesis and application of chiral bisphosphines through lithiation–conjugate addition tandem cyclization of chiral α, β, ψ, ω-unsaturated bisphosphine oxide Y Nagaoka, H Inoue, N El-Koussi, K Tomioka Chemical communications, 122-123, 2002 | 5 | 2002 |
SYNTHESIS OF 2-TRIFLUOROMETHYL-4, 7-DIHYDRO-7-OXO-(1, 2, 4) TRIAZOLO [1, 5-a] PYRIMIDINE-6-CARBOXYLIC ACID DERIVATIVES AS POTENTIAL ANTIMYCOBACTERIAL AND ANTIMICROBIAL AGENTS NA El-Koussi Bulletin of Pharmaceutical Sciences Assiut University 31 (1), 109-121, 2008 | 3 | 2008 |
Chemometrics assisted spectrophotometric method for simultaneous determination of certain fluoroquinolones and their decarboxylated degradants AI Mohamed, NA El-Koussi, NA Mohamed Bulletin of Pharmaceutical Sciences Assiut University 28 (2), 191-198, 2005 | 2 | 2005 |
A Novel Dipeptide‐based HIV Protease Inhibitor Containing Allophenylnorstatine HM Abdel‐Rahman, NA El‐Koussi, GS Alkaramany, AF Youssef, Y Kiso Archiv der Pharmazie: An International Journal Pharmaceutical and Medicinal …, 2004 | 2 | 2004 |
Recent progress in biological activities of dihydropyrimidine derivatives: An updated mini-review AM Elshamsy, TFS Ali, M Osman, NA El-Koussi Journal of advanced Biomedical and Pharmaceutical Sciences 6 (3), 114-123, 2023 | 1 | 2023 |