1, 4‐Diazabicyclo [2.2. 2] octane (DABCO) as an Efficient Reagent for the Synthesis of Isoxazole Derivatives from Primary Nitro Compounds and Dipolarophiles: The Role of the Base L Cecchi, F De Sarlo, F Machetti European Journal of Organic Chemistry 2006 (21), 4852-4860, 2006 | 104 | 2006 |
Synthesis of 4, 5‐Dihydroisoxazoles by Condensation of Primary Nitro Compounds with Alkenes by Using a Copper/Base Catalytic System L Cecchi, F De Sarlo, F Machetti Chemistry–A European Journal 14 (26), 7903-7912, 2008 | 78 | 2008 |
19-Nor-10-azasteroids: a novel class of inhibitors for human steroid 5α-reductases 1 and 2 A Guarna, C Belle, F Machetti, EG Occhiato, AH Payne, C Cassiani, ... Journal of medicinal chemistry 40 (7), 1112-1129, 1997 | 74 | 1997 |
Interactions of taurine and structurally related analogues with the GABAergic system and taurine binding sites of rabbit brain M Frosini, C Sesti, S Dragoni, M Valoti, M Palmi, HBF Dixon, F Machetti, ... British journal of pharmacology 138 (6), 1163-1171, 2003 | 65 | 2003 |
Acid–Base‐Catalysed Condensation Reaction in Water: Isoxazolines and Isoxazoles from Nitroacetates and Dipolarophiles E Trogu, C Vinattieri, F De Sarlo, F Machetti Chemistry–A European Journal 18 (7), 2081-2093, 2012 | 62 | 2012 |
Isoxazoline derivatives from activated primary nitrocompounds and tertiary diamines L Cecchi, F De Sarlo, F Machetti Tetrahedron letters 46 (46), 7877-7879, 2005 | 57 | 2005 |
A specific taurine recognition site in the rabbit brain is responsible for taurine effects on thermoregulation M Frosini, C Sesti, S Saponara, L Ricci, M Valoti, M Palmi, F Machetti, ... British journal of pharmacology 139 (3), 487-494, 2003 | 57 | 2003 |
Synthesis and reactivity of bicycles derived from tartaric acid and α-amino acids: a novel class of conformationally constrained dipeptide isosteres based upon enantiopure 3 … A Guarna, A Guidi, F Machetti, G Menchi, EG Occhiato, D Scarpi, S Sisi, ... The Journal of Organic Chemistry 64 (20), 7347-7364, 1999 | 57 | 1999 |
Isoxazoles D Giomi, F Cordero, F Machetti Comprehensive Heterocyclic Chemistry, 365-486, 2008 | 55 | 2008 |
Isoxazoles and Isoxazolines by 1, 3‐Dipolar Cycloaddition: Base‐Catalysed Condensation of Primary Nitro Compounds with Dipolarophiles F Machetti, L Cecchi, E Trogu, F De Sarlo European Journal of Organic Chemistry 2007 (26), 4352-4359, 2007 | 51 | 2007 |
Michael Additions versus Cycloaddition Condensations with Ethyl Nitroacetate and Electron‐Deficient Olefins E Trogu, F De Sarlo, F Machetti Chemistry–A European Journal 15 (32), 7940-7948, 2009 | 49 | 2009 |
Comprehensive Heterocyclic Chemistry III D Giomi, FM Cordero, F Machetti, A Katritzky, C Ramsden, RT E Scriven Elsevier: Oxford 4, 2008 | 47 | 2008 |
A new synthesis of (2S)-4-oxopipecolic acid by thermal rearrangement of enantiopure spirocyclopropaneisoxazolidine F Machetti, FM Cordero, F De Sarlo, A Guarna, A Brandi Tetrahedron letters 37 (24), 4205-4208, 1996 | 47 | 1996 |
Conjugate Addition versus Cycloaddition/Condensation of Nitro Compounds in Water: Selectivity, Acid–Base Catalysis, and Induction Period L Guideri, F De Sarlo, F Machetti Chemistry–A European Journal 19 (2), 665-677, 2013 | 42 | 2013 |
A new bicyclic dipeptide isostere with pyrrolizidinone skeleton FM Cordero, F Pisaneschi, K Meschini Batista, S Valenza, F Machetti, ... The Journal of Organic Chemistry 70 (3), 856-867, 2005 | 42 | 2005 |
Benzo[c]quinolizin-3-ones: A Novel Class of Potent and Selective Nonsteroidal Inhibitors of Human Steroid 5α-Reductase 1 A Guarna, F Machetti, EG Occhiato, D Scarpi, A Comerci, G Danza, ... Journal of medicinal chemistry 43 (20), 3718-3735, 2000 | 39 | 2000 |
Synthesis of a new enantiopure bicyclic γ/δ-amino acid (BTKa) derived from tartaric acid and α-amino acetophenone A Guarna, I Bucelli, F Machetti, G Menchi, EG Occhiato, D Scarpi, ... Tetrahedron 58 (49), 9865-9870, 2002 | 38 | 2002 |
A CONCISE ROUTE TO 19-NOR-10-AZASTEROIDS, A NEW CLASS OF STEROID 5-REDUCTASE INHIBITORS. 3.1 SYNTHESIS OF (+)-19-NOR-10-AZATESTOSTERONE AND (+)-17B-ACETYLOXY-(5B)-10-AZAESTR-1 … A Guarna, EG Occhiato, F Machetti, D Scarpi Journal of organic chemistry 63, 4111-4115, 1998 | 37 | 1998 |
Identification of Inhibitors of Drug-Resistant Candida albicans Strains from a Library of Bicyclic Peptidomimetic Compounds A Trabocchi, C Mannino, F Machetti, F De Bernardis, S Arancia, R Cauda, ... Journal of medicinal chemistry 53 (6), 2502-2509, 2010 | 36 | 2010 |
Design, synthesis, and applications of 3-aza-6, 8-dioxabicyclo [3.2. 1] octane-based scaffolds for peptidomimetic chemistry A Trabocchi, G Menchi, F Guarna, F Machetti, D Scarpi, A Guarna Synlett 2006 (03), 0331-0353, 2006 | 36 | 2006 |