| Design, synthesis and biological evaluation of novel potent MDM2/p53 small-molecule inhibitors YA Ivanenkov, SV Vasilevski, EK Beloglazkina, ME Kukushkin, ... Bioorganic & Medicinal Chemistry Letters 25 (2), 404-409, 2015 | 84 | 2015 |
| Small-molecule PSMA ligands. Current state, SAR and perspectives AE Machulkin, YA Ivanenkov, AV Aladinskaya, MS Veselov, VA Aladinskiy, ... Journal of drug targeting 24 (8), 679-693, 2016 | 61 | 2016 |
| Synthesis and biological evaluation of PSMA ligands with aromatic residues and fluorescent conjugates based on them AE Machulkin, RR Shafikov, AA Uspenskaya, SA Petrov, AP Ber, ... Journal of Medicinal Chemistry 64 (8), 4532-4552, 2021 | 28 | 2021 |
| Synthesis and biological evaluation of PSMA-targeting paclitaxel conjugates AE Machulkin, DA Skvortsov, YA Ivanenkov, AP Ber, MV Kavalchuk, ... Bioorganic & Medicinal Chemistry Letters 29 (16), 2229-2235, 2019 | 27 | 2019 |
| Synthesis and biological evaluation of Doxorubicin-containing conjugate targeting PSMA YA Ivanenkov, AE Machulkin, AS Garanina, DA Skvortsov, ... Bioorganic & medicinal chemistry letters 29 (10), 1246-1255, 2019 | 25 | 2019 |
| PSMA-targeted small-molecule docetaxel conjugate: Synthesis and preclinical evaluation AE Machulkin, AA Uspenskaya, NY Zyk, EA Nimenko, AP Ber, SA Petrov, ... European Journal of Medicinal Chemistry 227, 113936, 2022 | 19 | 2022 |
| Synthesis, characterization, and preclinical evaluation of a small-molecule prostate-specific membrane antigen-targeted monomethyl auristatin E conjugate AE Machulkin, AA Uspenskaya, NU Zyk, EA Nimenko, AP Ber, SA Petrov, ... Journal of Medicinal Chemistry 64 (23), 17123-17145, 2021 | 16 | 2021 |
| Polypeptide-based molecular platform and its docetaxel/sulfo-Cy5-containing conjugate for targeted delivery to prostate specific membrane antigen SA Petrov, AE Machulkin, AA Uspenskaya, NY Zyk, EA Nimenko, ... Molecules 25 (24), 5784, 2020 | 16 | 2020 |
| Nanohybride materials based on magnetite-gold nanoparticles for diagnostics of prostate cancer: synthesis and in vitro testing AE Machulkin, AS Garanina, OA Zhironkina, EK Beloglazkina, NV Zyk, ... Bull Exp Biol Med 161 (5), 706-710, 2016 | 13 | 2016 |
| 2-Pyrazol-1-yl-thiazole derivatives as novel highly potent antibacterials YA Ivanenkov, RS Yamidanov, IA Osterman, PV Sergiev, VA Aladinskiy, ... The Journal of antibiotics 72 (11), 827-833, 2019 | 12 | 2019 |
| Synthesis of PSMA-targeted 131- and 152-substituted chlorin e6 derivatives and their biological properties NV Suvorov, AE Machulkin, AV Ivanova, AM Popkov, EA Bondareva, ... Journal of Porphyrins and Phthalocyanines 22 (11), 1030-1038, 2018 | 12 | 2018 |
| PSMA-targeted low-molecular double conjugates for diagnostics and therapy SA Petrov, NY Zyk, AE Machulkin, EK Beloglazkina, AG Majouga European Journal of Medicinal Chemistry 225, 113752, 2021 | 10 | 2021 |
| The importance of linkers in the structure of PSMA ligands AA Uspenskaya, EA Nimenko, AE Machulkin, EK Beloglazkina, ... Current Medicinal Chemistry 29 (2), 268-298, 2022 | 9 | 2022 |
| Synthesis and organogelating behaviour of urea-and Fmoc-containing diphenylalanine based hexaamide SA Petrov, AE Machulkin, RA Petrov, AN Tavtorkin, GN Bondarenko, ... Journal of Molecular Structure 1234, 130127, 2021 | 8 | 2021 |
| Identification of pyrrolo-pyridine derivatives as novel class of antibacterials MS Veselov, YA Ivanenkov, RS Yamidanov, IA Osterman, PV Sergiev, ... Molecular Diversity 24, 233-239, 2020 | 8 | 2020 |
| Pharmacokinetic Properties of 68Ga-labelled Folic Acid Conjugates: Improvement Using HEHE Tag A Larenkov, M Rakhimov, K Lunyova, O Klementyeva, A Maruk, ... Molecules 25 (11), 2712, 2020 | 7 | 2020 |
| Bifunctional magnetite–gold nanoparticles for magneto-mechanical actuation and cancer cell destruction AS Garanina, MV Efremova, AE Machulkin, EV Lyubin, NS Vorobyeva, ... Magnetochemistry 8 (12), 185, 2022 | 6 | 2022 |
| Influence of the dipeptide linker configuration on the activity of PSMA ligands AA Uspenskaya, AE Machulkin, EA Nimenko, RR Shafikov, SA Petrov, ... Mendeleev Communications 30 (6), 756-759, 2020 | 6 | 2020 |
| Synthesis and Preclinical Evaluation of Small-Molecule Prostate-Specific Membrane Antigen-Targeted Abiraterone Conjugate AE Machulkin, EA Nimenko, NU Zyk, AA Uspenskaia, GB Smirnova, ... Molecules 27 (24), 8795, 2022 | 5 | 2022 |
| Synthesis and initial in vitro evaluation of PSMA-targeting ligands with a modified aromatic moiety at the lysine ε-nitrogen atom NY Zyk, AP Ber, EA Nimenko, RR Shafikov, SA Evteev, SA Petrov, ... Bioorganic & Medicinal Chemistry Letters 71, 128840, 2022 | 5 | 2022 |
