Inhibition of neuronal nitric oxide synthase activity by N1‐acetyl‐5‐methoxykynuramine, a brain metabolite of melatonin J León, G Escames, MI Rodríguez, LC López, V Tapias, A Entrena, ... Journal of neurochemistry 98 (6), 2023-2033, 2006 | 202 | 2006 |
Synthesis and antitumor activity of 1, 5-disubstituted 1, 2, 4-triazoles as cis-restricted combretastatin analogues R Romagnoli, PG Baraldi, O Cruz-Lopez, C Lopez Cara, MD Carrion, ... Journal of medicinal chemistry 53 (10), 4248-4258, 2010 | 194 | 2010 |
Synthesis and Biological Evaluation of 2- and 3-Aminobenzo[b]thiophene Derivatives as Antimitotic Agents and Inhibitors of Tubulin Polymerization R Romagnoli, PG Baraldi, MD Carrion, CL Cara, D Preti, F Fruttarolo, ... Journal of medicinal chemistry 50 (9), 2273-2277, 2007 | 180 | 2007 |
Effects of estrogen or estrogen/progestin regimens on heart disease risk factors in postmenopausal women: the postmenopausal estrogen/progestin interventions (PEPI) trial VT Miller, J LaRosa, V Barnabei, C Kessler, G Levin, A Smith-Roth, ... Jama 273 (3), 199-208, 1995 | 169 | 1995 |
Design, synthesis, and biological evaluation of thiophene analogues of chalcones R Romagnoli, PG Baraldi, MD Carrion, CL Cara, O Cruz-Lopez, D Preti, ... Bioorganic & medicinal chemistry 16 (10), 5367-5376, 2008 | 157 | 2008 |
Organocatalytic Approach to Benzofused Nitrogen‐Containing Heterocycles: Enantioselective Total Synthesis of (+)‐Angustureine. S Fustero, J Moscardo, D Jimenez, MD Pérez‐Carrión, ... ChemInform 40 (11), no-no, 2009 | 150 | 2009 |
Melatonin and its brain metabolite N1‐acetyl‐5‐methoxykynuramine prevent mitochondrial nitric oxide synthase induction in parkinsonian mice V Tapias, G Escames, LC López, A Lopez, E Camacho, MD Carrión, ... Journal of neuroscience research 87 (13), 3002-3010, 2009 | 136 | 2009 |
Synthesis and biological evaluation of 1-methyl-2-(3′, 4′, 5′-trimethoxybenzoyl)-3-aminoindoles as a new class of antimitotic agents and tubulin inhibitors R Romagnoli, PG Baraldi, T Sarkar, MD Carrion, CL Cara, O Cruz-Lopez, ... Journal of medicinal chemistry 51 (5), 1464-1468, 2008 | 119 | 2008 |
Design, synthesis and structure–activity relationship of 2-(3′, 4′, 5′-trimethoxybenzoyl)-benzo [b] furan derivatives as a novel class of inhibitors of tubulin polymerization R Romagnoli, PG Baraldi, MD Carrion, CL Cara, O Cruz-Lopez, ... Bioorganic & medicinal chemistry 17 (19), 6862-6871, 2009 | 90 | 2009 |
4,5-Dihydro-1H-pyrazole Derivatives with Inhibitory nNOS Activity in Rat Brain: Synthesis and Structure−Activity Relationships ME Camacho, J León, A Entrena, G Velasco, MD Carrión, G Escames, ... Journal of medicinal chemistry 47 (23), 5641-5650, 2004 | 88 | 2004 |
Hybrid α-bromoacryloylamido chalcones. Design, synthesis and biological evaluation R Romagnoli, PG Baraldi, MD Carrion, O Cruz-Lopez, CL Cara, ... Bioorganic & Medicinal Chemistry Letters 19 (7), 2022-2028, 2009 | 72 | 2009 |
Synthesis and biological evaluation of 2-(3 ‘, 4 ‘, 5 ‘-trimethoxybenzoyl)-3-amino 5-aryl thiophenes as a new class of tubulin inhibitors R Romagnoli, PG Baraldi, V Remusat, MD Carrion, CL Cara, D Preti, ... Journal of medicinal chemistry 49 (21), 6425-6428, 2006 | 72 | 2006 |
2-Arylamino-4-amino-5-aroylthiazoles.“One-pot” synthesis and biological evaluation of a new class of inhibitors of tubulin polymerization R Romagnoli, PG Baraldi, MD Carrion, O Cruz-Lopez, C Lopez Cara, ... Journal of medicinal chemistry 52 (17), 5551-5555, 2009 | 68 | 2009 |
Kynurenamines as neural nitric oxide synthase inhibitors A Entrena, ME Camacho, MD Carrión, LC López-Cara, G Velasco, J León, ... Journal of medicinal chemistry 48 (26), 8174-8181, 2005 | 66 | 2005 |
Synthesis and biological evaluation of 2-(3′, 4′, 5′-trimethoxybenzoyl)-3-N, N-dimethylamino benzo [b] furan derivatives as inhibitors of tubulin polymerization R Romagnoli, PG Baraldi, T Sarkar, MD Carrion, O Cruz-Lopez, CL Cara, ... Bioorganic & medicinal chemistry 16 (18), 8419-8426, 2008 | 65 | 2008 |
Pyrazoles and pyrazolines as neural and inducible nitric oxide synthase (nNOS and iNOS) potential inhibitors (III) MD Carrión, LCL Cara, ME Camacho, V Tapias, G Escames, ... European journal of medicinal chemistry 43 (11), 2579-2591, 2008 | 61 | 2008 |
Synthesis and biological evaluation of 2-amino-3-(4-chlorobenzoyl)-4-[N-(substituted) piperazin-1-yl] thiophenes as potent allosteric enhancers of the A1 adenosine receptor R Romagnoli, PG Baraldi, MD Carrion, CL Cara, O Cruz-Lopez, ... Journal of medicinal chemistry 51 (18), 5875-5879, 2008 | 56 | 2008 |
Substituted 2-(3′, 4′, 5′-trimethoxybenzoyl)-benzo [b] thiophene derivatives as potent tubulin polymerization inhibitors R Romagnoli, PG Baraldi, MD Carrion, O Cruz-Lopez, M Tolomeo, ... Bioorganic & medicinal chemistry 18 (14), 5114-5122, 2010 | 54 | 2010 |
Allosteric enhancers for A1 adenosine receptor. PG Baraldi, MA Iaconinoto, AR Moorman, MD Carrion, CL Cara, D Preti, ... Mini reviews in medicinal chemistry 7 (6), 559-569, 2007 | 51 | 2007 |
Phenylpyrrole derivatives as neural and inducible nitric oxide synthase (nNOS and iNOS) inhibitors LCL Cara, ME Camacho, MD Carrión, V Tapias, MA Gallo, G Escames, ... European journal of medicinal chemistry 44 (6), 2655-2666, 2009 | 46 | 2009 |