Structure–activity study of bioisosteric trifluoromethyl and pentafluorosulfanyl indole inhibitors of the AAA ATPase p97 C Alverez, MR Arkin, SL Bulfer, R Colombo, M Kovaliov, MG LaPorte, ... ACS medicinal chemistry letters 6 (12), 1225-1230, 2015 | 58 | 2015 |
SuFEx postpolymerization modification kinetics and reactivity in polymer brushes K Durie, J Yatvin, M Kovaliov, GH Crane, J Horn, S Averick, J Locklin Macromolecules 51 (2), 297-305, 2018 | 49 | 2018 |
Synthesis of lipase polymer hybrids with retained or enhanced activity using the grafting-from strategy M Kovaliov, ML Allegrezza, B Richter, D Konkolewicz, S Averick Polymer 137, 338-345, 2018 | 47 | 2018 |
Therapeutic and prophylactic vaccines to counteract fentanyl use disorders and toxicity C Robinson, V Gradinati, F Hamid, C Baehr, B Crouse, S Averick, ... Journal of medicinal chemistry 63 (23), 14647-14667, 2020 | 28 | 2020 |
Covalent poly (lactic acid) nanoparticles for the sustained delivery of naloxone AJ Kassick, HN Allen, SS Yerneni, F Pary, M Kovaliov, C Cheng, ... ACS applied bio materials 2 (8), 3418-3428, 2019 | 25 | 2019 |
Extended-release of opioids using fentanyl-based polymeric nanoparticles for enhanced pain management M Kovaliov, S Li, E Korkmaz, D Cohen-Karni, N Tomycz, OB Ozdoganlar, ... RSC advances 7 (76), 47904-47912, 2017 | 23 | 2017 |
Grafting challenging monomers from proteins using aqueous ICAR ATRP under bio-relevant conditions D Cohen-Karni, M Kovaliov, T Ramelot, D Konkolewicz, S Graner, ... Polymer Chemistry 8 (27), 3992-3998, 2017 | 23 | 2017 |
In‐situ Chemiluminescence‐Driven Reversible Addition–Fragmentation Chain‐Transfer Photopolymerization N De Alwis Watuthanthrige, ML Allegrezza, MT Dolan, AJ Kloster, ... Angewandte Chemie International Edition 58 (34), 11826-11829, 2019 | 20 | 2019 |
Asymmetric total synthesis and biological evaluation of (+)-cycloclavine SR McCabe, P Wipf Synthesis 51 (01), 213-224, 2019 | 18 | 2019 |
Synthesis of orthogonally protected optically pure ketopiperazine, diketopiperazine, ketodiazepane, and 3-aminopyrrolidone building blocks for peptidomimetic combinatorial … G Gellerman, E Hazan, M Kovaliov, A Albeck, S Shatzmiler Tetrahedron 65 (7), 1389-1396, 2009 | 18 | 2009 |
Grafting-from lipase: utilization of a common amino acid residue as a new grafting site M Kovaliov, C Cheng, B Cheng, S Averick Polymer Chemistry 9 (37), 4651-4659, 2018 | 17 | 2018 |
Affinity capture of p97 with small-molecule ligand bait reveals a 3.6 Å double-hexamer cryoelectron microscopy structure MR Hoq, FS Vago, K Li, M Kovaliov, RJ Nicholas, DM Huryn, P Wipf, ... ACS nano 15 (5), 8376-8385, 2021 | 15 | 2021 |
Fentanyl initiated polymers prepared by atrp for targeted delivery D Cohen-Karni, M Kovaliov, S Li, S Jaffee, ND Tomycz, S Averick Bioconjugate Chemistry 28 (4), 1251-1259, 2017 | 14 | 2017 |
A threonine turnstile defines a dynamic amphiphilic binding motif in the AAA ATPase p97 allosteric binding site JC Burnett, C Lim, BD Peyser, LP Samankumara, M Kovaliov, R Colombo, ... Organic & biomolecular chemistry 15 (19), 4096-4114, 2017 | 14 | 2017 |
Toward next-generation biohybrid catalyst design: influence of degree of polymerization on enzyme activity M Kovaliov, TA Wright, B Cheng, RT Mathers, X Zhang, D Meng, ... Bioconjugate Chemistry 31 (3), 939-947, 2020 | 13 | 2020 |
Grafting strategies for the synthesis of active DNase I polymer biohybrids M Kovaliov, D Cohen-Karni, KA Burridge, D Mambelli, S Sloane, ... European Polymer Journal 107, 15-24, 2018 | 13 | 2018 |
Synthesis and evaluation of a photoresponsive quencher for fluorescent hybridization probes M Kovaliov, C Wachtel, E Yavin, B Fischer Organic & biomolecular chemistry 12 (39), 7844-7858, 2014 | 13 | 2014 |
Antimicrobial benzodiazepine‐based short cationic peptidomimetics GM Zats, M Kovaliov, A Albeck, S Shatzmiller Journal of Peptide Science 21 (6), 512-519, 2015 | 11 | 2015 |
Phenyl-imidazolo-cytidine Analogues: Structure–Photophysical Activity Relationship and Ability To Detect Single DNA Mismatch M Kovaliov, M Weitman, DT Major, B Fischer The Journal of Organic Chemistry 79 (15), 7051-7062, 2014 | 11 | 2014 |
Fluorescent p-substituted-phenyl-imidazolo-cytidine analogues M Kovaliov, M Segal, B Fischer Tetrahedron 69 (18), 3698-3705, 2013 | 11 | 2013 |