Peptidotriazoles on solid phase:[1, 2, 3]-triazoles by regiospecific copper (I)-catalyzed 1, 3-dipolar cycloadditions of terminal alkynes to azides CW Tornøe, C Christensen, M Meldal The Journal of organic chemistry 67 (9), 3057-3064, 2002 | 10580 | 2002 |
Cu-catalyzed azide− alkyne cycloaddition M Meldal, CW Tornøe Chemical reviews 108 (8), 2952-3015, 2008 | 5336 | 2008 |
Combinatorial Library of Peptidotriazoles: Identification of [1,2,3]-Triazole Inhibitors against a Recombinant Leishmania mexicana Cysteine Protease CW Tornøe, SJ Sanderson, JC Mottram, GH Coombs, M Meldal Journal of Combinatorial Chemistry 6 (3), 312-324, 2004 | 210 | 2004 |
Peptidotriazoles: Copper (I)-catalyzed 1, 3-dipolar cycloadditions on solid-phase CW Tornøe, M Meldal Peptides: The Wave of the Future: Proceedings of the Second International …, 2001 | 149 | 2001 |
Palladium‐Catalyzed Three‐Component Approach to Promazine with Formation of One Carbon–Sulfur and Two Carbon–Nitrogen Bonds T Dahl, CW Tornøe, B Bang‐Andersen, P Nielsen, M Jørgensen Angewandte Chemie International Edition 47 (9), 1726-1728, 2008 | 146 | 2008 |
α‐Azido acids for direct use in solid‐phase peptide synthesis CW Tornøe, P Davis, F Porreca, M Meldal Journal of Peptide Science: An Official Publication of the European Peptide …, 2000 | 34 | 2000 |
Efficient synthesis of diverse 5-thio-or 5-selenotriazoles: One-pot multicomponent reaction from elemental sulfur or selenium LL Zhang, YT Li, T Gao, SS Guo, B Yang, ZH Meng, QP Dai, ZB Xu, ... Synthesis 51 (22), 4170-4182, 2019 | 29 | 2019 |
Anti-Markovnikov hydroazidation of activated olefins via organic photoredox catalysis NPR Onuska, ME Schutzbach-Horton, JLR Collazo, DA Nicewicz Synlett 31 (01), 55-59, 2020 | 21 | 2020 |
One-pot, metal-and azide-free synthesis of 1, 2, 3-triazoles from α-ketoacetals and amines LR Zehnder, JM Hawkins, SC Sutton Synlett 31 (02), 175-178, 2020 | 19 | 2020 |
A mild multi-component reaction for the synthesis of 4, 5-disubstituted 1H-1, 2, 3-Triazoles from phosphonium salts, aldehydes, and sodium azide GL Wu, QP Wu Synthesis 50 (14), 2768-2774, 2018 | 19 | 2018 |
Ralph F. Hirschmann award address 2009: Merger of organic chemistry with peptide diversity M Meldal, CW Tornøe, TE Nielsen, F Diness, ST Le Quement, ... Peptide Science: Original Research on Biomolecules 94 (2), 161-182, 2010 | 19 | 2010 |
Divergent protein synthesis of Bowman–Birk protease inhibitors, their hydrodynamic behavior and co-crystallization with α-chymotrypsin CW Tornøe, E Johansson, PO Wahlund Synlett 28 (15), 1901-1906, 2017 | 15 | 2017 |
Enzymatic and chiral HPLC resolution of α-azido acids and amides CW Tornøe, T Sonke, I Maes, HE Schoemaker, M Meldal Tetrahedron: Asymmetry 11 (5), 1239-1248, 2000 | 15 | 2000 |
Substituted morpholine and thiomorpholine derivatives CW Tornøe, M Rottländer, N Khanzhin, A Ritzèn, WP Watson US Patent 7,501,414, 2009 | 14* | 2009 |
EXPO3000—a new expandable polymer for synthesis and enzymatic assays CW Tornøe, M Meldal Tetrahedron letters 43 (36), 6409-6411, 2002 | 14 | 2002 |
Solid‐phase synthesis of chemotactic peptides using α‐azido acids CW Tornøe, H Sengeløv, M Meldal Journal of peptide science: an official publication of the European Peptide …, 2000 | 14 | 2000 |
Dipolar Cycloaddition Reactions in Peptide Chemistry CW Tornøe, M Meldal Organic Azides: Syntheses and Applications, 285, 2009 | 13 | 2009 |
A multifunctional HBED-type chelator with dual conjugation capabilities for radiopharmaceutical development A Makarem, MK Sarvestani, KD Klika, K Kopka Synlett 30 (15), 1795-1798, 2019 | 12 | 2019 |
Derivatives of GLP-1 like peptides, and uses thereof S Reedtz-Runge, J Kofoed, CW Tornoee, P Sauerberg US Patent 9,498,534, 2016 | 12 | 2016 |
Substituted aniline derivatives D Greve, M Rottlander, W Watson US Patent App. 10/549,345, 2006 | 12* | 2006 |