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Nikolina MAČEK HRVAT
Nikolina MAČEK HRVAT
Scientific Associate, Institute for Medical Research and Occupational Health
在 imi.hr 的电子邮件经过验证
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引用次数
引用次数
年份
Centrally acting oximes in reactivation of tabun-phosphoramidated AChE
Z Kovarik, N Maček, RK Sit, Z Radić, VV Fokin, KB Sharpless, P Taylor
Chemico-biological interactions 203 (1), 77-80, 2013
762013
Potent 3‐Hydroxy‐2‐Pyridine Aldoxime Reactivators of Organophosphate‐Inhibited Cholinesterases with Predicted Blood–Brain Barrier Penetration
T Zorbaz, A Braïki, N Maraković, J Renou, E de La Mora, N Maček Hrvat, ...
Chemistry–A European Journal 24 (38), 9675-9691, 2018
682018
Pyridinium Oximes with Ortho-Positioned Chlorine Moiety Exhibit Improved Physicochemical Properties and Efficient Reactivation of Human Acetylcholinesterase …
T Zorbaz, D Malinak, N Maraković, N Maček Hrvat, A Zandona, ...
Journal of medicinal chemistry 61 (23), 10753-10766, 2018
612018
A comprehensive evaluation of novel oximes in creation of butyrylcholinesterase-based nerve agent bioscavengers
M Katalinić, NM Hrvat, K Baumann, SM Piperčić, S Makarić, S Tomić, ...
Toxicology and applied pharmacology 310, 195-204, 2016
522016
Catalytic soman scavenging by the Y337A/F338A acetylcholinesterase mutant assisted with novel site-directed aldoximes
Z Kovarik, N Maček Hrvat, M Katalinić, RK Sit, A Paradyse, S Žunec, ...
Chemical research in toxicology 28 (5), 1036-1044, 2015
502015
Pharmacology, pharmacokinetics, and tissue disposition of zwitterionic hydroxyiminoacetamido alkylamines as reactivating antidotes for organophosphate exposure
RK Sit, Z Kovarik, NM Hrvat, S Žunec, C Green, VV Fokin, KB Sharpless, ...
Journal of Pharmacology and Experimental Therapeutics 367 (2), 363-372, 2018
482018
Counteracting poisoning with chemical warfare nerve agents
N Maček Hrvat, Z Kovarik
Arhiv za higijenu rada i toksikologiju 71 (4), 284-284, 2020
432020
Oxime-assisted reactivation of tabun-inhibited acetylcholinesterase analysed by active site mutations
M Katalinić, G Šinko, NM Hrvat, T Zorbaz, A Bosak, Z Kovarik
Toxicology 406, 104-113, 2018
342018
Pharmacokinetic evaluation of brain penetrating morpholine-3-hydroxy-2-pyridine oxime as an antidote for nerve agent poisoning
T Zorbaz, P Mišetić, N Probst, S Žunec, A Zandona, G Mendaš, ...
ACS chemical neuroscience 11 (7), 1072-1084, 2020
332020
The estimation of oxime efficiency is affected by the experimental design of phosphylated acetylcholinesterase reactivation
NM Hrvat, T Zorbaz, G Šinko, Z Kovarik
Toxicology letters 293, 222-228, 2018
332018
Reversal of Tabun Toxicity Enabled by a Triazole‐Annulated Oxime Library—Reactivators of Acetylcholinesterase
Z Kovarik, J Kalisiak, NM Hrvat, M Katalinić, T Zorbaz, S Žunec, C Green, ...
Chemistry–A European Journal 25 (16), 4100-4114, 2019
312019
HI-6 assisted catalytic scavenging of VX by acetylcholinesterase choline binding site mutants
NM Hrvat, S Žunec, P Taylor, Z Radić, Z Kovarik
Chemico-biological interactions 259, 148-153, 2016
272016
Translation of in vitro to in vivo pyridinium oxime potential in tabun poisoning/Translacija učinkovitosti piridinijevih oksima kod trovanja tabunom iz in vitro sustava u in …
M Katalinić, NM Hrvat, JŽ Karasová, J Misik, Z Kovarik
Archives of Industrial Hygiene and Toxicology 66 (4), 291-298, 2015
252015
Evaluation of high-affinity phenyltetrahydroisoquinoline aldoximes, linked through anti-triazoles, as reactivators of phosphylated cholinesterases
NM Hrvat, J Kalisiak, G Šinko, Z Radić, KB Sharpless, P Taylor, Z Kovarik
Toxicology letters 321, 83-89, 2020
212020
Design, synthesis and cholinesterase inhibitory properties of new oxazole benzylamine derivatives
I Šagud, N Maček Hrvat, A Grgičević, T Čadež, J Hodak, M Dragojević, ...
Journal of enzyme inhibition and medicinal chemistry 35 (1), 460-467, 2020
202020
Halogen substituents enhance oxime nucleophilicity for reactivation of cholinesterases inhibited by nerve agents
T Zorbaz, D Malinak, T Hofmanova, N Maraković, S Žunec, NM Hrvat, ...
European Journal of Medicinal Chemistry 238, 114377, 2022
132022
Efficient detoxification of nerve agents by oxime-assisted reactivation of acetylcholinesterase mutants
Z Kovarik, NM Hrvat
Neuropharmacology 171, 108111, 2020
132020
Counteracting tabun inhibition by reactivation by pyridinium aldoximes that interact with active center gorge mutants of acetylcholinesterase
Z Kovarik, NM Hrvat, J Kalisiak, M Katalinić, RK Sit, T Zorbaz, Z Radić, ...
Toxicology and applied pharmacology 372, 40-46, 2019
122019
Who's in, who's out? Re‐evaluation of lipid raft residents
K Mlinac‐Jerkovic, K Ilic, M Zjalić, D Mandić, Ž Debeljak, M Balog, ...
Journal of neurochemistry 158 (3), 657-672, 2021
82021
Benzobicyclo [3.2. 1] octene derivatives as a new class of cholinesterase inhibitors
T Čadež, A Grgičević, R Ahmetović, D Barić, NM Hrvat, Z Kovarik, I Škorić
Molecules 25 (21), 4872, 2020
82020
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