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Katrin Szardenings
Katrin Szardenings
Janssen
在 its.jnj.com 的电子邮件经过验证
标题
引用次数
引用次数
年份
Early clinical PET imaging results with the novel PHF-tau radioligand [F-18]-T807
DT Chien, S Bahri, AK Szardenings, JC Walsh, F Mu, MY Su, WR Shankle, ...
Journal of Alzheimer's Disease 34 (2), 457-468, 2013
7582013
[18F] T807, a novel tau positron emission tomography imaging agent for Alzheimer's disease
CF Xia, J Arteaga, G Chen, U Gangadharmath, LF Gomez, D Kasi, C Lam, ...
Alzheimer's & Dementia 9 (6), 666-676, 2013
5462013
Functional interrogation of the kinome using nucleotide acyl phosphates
MP Patricelli, AK Szardenings, M Liyanage, TK Nomanbhoy, M Wu, ...
Biochemistry 46 (2), 350-358, 2007
4732007
Early clinical PET imaging results with the novel PHF-tau radioligand [F18]-T808
DT Chien, AK Szardenings, S Bahri, JC Walsh, F Mu, C Xia, WR Shankle, ...
Journal of Alzheimer's Disease 38 (1), 171-184, 2014
3132014
A highly selective and specific PET tracer for imaging of tau pathologies
W Zhang, J Arteaga, DK Cashion, G Chen, U Gangadharmath, LF Gomez, ...
Journal of Alzheimer's Disease 31 (3), 601-612, 2012
2342012
A simple procedure for the solid phase synthesis of diketopiperazine and diketomorpholine derivatives
AK Szardenings, TS Burkoth, HH Lu, DW Tien, DA Campbell
Tetrahedron 53 (19), 6573-6593, 1997
1781997
A reductive alkylation procedure applicable to both solution-and solid-phase syntheses of secondary amines
AK Szardenings, TS Burkoth, GC Look, DA Campbell
The Journal of organic chemistry 61 (19), 6720-6722, 1996
1421996
Identification of highly selective inhibitors of collagenase-1 from combinatorial libraries of diketopiperazines
AK Szardenings, V Antonenko, DA Campbell, N DeFrancisco, S Ida, L Shi, ...
Journal of medicinal chemistry 42 (8), 1348-1357, 1999
1071999
Functional profiling of the proteome with affinity labels
DA Campbell, AK Szardenings
Current opinion in chemical biology 7 (2), 296-303, 2003
972003
Method for synthesis of diketopiperazine and diketomorpholine derivatives
AK Szardenings, D Campbell
US Patent 5,817,751, 1998
961998
Rational design and combinatorial evaluation of enzyme inhibitor scaffolds: identification of novel inhibitors of matrix metalloproteinases
AK Szardenings, D Harris, S Lam, L Shi, D Tien, Y Wang, DV Patel, ...
Journal of medicinal chemistry 41 (13), 2194-2200, 1998
951998
Synthesis and Structure–activity Relationship of N-alkyl Gly-boro-Pro Inhibitors of DPP4, FAP, and DPP7
Y Hu, L Ma, M Wu, MS Wong, B Li, S Corral, Z Yu, T Nomanbhoy, ...
Bioorganic & Medicinal Chemistry Letters 15 (19), 4239-4242, 2005
932005
2, 5-Diketopiperazines as potent and selective oxytocin antagonists 1: Identification, stereochemistry and initial SAR
PG Wyatt, MJ Allen, AD Borthwick, DE Davies, AM Exall, RJD Hatley, ...
Bioorganic & medicinal chemistry letters 15 (10), 2579-2582, 2005
892005
α, α-Difluoro-β-ketophosphonates as potent inhibitors of protein tyrosine phosphatase 1B
X Li, A Bhandari, CP Holmes, AK Szardenings
Bioorganic & medicinal chemistry letters 14 (16), 4301-4306, 2004
812004
Chemiluminescent nitrogen detection for HPLC: an important new tool in organic analytical chemistry
WL Fitch, AK Szardenings, EM Fujinari
Tetrahedron letters 38 (10), 1689-1692, 1997
811997
Imaging agents for detecting neurological disorders
UB Gangadharmath, HC Kolb, PJH Scott, JC Walsh, W Zhang, ...
US Patent 8,491,869, 2013
752013
Repeatability of hypoxia PET imaging using [18F]HX4 in lung and head and neck cancer patients: a prospective multicenter trial
CML Zegers, W van Elmpt, K Szardenings, H Kolb, A Waxman, ...
European journal of nuclear medicine and molecular imaging 42, 1840-1849, 2015
712015
Collagenase-1 and stromelysin-1 inhibitors, pharmaceutical compositions comprising same and methods of their use
D Campbell, GC Look, AK Szardenings, DV Patel
US Patent 5,932,579, 1999
651999
Imaging agents for detecting neurological disorders
AK Szardenings, W Zhang, D Kasi, A Sinha, UB Gangadharmath, ...
US Patent 8,691,187, 2014
612014
PET Imaging of the P2X7 Ion Channel with a Novel Tracer [18F]JNJ-64413739 in a Rat Model of Neuroinflammation
T Berdyyeva, C Xia, N Taylor, Y He, G Chen, C Huang, W Zhang, H Kolb, ...
Molecular Imaging and Biology 21, 871-878, 2019
582019
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