Early clinical PET imaging results with the novel PHF-tau radioligand [F-18]-T807 DT Chien, S Bahri, AK Szardenings, JC Walsh, F Mu, MY Su, WR Shankle, ... Journal of Alzheimer's Disease 34 (2), 457-468, 2013 | 758 | 2013 |
[18F] T807, a novel tau positron emission tomography imaging agent for Alzheimer's disease CF Xia, J Arteaga, G Chen, U Gangadharmath, LF Gomez, D Kasi, C Lam, ... Alzheimer's & Dementia 9 (6), 666-676, 2013 | 546 | 2013 |
Functional interrogation of the kinome using nucleotide acyl phosphates MP Patricelli, AK Szardenings, M Liyanage, TK Nomanbhoy, M Wu, ... Biochemistry 46 (2), 350-358, 2007 | 473 | 2007 |
Early clinical PET imaging results with the novel PHF-tau radioligand [F18]-T808 DT Chien, AK Szardenings, S Bahri, JC Walsh, F Mu, C Xia, WR Shankle, ... Journal of Alzheimer's Disease 38 (1), 171-184, 2014 | 313 | 2014 |
A highly selective and specific PET tracer for imaging of tau pathologies W Zhang, J Arteaga, DK Cashion, G Chen, U Gangadharmath, LF Gomez, ... Journal of Alzheimer's Disease 31 (3), 601-612, 2012 | 234 | 2012 |
A simple procedure for the solid phase synthesis of diketopiperazine and diketomorpholine derivatives AK Szardenings, TS Burkoth, HH Lu, DW Tien, DA Campbell Tetrahedron 53 (19), 6573-6593, 1997 | 178 | 1997 |
A reductive alkylation procedure applicable to both solution-and solid-phase syntheses of secondary amines AK Szardenings, TS Burkoth, GC Look, DA Campbell The Journal of organic chemistry 61 (19), 6720-6722, 1996 | 142 | 1996 |
Identification of highly selective inhibitors of collagenase-1 from combinatorial libraries of diketopiperazines AK Szardenings, V Antonenko, DA Campbell, N DeFrancisco, S Ida, L Shi, ... Journal of medicinal chemistry 42 (8), 1348-1357, 1999 | 107 | 1999 |
Functional profiling of the proteome with affinity labels DA Campbell, AK Szardenings Current opinion in chemical biology 7 (2), 296-303, 2003 | 97 | 2003 |
Method for synthesis of diketopiperazine and diketomorpholine derivatives AK Szardenings, D Campbell US Patent 5,817,751, 1998 | 96 | 1998 |
Rational design and combinatorial evaluation of enzyme inhibitor scaffolds: identification of novel inhibitors of matrix metalloproteinases AK Szardenings, D Harris, S Lam, L Shi, D Tien, Y Wang, DV Patel, ... Journal of medicinal chemistry 41 (13), 2194-2200, 1998 | 95 | 1998 |
Synthesis and Structure–activity Relationship of N-alkyl Gly-boro-Pro Inhibitors of DPP4, FAP, and DPP7 Y Hu, L Ma, M Wu, MS Wong, B Li, S Corral, Z Yu, T Nomanbhoy, ... Bioorganic & Medicinal Chemistry Letters 15 (19), 4239-4242, 2005 | 93 | 2005 |
2, 5-Diketopiperazines as potent and selective oxytocin antagonists 1: Identification, stereochemistry and initial SAR PG Wyatt, MJ Allen, AD Borthwick, DE Davies, AM Exall, RJD Hatley, ... Bioorganic & medicinal chemistry letters 15 (10), 2579-2582, 2005 | 89 | 2005 |
α, α-Difluoro-β-ketophosphonates as potent inhibitors of protein tyrosine phosphatase 1B X Li, A Bhandari, CP Holmes, AK Szardenings Bioorganic & medicinal chemistry letters 14 (16), 4301-4306, 2004 | 81 | 2004 |
Chemiluminescent nitrogen detection for HPLC: an important new tool in organic analytical chemistry WL Fitch, AK Szardenings, EM Fujinari Tetrahedron letters 38 (10), 1689-1692, 1997 | 81 | 1997 |
Imaging agents for detecting neurological disorders UB Gangadharmath, HC Kolb, PJH Scott, JC Walsh, W Zhang, ... US Patent 8,491,869, 2013 | 75 | 2013 |
Repeatability of hypoxia PET imaging using [18F]HX4 in lung and head and neck cancer patients: a prospective multicenter trial CML Zegers, W van Elmpt, K Szardenings, H Kolb, A Waxman, ... European journal of nuclear medicine and molecular imaging 42, 1840-1849, 2015 | 71 | 2015 |
Collagenase-1 and stromelysin-1 inhibitors, pharmaceutical compositions comprising same and methods of their use D Campbell, GC Look, AK Szardenings, DV Patel US Patent 5,932,579, 1999 | 65 | 1999 |
Imaging agents for detecting neurological disorders AK Szardenings, W Zhang, D Kasi, A Sinha, UB Gangadharmath, ... US Patent 8,691,187, 2014 | 61 | 2014 |
PET Imaging of the P2X7 Ion Channel with a Novel Tracer [18F]JNJ-64413739 in a Rat Model of Neuroinflammation T Berdyyeva, C Xia, N Taylor, Y He, G Chen, C Huang, W Zhang, H Kolb, ... Molecular Imaging and Biology 21, 871-878, 2019 | 58 | 2019 |