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Khuloud takrouri
Khuloud takrouri
Medicinal Chemist, PhD
在 mail.huji.ac.il 的电子邮件经过验证
标题
引用次数
引用次数
年份
Structure of the eukaryotic translation initiation factor eIF4E in complex with 4EGI-1 reveals an allosteric mechanism for dissociating eIF4G
E Papadopoulos, S Jenni, E Kabha, KJ Takrouri, T Yi, N Salvi, RE Luna, ...
Proceedings of the National Academy of Sciences 111 (31), E3187-E3195, 2014
962014
New reduction pathways for ctc-[PtCl 2 (CH 3 CO 2) 2 (NH 3)(Am)] anticancer prodrugs
A Nemirovski, I Vinograd, K Takrouri, A Mijovilovich, A Rompel, D Gibson
Chemical Communications 46 (11), 1842-1844, 2010
892010
Progress against Escherichia coli with the Oxazolidinone Class of Antibacterials: Test Case for a General Approach To Improving Whole-Cell Gram-Negative Activity
K Takrouri, HD Cooper, A Spaulding, P Zucchi, B Koleva, DC Cleary, ...
ACS Infectious Diseases 2 (6), 405-426, 2016
342016
Explorations of substituted urea functionality for the discovery of new activators of the heme-regulated inhibitor kinase
T Chen, K Takrouri, S Hee-Hwang, S Rana, R Yefidoff-Freedman, ...
Journal of medicinal chemistry 56 (23), 9457-9470, 2013
312013
Structure–activity relationship study of 4EGI-1, small molecule eIF4E/eIF4G protein–protein interaction inhibitors
K Takrouri, T Chen, E Papadopoulos, R Sahoo, E Kabha, H Chen, ...
European journal of medicinal chemistry 77, 361-377, 2014
302014
Synthesis of rigidified eIF4E/eIF4G inhibitor-1 (4EGI-1) mimetic and their in vitro characterization as inhibitors of protein–protein interaction
P Mahalingam, K Takrouri, T Chen, R Sahoo, E Papadopoulos, L Chen, ...
Journal of medicinal chemistry 57 (12), 5094-5111, 2014
292014
Pharmacologically active boranes
A Jabbour, R Smoum, K Takrouri, E Shalom, B Zaks, D Steinberg, ...
Pure and applied chemistry 78 (7), 1425-1453, 2006
272006
Synthesis and antifungal activity of a novel series of alkyldimethylamine cyanoboranes and their derivatives
K Takrouri, G Oren, I Polacheck, E Sionov, E Shalom, J Katzhendler, ...
Journal of medicinal chemistry 49 (16), 4879-4885, 2006
252006
C-Lithiation/alkylation of trimethylamine cyanoborane
K Takrouri, J Katzhendler, M Srebnik
Organometallics 23 (11), 2817-2820, 2004
232004
Effect of surfactants on the thermodynamic properties of Methyl Orange dye in buffered solutions
M Dakiky, M Khamis, A Manasra, K Takrouri
Coloration technology 118 (4), 191-197, 2002
172002
Compound design guidelines for evading the efflux and permeation barriers of Escherichia coli with the oxazolidinone class of antibacterials: Test case for a general approach …
A Spaulding, K Takrouri, P Mahalingam, DC Cleary, HD Cooper, P Zucchi, ...
Bioorganic & Medicinal Chemistry Letters 27 (23), 5310-5321, 2017
152017
Preparation and Structure Determination of Trimethylamine− Dibromocarboxyborane Esters
E Shalom, K Takrouri, I Goldberg, J Katzhendler, M Srebnik
Organometallics 23 (19), 4396-4399, 2004
152004
Diborane (4) derivatives via coupling of amine monobromocyanoboranes: Study of the bromination of amine cyanoborane and molecular structures of the amine dibromocyanoboranes
K Takrouri, E Shalom, I Goldberg, J Katzhendler, M Srebnik
Journal of organometallic chemistry 690 (18), 4150-4158, 2005
102005
Insight into acid driven formation of spiro-[oxindole] xanthenes from isatin and phenols
H Yang, K Takrouri, M Chorev
Current Organic Chemistry 16 (13), 1581-1593, 2012
92012
Semiautomated synthesis of a novel [18F] amine fluorocyanoborane for PET imaging studies. Radiosynthesis and in vivo characterization in rats
E Shalom, K Takrouri, N Metsuyanim, A Grufi, J Katzhendler, M Srebnik
Applied radiation and isotopes 65 (2), 204-208, 2007
62007
Preparation of novel fluoro derivatives of amine cyanoboranes and amine carboxyborane esters
E Shalom, K Takrouri, I Goldberg, J Katzhendler, M Srebnik
Organometallics 24 (23), 5776-5779, 2005
42005
α-Aminoboronic acids, amine cyanoboranes, amine carboxyboranes and their derivatives
K Takrouri, VM Dembistky, M Srebnik
Studies in Inorganic Chemistry 22, 495-549, 2005
42005
Novel amine-borane compounds and uses thereof
M Srebnik, K Takrouri, E Shalom
US Patent App. 11/991,850, 2010
32010
Crystallographic report: Dimethyl‐2‐phenylethan‐2‐olamine cyanoborane
K Takrouri, E Shalom, I Goldberg, J Katzhendler, M Srebnik
Applied organometallic chemistry 19 (3), 386-387, 2005
32005
Crystallographic report: Trimethylaminedibromopropoxycarbonylborane
E Shalom, K Takrouri, I Goldberg, J Katzhendler, M Srebnik
Applied organometallic chemistry 19 (3), 391-392, 2005
32005
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