Validation and development of MTH1 inhibitors for treatment of cancer UW Berglund, K Sanjiv, H Gad, C Kalderen, T Koolmeister, T Pham, ... Annals of oncology 27 (12), 2275-2283, 2016 | 141 | 2016 |
Base-Mediated Hydroamination of Propargylamine: A Regioselective Intramolecular 5-exo-dig Cycloisomerization en Route to Imidazole-2-thione A Ranjan, R Yerande, PB Wakchaure, SG Yerande, DH Dethe Organic letters 16 (21), 5788-5791, 2014 | 76 | 2014 |
Facile air-oxidation of N-homopiperonyl-5, 6-dimethoxyhomophthalimide: simple and efficient access to nuevamine PB Wakchaure, S Easwar, VG Puranik, NP Argade Tetrahedron 64 (8), 1786-1791, 2008 | 43 | 2008 |
Thermal and Microwave‐Assisted Conjugate Additions of Indole on Electron‐Deficient Nitro‐olefins RS Kusurkar, NAH Alkobati, AS Gokule, PM Chaudhari, PB Waghchaure Synthetic communications 36 (8), 1075-1081, 2006 | 28 | 2006 |
Synthesis of Vinyl‐ and Aryl–Acyl Sulfonimidamides Through Pd‐Catalyzed Carbonylation Using Mo(CO)6 as ex situ CO Source PB Wakchaure, SR Borhade, A Sandström, PI Arvidsson European Journal of Organic Chemistry 2015 (1), 213-219, 2015 | 26 | 2015 |
MTH1 promotes mitotic progression to avoid oxidative DNA damage in cancer cells H Gad, O Mortusewicz, SG Rudd, A Stolz, N Amaral, L Brautigham, ... BioRxiv, 575290, 2019 | 21 | 2019 |
Synthesis of the reported protoberberine gusanlung D PB Wakchaure, S Easwar, NP Argade Synthesis 2009 (10), 1667-1672, 2009 | 18 | 2009 |
Pd-catalyzed C–N coupling of vinylbromides and sulfonimidamides: a facile synthesis of N′-vinylsulfonimidamides GC Nandi, SR Kota, PB Wakchaure, PK Chinthakindi, T Govender, ... RSC advances 5 (76), 62084-62090, 2015 | 13 | 2015 |
Intramolecular chemoselective acylation of a suitably substituted isoindole: synthesis of (±)-chilenine and (±)-deoxychilenine PB Wakchaure, NP Argade Synthesis 2011 (17), 2838-2842, 2011 | 13 | 2011 |
NUDT15-mediated hydrolysis limits the efficacy of anti-HCMV drug ganciclovir SM Zhang, D Rehling, AS Jemth, A Throup, N Landázuri, I Almlöf, ... Cell chemical biology 28 (12), 1693-1702. e6, 2021 | 12 | 2021 |
Synthesis of enantiopure angiotensin II type 2 receptor [AT2R] antagonist EMA401 PB Wakchaure, U Bremberg, J Wannberg, M Larhed Tetrahedron 71 (38), 6881-6887, 2015 | 11 | 2015 |
Stereoselective synthesis of (+)-isoindolo-β-carboline PB Wakchaure, VG Puranik, NP Argade Tetrahedron: Asymmetry 20 (2), 220-224, 2009 | 10 | 2009 |
Activation of Primary Amines by Copper (I)-Based Lewis Acid Promoters in the Solventless Synthesis of Secondary Propargylamines C Cimarelli, F Navazio, FV Rossi, F Del Bello, E Marcantoni Synthesis 51 (11), 2387-2396, 2019 | 7 | 2019 |
Easwar. S.; Puranik. VG; Argade, NP PB Wakchaure Tetrahedron 64, 1786, 2008 | 7 | 2008 |
Palladium‐Catalyzed Carbonylation of Aryl Iodides with Sulfinamides AK Belfrage, P Wakchaure, M Larhed, A Sandström European Journal of Organic Chemistry 2015 (32), 7069-7074, 2015 | 6 | 2015 |
A facile biogenetic synthesis of pulcheotine A PB Wakchaure, NP Argade Synthesis 2008 (15), 2321-2322, 2008 | 6 | 2008 |
Fries rearrangement: scalable synthesis of key fluoro building blocks 3-fluoro-4-methoxybenzoyl chloride and 1, 2-diethoxy-3-fluorobenzene SG Yerande, DM Shendage, PB Wakchaure, GR Phadtare, MY Bhoite, ... Tetrahedron Letters 55 (15), 2426-2429, 2014 | 5 | 2014 |
Regioselective NaBH4 and DIBAL-H reductions of 3,4-dimethoxyhomopiperonylphthalimide: Concise and efficient synthesis of nuevamine and isonuevamine PB Wakchaure, SS Kunte, NP Argade NISCAIR-CSIR, India, 2011 | 5 | 2011 |
Coupling cellular drug-target engagement to downstream pharmacology with CeTEAM NCK Valerie, K Sanjiv, O Mortusewicz, SM Zhang, S Alam, MJ Pires, ... bioRxiv, 2022.09. 19.505646, 2022 | | 2022 |
Mechanistic Investigation of Palladium (II)-Catalyzed Decarboxylative Synthesis of Electron Rich Styrenes and 1, 1-Diarylethenes F Svensson, A Fardost, B Skillinghaug, P Wakchaure, M Wejdemar, ... | | 2015 |