Quinazoline‐4‐piperidine sulfamides are specific inhibitors of human NPP 1 and prevent pathological mineralization of valve interstitial cells EE Shayhidin, E Forcellini, MC Boulanger, A Mahmut, S Dautrey, ... British journal of pharmacology 172 (16), 4189-4199, 2015 | 40 | 2015 |
Synthesis and biological evaluation of novel quinazoline-4-piperidinesulfamide derivatives as inhibitors of NPP1 E Forcellini, S Boutin, CA Lefebvre, EE Shayhidin, MC Boulanger, ... European Journal of Medicinal Chemistry 147, 130-149, 2018 | 28 | 2018 |
Synthesis of novel substituted pyrimidine derivatives bearing a sulfamide group and their in vitro cancer growth inhibition activity CA Lefebvre, E Forcellini, S Boutin, MF Côté, C René, P Mathieu, P Lagüe, ... Bioorganic & Medicinal Chemistry Letters 27 (2), 299-302, 2017 | 25 | 2017 |
Synthesis and pharmacological evaluation of a new series of radiolabeled ligands for 5-HT7 receptor PET neuroimaging J Colomb, G Becker, E Forcellini, S Meyer, L Buisson, L Zimmer, T Billard Nuclear Medicine and Biology 41 (4), 330-337, 2014 | 21 | 2014 |
Systematic study of the reactivity of (E)-4, 4, 4-trifluorobut-2-en-1-yl 4-methylbenzenesulfonate towards different classes of nucleophiles E Forcellini, R Hemelaere, J Desroches, JF Paquin Journal of Fluorine Chemistry 180, 216-221, 2015 | 8 | 2015 |
RC-Gaudreault, P. Mathieu, P. Lagüe, JF Paquin CA Lefebvre, E Forcellini, S Boutin, MF Côté Bioorg. Med. Chem. Lett 27, 299-302, 2017 | 7 | 2017 |
Complementary Methods for the Introduction of the (E)‐3‐(Pentafluorosulfanyl)allyl Chain unto O‐, N‐, S‐, and C‐Based Nucleophiles J Desroches, E Forcellini, JF Paquin European Journal of Organic Chemistry 2016 (27), 4611-4620, 2016 | 4 | 2016 |
Synthesis and in vitro activity of ectonucleotide pyrophosphatase/phosphodiesterase 1 inhibitors E Forcellini, EE Shayhidin, MC Boulanger, A Mahmut, CA Lefevbre, ... ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 251, 2016 | | 2016 |
Conception, synthèse et évaluation de l'activité biologique d'inhibiteurs d'une ectonucléotide pyrophosphatase/phosphodiestérase de type 1 (NPP1) E Forcellini | | 2016 |
A Novel Class of Inhibitors That Are Specific to Human NPP1 Prevent Pathologic Mineralization of Valve Interstitial Cells EE Shayhidin, E Forcellini, MC Boulanger, M Ablajan, S Dautrey, ... Circulation 130 (suppl_2), A16349-A16349, 2014 | | 2014 |
QUINAZOLIN-4-PIPERIDIN-4-METHYL SULFAMIDE COMPOUNDS ARE SPECIFIC INHIBITORS OF HUMAN NPP1 AND PREVENT CALCIFICATION OF VALVE INTERSTITIAL CELLS EE Shayhidin, E Forcellini, M Boulanger, A Mahmut, S Dautrey, ... Canadian Journal of Cardiology 10 (30), S245-S246, 2014 | | 2014 |