A catalytic asymmetric chlorocyclization of unsaturated amides A Jaganathan, A Garzan, DC Whitehead, RJ Staples, B Borhan Angewandte Chemie International Edition 50 (11), 2593-2596, 2011 | 206 | 2011 |
Solvent‐Dependent Enantiodivergence in the Chlorocyclization of Unsaturated Carbamates A Garzan, A Jaganathan, N Salehi Marzijarani, R Yousefi, DC Whitehead, ... Chemistry–A European Journal 19 (27), 9015-9021, 2013 | 84 | 2013 |
Pronounced catalytic effect of micellar solution of sodium dodecyl sulfate (SDS) for regioselective iodination of aromatic compounds with a sodium iodide/cerium (IV … H Firouzabadi, N Iranpoor, A Garzan Advanced Synthesis & Catalysis 347 (15), 1925-1928, 2005 | 74 | 2005 |
Structural basis for backbone N-methylation by an interrupted adenylation domain S Mori, AH Pang, TA Lundy, A Garzan, OV Tsodikov, ... Nature chemical biology, 1, 2018 | 71 | 2018 |
Novel alkylated azoles as potent antifungals SK Shrestha, A Garzan, S Garneau-Tsodikova European Journal of Medicinal Chemistry, 2017 | 64 | 2017 |
Repurposing antipsychotic drugs into antifungal agents: Synergistic combinations of azoles and bromperidol derivatives in the treatment of various fungal infections SYL Holbrook, A Garzan, EK Dennis, SK Shrestha, S Garneau-Tsodikova European Journal of Medicinal Chemistry, 2017 | 49 | 2017 |
Highly efficient halogenation of organic compounds with halides catalyzed by cerium (III) chloride heptahydrate using hydrogen peroxide as the terminal oxidant in water H Firouzabadi, N Iranpoor, S Kazemi, A Ghaderi, A Garzan Advanced Synthesis & Catalysis 351 (11‐12), 1925-1932, 2009 | 47 | 2009 |
Combating Enhanced Intracellular Survival (Eis)-Mediated Kanamycin Resistance of Mycobacterium tuberculosis by Novel Pyrrolo[1,5-a]pyrazine-Based Eis … A Garzan, MJ Willby, HX Ngo, CS Gajadeera, KD Green, SYL Holbrook, ... ACS Infectious Diseases, 2017 | 46 | 2017 |
Sulfonamide-Based Inhibitors of Aminoglycoside Acetyltransferase Eis Abolish Resistance to Kanamycin in Mycobacterium tuberculosis A Garzan, MJ Willby, KD Green, CS Gajadeera, C Hou, OV Tsodikov, ... Journal of Medicinal Chemistry 59 (23), 10619-10628, 2016 | 40 | 2016 |
Optimization of pyrazole-containing 1,2,4-triazolo-[3,4-b]thiadiazines, a new class of STAT3 pathway inhibitors MG LaPorte, Z Wang, R Colombo, A Garzan, VA Peshkov, M Liang, ... Bioorganic & Medicinal Chemistry Letters 26 (15), 3581-3585, 2016 | 32 | 2016 |
Discovery and Optimization of Two Eis Inhibitor Families as Kanamycin Adjuvants against Drug-Resistant M. tuberculosis A Garzan, MJ Willby, KD Green, OV Tsodikov, JE Posey, ... ACS Medicinal Chemistry Letters, 2016 | 31 | 2016 |
Pyrimidone inhibitors targeting Chikungunya Virus nsP3 macrodomain by fragment-based drug design S Zhang, A Garzan, N Haese, R Bostwick, Y Martinez-Gzegozewska, ... PLOS ONE 16 (1), e0245013, 2021 | 28 | 2021 |
Potent 1,2,4-Triazino[5,6b]indole-3-thioether Inhibitors of the Kanamycin Resistance Enzyme Eis from Mycobacterium tuberculosis HX Ngo, KD Green, CS Gajadeera, MJ Willby, SYL Holbrook, C Hou, ... ACS infectious diseases, 2018 | 24 | 2018 |
Deciphering Nature’s Intricate Way of N,S-Dimethylating l-Cysteine: Sequential Action of Two Bifunctional Adenylation Domains S Mori, A Garzan, OV Tsodikov, S Garneau-Tsodikova Biochemistry, 2017 | 24 | 2017 |
Discovery of Allosteric and Selective Inhibitors of Inorganic Pyrophosphatase from Mycobacterium tuberculosis AH Pang, A Garzan, MJ Larsen, TJ McQuade, S Garneau-Tsodikova, ... ACS Chemical Biology 11 (11), 3084-3092, 2016 | 21 | 2016 |
Facile Ring‐Expansion Substitution Reactions of 1, 3‐Dithiolanes and 1, 3‐Dithianes Initiated by Electrophilic Reagents to Produce Monohalo‐,‐cyano‐,‐azido‐and‐thiocyanato‐1, 4 … H Firouzabadi, N Iranpoor, A Garzan, HR Shaterian, F Ebrahimzadeh European journal of organic chemistry 2005 (2), 416-428, 2005 | 17 | 2005 |
Enzymatic Evidence for a Revised Congocidine Biosynthetic Pathway AH Al‐Mestarihi, A Garzan, JM Kim, S Garneau‐Tsodikova ChemBioChem 16 (9), 1307-1313, 2015 | 16 | 2015 |
Interfering with DNA decondensation as a strategy against Mycobacteria. E Scutigliani, E Scholl, A Grootemaat, S Khanal, J Kochan, P Krawczyk, ... Frontiers in microbiology 9, 2034, 2018 | 13 | 2018 |
Structure-based design of haloperidol analogues as inhibitors of acetyltransferase Eis from Mycobacterium tuberculosis to overcome kanamycin resistance A Punetha, KD Green, A Garzan, NT Chandrika, MJ Willby, AH Pang, ... RSC Medicinal Chemistry, 2021 | 12 | 2021 |
Activation and loading of the starter unit during thiocoraline biosynthesis S Mori, SK Shrestha, J Fernández, M Álvarez San Millán, A Garzan, ... Biochemistry, 2017 | 11 | 2017 |