The first one-pot ambient-temperature synthesis of 1, 2, 4-oxadiazoles from amidoximes and carboxylic acid esters S Baykov, T Sharonova, A Shetnev, S Rozhkov, S Kalinin, AV Smirnov Tetrahedron 73 (7), 945-951, 2017 | 93 | 2017 |
Continued exploration of 1, 2, 4-oxadiazole periphery for carbonic anhydrase-targeting primary arene sulfonamides: Discovery of subnanomolar inhibitors of membrane-bound hCA IX … M Krasavin, A Shetnev, T Sharonova, S Baykov, S Kalinin, A Nocentini, ... European Journal of Medicinal Chemistry 164, 92-105, 2019 | 82 | 2019 |
A convenient and mild method for 1, 2, 4-oxadiazole preparation: cyclodehydration of O-acylamidoximes in the superbase system MOH/DMSO S Baykov, T Sharonova, A Osipyan, S Rozhkov, A Shetnev, A Smirnov Tetrahedron Letters 57 (26), 2898-2900, 2016 | 69 | 2016 |
Heterocyclic periphery in the design of carbonic anhydrase inhibitors: 1, 2, 4-Oxadiazol-5-yl benzenesulfonamides as potent and selective inhibitors of cytosolic hCA II and … M Krasavin, A Shetnev, T Sharonova, S Baykov, T Tuccinardi, S Kalinin, ... Bioorganic Chemistry 76, 88-97, 2018 | 63 | 2018 |
Room-temperature synthesis of pharmaceutically important carboxylic acids bearing the 1, 2, 4-oxadiazole moiety M Tarasenko, N Duderin, T Sharonova, S Baykov, A Shetnev, AV Smirnov Tetrahedron Letters 58 (37), 3672-3677, 2017 | 56 | 2017 |
1, 2, 4-oxadiazole/2-imidazoline hybrids: multi-target-directed compounds for the treatment of infectious diseases and cancer A Shetnev, S Baykov, S Kalinin, A Belova, V Sharoyko, A Rozhkov, ... International Journal of Molecular Sciences 20 (7), 1699, 2019 | 53 | 2019 |
Novel monoamine oxidase inhibitors based on the privileged 2-imidazoline molecular framework A Shetnev, A Osipyan, S Baykov, A Sapegin, Z Chirkova, M Korsakov, ... Bioorganic & Medicinal Chemistry Letters 29 (1), 40-46, 2019 | 51 | 2019 |
Facile room-temperature assembly of the 1, 2, 4-oxadiazole core from readily available amidoximes and carboxylic acids T Sharonova, V Pankrat'eva, P Savko, S Baykov, A Shetnev Tetrahedron Letters 59 (29), 2824-2827, 2018 | 48 | 2018 |
Recent advances of 1, 3, 5-triazinanes in aminomethylation and cycloaddition reactions D Liang, WJ Xiao, JR Chen Synthesis 52 (17), 2469-2482, 2020 | 47 | 2020 |
An efficient synthesis and antimicrobial evaluation of 5-alkenyl-and 5-styryl-1, 2, 4-oxadiazoles M Tarasenko, V Sidneva, A Belova, A Romanycheva, T Sharonova, ... Arkivoc 7, 458-470, 2018 | 35 | 2018 |
Copper‐Catalyzed Selective N‐Arylation of Oxadiazolones by Diaryliodonium Salts NS Soldatova, AV Semenov, KK Geyl, SV Baykov, AA Shetnev, ... Advanced Synthesis & Catalysis 363 (14), 3566-3576, 2021 | 33 | 2021 |
Pyridazinone-substituted benzenesulfonamides display potent inhibition of membrane-bound human carbonic anhydrase IX and promising antiproliferative activity against cancer … M Krasavin, A Shetnev, S Baykov, S Kalinin, A Nocentini, V Sharoyko, ... European Journal of Medicinal Chemistry 168, 301-314, 2019 | 30 | 2019 |
1, 3, 4-Oxadiazol-2-ylbenzenesulfonamides as privileged structures for the inhibition of monoamine oxidase B A Shetnev, R Shlenev, J Efimova, S Ivanovskii, A Tarasov, A Petzer, ... Bioorganic & medicinal chemistry letters 29 (21), 126677, 2019 | 27 | 2019 |
The latest advances in chemistry of 1, 2, 4-oxadiazines (microreview) AA Shetnev, FI Zubkov Chemistry of Heterocyclic Compounds 53, 495-497, 2017 | 24 | 2017 |
Entry into (E)-3-(1, 2, 4-oxadiazol-5-yl) acrylic acids via a one-pot ring-opening/ring-closing/retro-Diels-Alder reaction sequence S Presnukhina, M Tarasenko, S Baykov, SN Smirnov, VP Boyarskiy, ... Tetrahedron Letters 61 (9), 151543, 2020 | 18 | 2020 |
A Condensation of Biginelli Products with 1,3‐Benzenediols: a Facile Access to Diastereomerically Pure Hexahydro‐5H‐chromeno[4,3‐d]pyrimidin‐5‐ones SI Filimonov, ZV Chirkova, MV Kabanova, ES Makarova, AA Shetnev, ... ChemistrySelect 4 (33), 9550-9555, 2019 | 16 | 2019 |
Diastereoselective Opening of Bridged Anhydrides by Amidoximes Providing Access to 1, 2, 4‐Oxadiazole/Norborna (e) ne Hybrids S Baykov, M Tarasenko, LE Zelenkov, S Kasatkina, P Savko, A Shetnev European Journal of Organic Chemistry 2019 (33), 5685-5693, 2019 | 15 | 2019 |
Synthesis of substituted 5-hydroxypyrazolo [1, 5-a] quinoxalin-4-ones VA Panova, MK Korsakov, AA Shetnev, SI Filimonov Mendeleev Communications 29 (1), 114-115, 2019 | 13 | 2019 |
2, 5-Dibromothiophenes: Halogen bond involving packing patterns and their relevance to solid-state polymerization SV Baykov, SI Presnukhina, AS Novikov, AA Shetnev, VP Boyarskiy, ... Crystal Growth & Design 21 (4), 2526-2540, 2021 | 12 | 2021 |
Investigation of pyrazolo [1, 5-a] quinoxalin-4-ones as novel monoamine oxidase inhibitors VA Panova, SI Filimonov, ZV Chirkova, MV Kabanova, AA Shetnev, ... Bioorganic Chemistry 108, 104563, 2021 | 12 | 2021 |