SF2312 is a natural phosphonate inhibitor of enolase PG Leonard, N Satani, D Maxwell, YH Lin, N Hammoudi, Z Peng, ... Nature chemical biology 12 (12), 1053-1058, 2016 | 89 | 2016 |
New synthesis of β-lactams by ethylene extrusion from spirocyclopropane isoxazolidines FM Cordero, F Pisaneschi, A Goti, J Ollivier, J Salaün, A Brandi Journal of the American Chemical Society 122 (33), 8075-8076, 2000 | 75 | 2000 |
Development of a new epidermal growth factor receptor positron emission tomography imaging agent based on the 3-cyanoquinoline core: synthesis and biological evaluation F Pisaneschi, QD Nguyen, E Shamsaei, M Glaser, E Robins, M Kaliszczak, ... Bioorganic & medicinal chemistry 18 (18), 6634-6645, 2010 | 63 | 2010 |
A novel mitochondrial inhibitor blocks MAPK pathway and overcomes MAPK inhibitor resistance in melanoma YN Vashisht Gopal, S Gammon, R Prasad, B Knighton, F Pisaneschi, ... Clinical Cancer Research 25 (21), 6429-6442, 2019 | 59 | 2019 |
An enolase inhibitor for the targeted treatment of ENO1-deleted cancers YH Lin, N Satani, N Hammoudi, VC Yan, Y Barekatain, S Khadka, ... Nature metabolism 2 (12), 1413-1426, 2020 | 50 | 2020 |
Selective ring contraction of 5-spirocyclopropane isoxazolidines mediated by acids FM Cordero, F Pisaneschi, M Salvati, V Paschetta, J Ollivier, J Salaün, ... The Journal of Organic Chemistry 68 (8), 3271-3280, 2003 | 48 | 2003 |
A new bicyclic dipeptide isostere with pyrrolizidinone skeleton FM Cordero, F Pisaneschi, K Meschini Batista, S Valenza, F Machetti, ... The Journal of Organic Chemistry 70 (3), 856-867, 2005 | 42 | 2005 |
Diastereoselective cycloaddition of alkylidenecyclopropane nitrones from palladium (0)-catalyzed nucleophilic substitution of asymmetric 1-alkenylcyclopropyl esters by amino acids F Pisaneschi, FM Cordero, A Goti, R Paugam, J Ollivier, A Brandi, ... Tetrahedron: Asymmetry 11 (4), 897-909, 2000 | 35 | 2000 |
Positron emission tomographic imaging of CXCR4 in cancer: challenges and promises GPC George, F Pisaneschi, QD Nguyen, EO Aboagye Molecular imaging 14 (1), 7290.2014. 00041, 2015 | 33 | 2015 |
Preclinical evaluation of a CXCR4-specific 68Ga-labelled TN14003 derivative for cancer PET imaging GPC George, E Stevens, O Åberg, QD Nguyen, F Pisaneschi, AC Spivey, ... Bioorganic & Medicinal Chemistry 22 (2), 796-803, 2014 | 33 | 2014 |
New developments in the synthesis of pyrrolizidinone-based dipeptide isosteres M Salvati, FM Cordero, F Pisaneschi, F Bucelli, A Brandi Tetrahedron 61 (37), 8836-8847, 2005 | 30 | 2005 |
Solid-phase access to polyhydroxypyrrolizidines by 1,3-dipolar cycloaddition of (S)-3-alkoxypyrroline N-oxide to maleate and crotonate derivatives F Pisaneschi, C Della Monica, FM Cordero, A Brandi Tetrahedron letters 43 (33), 5711-5714, 2002 | 30 | 2002 |
Novel Prospects of the Acidic Thermal Rearrangement of Spiro [cyclopropane‐1, 5′‐isoxazolidines] to β‐Lactams FM Cordero, M Salvati, F Pisaneschi, A Brandi European Journal of Organic Chemistry 2004 (10), 2205-2213, 2004 | 29 | 2004 |
Preclinical evaluation of 3-18F-fluoro-2, 2-dimethylpropionic acid as an imaging agent for tumor detection TH Witney, F Pisaneschi, IS Alam, S Trousil, M Kaliszczak, F Twyman, ... Journal of Nuclear Medicine 55 (9), 1506-1512, 2014 | 28 | 2014 |
Mechanism-Specific Pharmacodynamics of a Novel Complex-I Inhibitor Quantified by Imaging Reversal of Consumptive Hypoxia with [18F]FAZA PET In Vivo ST Gammon, F Pisaneschi, ML Bandi, MG Smith, Y Sun, Y Rao, F Muller, ... Cells 8 (12), 1487, 2019 | 26 | 2019 |
Multiwalled carbon nanotubes for combination therapy: A biodistribution and efficacy pilot study G Biagiotti, F Pisaneschi, ST Gammon, F Machetti, MC Ligi, ... Journal of Materials Chemistry B 7 (16), 2678-2687, 2019 | 25 | 2019 |
18F-labelling of a cyclic pentapeptide inhibitor of the chemokine receptor CXCR4 O Åberg, F Pisaneschi, G Smith, QD Nguyen, E Stevens, EO Aboagye Journal of Fluorine Chemistry 135, 200-206, 2012 | 24 | 2012 |
Caspase-3 substrates for noninvasive pharmacodynamic imaging of apoptosis by PET/CT BJ Engel, ST Gammon, R Chaudhari, Z Lu, F Pisaneschi, H Yang, ... Bioconjugate chemistry 29 (9), 3180-3195, 2018 | 20 | 2018 |
Combined therapies with nanostructured carbon materials: there is room still available at the bottom G Biagiotti, S Fedeli, G Tuci, L Luconi, G Giambastiani, A Brandi, ... Journal of Materials Chemistry B 6 (14), 2022-2035, 2018 | 19 | 2018 |
Stereoselective synthesis of a new trihydroxyindolizidine lactone F Pisaneschi, M Piacenti, FM Cordero, A Brandi Tetrahedron: Asymmetry 17 (2), 292-296, 2006 | 19 | 2006 |