关注
Krisztina Takács-Novák
Krisztina Takács-Novák
Professor of Department of Pharmaceutical Chemistry, Semmelweis University
在 pharma.semmelweis-univ.hu 的电子邮件经过验证
标题
引用次数
引用次数
年份
Study of equilibrium solubility measurement by saturation shake-flask method using hydrochlorothiazide as model compound
E Baka, JEA Comer, K Takács-Novák
Journal of pharmaceutical and biomedical analysis 46 (2), 335-341, 2008
5242008
Protonation equilibria of quinolone antibacterials
K Takács-Novák, B Noszál, I Hermecz, G Keresztúri, B Podányi, G Szasz
Journal of pharmaceutical sciences 79 (11), 1023-1028, 1990
2711990
Multi-wavelength spectrophotometric determination of acid dissociation constants: a validation study
KY Tam, K Takács-Novák
Analytica chimica acta 434 (1), 157-167, 2001
2242001
Skin–PAMPA: A new method for fast prediction of skin penetration
B Sinkó, TM Garrigues, GT Balogh, ZK Nagy, O Tsinman, A Avdeef, ...
European Journal of Pharmaceutical Sciences 45 (5), 698-707, 2012
2182012
Potentiometric pKa determination of water-insoluble compounds: validation study in methanol/water mixtures
K Takács-Novák, KJ Box, A Avdeef
International journal of pharmaceutics 151 (2), 235-248, 1997
2181997
Lipophilicity of antibacterial fluoroquinolones
K Takács-Novák, M Józan, I Hermecz, G Szász
International Journal of Pharmaceutics 79 (1-3), 89-96, 1992
2161992
Potentiometric and spectrophotometric pKa determination of water-insoluble compounds: validation study in a new cosolvent system
G Völgyi, R Ruiz, K Box, J Comer, E Bosch, K Takács-Novák
Analytica chimica acta 583 (2), 418-428, 2007
2142007
On the partition of ampholytes: application to blood–brain distribution
MH Abraham, K Takács-Novák, RC Mitchell
Journal of pharmaceutical sciences 86 (3), 310-315, 1997
1781997
Study of pH-dependent solubility of organic bases. Revisit of Henderson-Hasselbalch relationship
G Völgyi, E Baka, KJ Box, JEA Comer, K Takács-Novák
Analytica Chimica Acta 673 (1), 40-46, 2010
1402010
Reliability of logP predictions based on calculated molecular descriptors: a critical review
D Eros, I Kovesdi, L Orfi, K Takacs-Novak, G Acsády, G Kéri
Current medicinal chemistry 9 (20), 1819-1829, 2002
1362002
Equilibrium versus kinetic measurements of aqueous solubility, and the ability of compounds to supersaturate in solution—a validation study
KJ Box, G Völgyi, E Baka, M Stuart, K Takács-Novák, JEA Comer
Journal of pharmaceutical sciences 95 (6), 1298-1307, 2006
1342006
Equilibrium solubility measurement of ionizable drugs–consensus recommendations for improving data quality
A Avdeef, E Fuguet, A Llinàs, C Ràfols, E Bosch, G Völgyi, T Verbić, ...
Admet and Dmpk 4 (2), 117-178, 2016
1212016
Multiwavelength spectrophotometric determination of acid dissociation constants: Part V: microconstants and tautomeric ratios of diprotic amphoteric drugs
K Takács-Novák, KY Tam
Journal of pharmaceutical and biomedical analysis 21 (6), 1171-1182, 2000
1122000
Correlations between cytotoxicity and topography of some 2-arylidenebenzocycloalkanones determined by X-ray crystallography
JR Dimmock, GA Zello, EO Oloo, JW Quail, HB Kraatz, P Perjési, F Aradi, ...
Journal of Medicinal Chemistry 45 (14), 3103-3111, 2002
1052002
Lipophilicity of amphoteric molecules expressed by the true partition coefficient
K Takács-Novák, M Józan, G Szász
International journal of pharmaceutics 113 (1), 47-55, 1995
1011995
Determination of protonation macro-and microconstants and octanol/water partition coefficient of the antiinflammatory drug niflumic acid
K Takács-Novák, A Avdeef, KJ Box, B Podányi, G Szász
Journal of pharmaceutical and biomedical analysis 12 (11), 1369-1377, 1994
941994
Acid-base properties and proton-speciation of vancomycin
K Takács-Novák, B Noszál, M Tókés-Kövesdi, G Szász
International journal of pharmaceutics 89 (3), 261-263, 1993
841993
Ion-pair partition of quaternary ammonium drugs: The influence of counter ions of different lipophilicity, size, and flexibility
K Takács-Novák, G Szász
Pharmaceutical research 16, 1633-1638, 1999
801999
Theoretical conformational analysis for neurotransmitters in the gas phase and in aqueous solution. Norepinephrine
PI Nagy, G Alagona, C Ghio, K Takács-Novák
Journal of the American Chemical Society 125 (9), 2770-2785, 2003
702003
Microscopic Protonation/Deprotonation Equilibria of the Anti‐Inflammatory Agent Piroxicam
K Takács‐Novák, J Kökösi, B Podányi, B Noszál, RS Tsai, G Lisa, ...
Helvetica chimica acta 78 (3), 553-562, 1995
651995
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