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h5 指数:41
h5 中位数:50

h5 指数是指在过去整整 5 年中所发表文章的 h 指数。h 指在 2018-2022 年间发表的 h 篇文章每篇至少都被引用过 h 次的最大值。隐藏

出版物的 h5 中位数，是指出版物的 h5 指数所涵盖的所有文章获得的引用次数的中位值。隐藏

#11 Medicinal Chemistry

标题/作者	引用次数	年份
The Ecstasy and Agony of Assay Interference Compounds C Aldrich, C Bertozzi, GI Georg, L Kiessling, C Lindsley, D Liotta, ... ACS Medicinal Chemistry Letters 8 (4), 379-382	136	2017
Distinct Binding Mode of Multikinase Inhibitor Lenvatinib Revealed by Biochemical Characterization K Okamoto, M Ikemori-Kawada, A Jestel, K von König, Y Funahashi, ... ACS Medicinal Chemistry Letters 6 (1), 89-94	131	2015
Biocatalysis in the Pharmaceutical Industry: The Need for Speed MD Truppo ACS Medicinal Chemistry Letters 8 (5), 476-480	128	2017
INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2, 3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology EW Yue, R Sparks, P Polam, D Modi, B Douty, B Wayland, B Glass, ... ACS Medicinal Chemistry Letters 8 (5), 486-491	115	2017
Discovery of AG-120 (Ivosidenib): A First-in-Class Mutant IDH1 Inhibitor for the Treatment of IDH1 Mutant Cancers J Popovici-Muller, RM Lemieux, E Artin, JO Saunders, FG Salituro, ... ACS Medicinal Chemistry Letters 9 (4), 300-305	92	2018
Practical High-Throughput Experimentation for Chemists M Shevlin ACS Medicinal Chemistry Letters 8 (6), 601-607	84	2017
Design and Synthesis of Tesirine, a Clinical Antibody–Drug Conjugate Pyrrolobenzodiazepine Dimer Payload AC Tiberghien, JN Levy, LA Masterson, NV Patel, LR Adams, S Corbett, ... ACS Medicinal Chemistry Letters 7 (11), 983-987	79	2016
EPZ011989, A Potent, Orally-Available EZH2 Inhibitor with Robust in Vivo Activity JE Campbell, KW Kuntz, SK Knutson, NM Warholic, H Keilhack, TJ Wigle, ... ACS Medicinal Chemistry Letters 6 (5), 491-495	74	2015
Molecular Property Design: Does Everyone Get It? PD Leeson, RJ Young ACS Medicinal Chemistry Letters 6 (7), 722-725	66	2015
Aryl Pyrazoles as Potent Inhibitors of Arginine Methyltransferases: Identification of the First PRMT6 Tool Compound LH Mitchell, AE Drew, SA Ribich, N Rioux, KK Swinger, SL Jacques, ... ACS Medicinal Chemistry Letters 6 (6), 655-659	63	2015
Hope and Disappointment: Covalent Inhibitors to Overcome Drug Resistance in Non-Small Cell Lung Cancer J Engel, J Lategahn, D Rauh ACS Medicinal Chemistry Letters 7 (1), 2-5	60	2016
Mitochondria-Localized Fluorescent BODIPY-Platinum Conjugate T Sun, X Guan, M Zheng, X Jing, Z Xie ACS Medicinal Chemistry Letters 6 (4), 430-433	60	2015
Switch in Site of Inhibition: A Strategy for Structure-Based Discovery of Human Topoisomerase IIα Catalytic Inhibitors AT Baviskar, SM Amrutkar, N Trivedi, V Chaudhary, A Nayak, SK Guchhait, ... ACS Medicinal Chemistry Letters 6 (4), 481-485	59	2015
Discovery of Aryl Sulfonamides as Isoform-Selective Inhibitors of NaV1. 7 with Efficacy in Rodent Pain Models T Focken, S Liu, N Chahal, M Dauphinais, ME Grimwood, S Chowdhury, ... ACS Medicinal Chemistry Letters 7 (3), 277-282	57	2016
Small-Molecule CD4-Mimics: Structure-Based Optimization of HIV-1 Entry Inhibition B Melillo, S Liang, J Park, A Schön, JR Courter, JM LaLonde, ... ACS Medicinal Chemistry Letters 7 (3), 330-334	54	2016
Fragment-Based Discovery of a Selective and Cell-Active Benzodiazepinone CBP/EP300 Bromodomain Inhibitor (CPI-637) AM Taylor, A Côté, MC Hewitt, R Pastor, Y Leblanc, CG Nasveschuk, ... ACS Medicinal Chemistry Letters 7 (5), 531-536	53	2016
High-Throughput Screening of Patient-Derived Cultures Reveals Potential for Precision Medicine in Glioblastoma CE Quartararo, E Reznik, AC deCarvalho, T Mikkelsen, BR Stockwell ACS Medicinal Chemistry Letters 6 (8), 948-952	53	2015
BRD4 Structure–Activity Relationships of Dual PLK1 Kinase/BRD4 Bromodomain Inhibitor BI-2536 L Chen, JL Yap, M Yoshioka, ME Lanning, RN Fountain, M Raje, ... ACS Medicinal Chemistry Letters 6 (7), 764-769	53	2015
Structure and Property Guided Design in the Identification of PRMT5 Tool Compound EPZ015666 KW Duncan, N Rioux, PA Boriack-Sjodin, MJ Munchhof, LA Reiter, ... ACS Medicinal Chemistry Letters 7 (2), 162-166	51	2016
Discovery of a Dual PRMT5–PRMT7 Inhibitor D Smil, MS Eram, F Li, S Kennedy, MM Szewczyk, PJ Brown, ... ACS Medicinal Chemistry Letters 6 (4), 408-412	51	2015

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