| Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors S Castellano, D Kuck, M Viviano, J Yoo, F López-Vallejo, P Conti, ... Journal of medicinal chemistry 54 (21), 7663-7677, 2011 | 178 | 2011 |
| An overview of coumarin as a versatile and readily accessible scaffold with broad-ranging biological activities F Annunziata, C Pinna, S Dallavalle, L Tamborini, A Pinto International journal of molecular sciences 21 (13), 4618, 2020 | 171 | 2020 |
| Drug discovery targeting amino acid racemases P Conti, L Tamborini, A Pinto, A Blondel, P Minoprio, A Mozzarelli, ... Chemical reviews 111 (11), 6919-6946, 2011 | 118 | 2011 |
| Inhibition of rhodesain as a novel therapeutic modality for human African trypanosomiasis R Ettari, L Tamborini, IC Angelo, N Micale, A Pinto, C De Micheli, P Conti Journal of Medicinal Chemistry 56 (14), 5637-5658, 2013 | 96 | 2013 |
| The synthesis of Azadirachtin: a potent insect antifeedant SV Ley, A Abad‐Somovilla, JC Anderson, C Ayats, R Bänteli, ... Chemistry–A European Journal 14 (34), 10683-10704, 2008 | 63 | 2008 |
| Antimicrobial activity of resveratrol-derived monomers and dimers against foodborne pathogens LM Mattio, S Dallavalle, L Musso, R Filardi, L Franzetti, L Pellegrino, ... Scientific Reports 9 (1), 19525, 2019 | 57 | 2019 |
| An efficient method for the lipase-catalysed resolution and in-line purification of racemic flurbiprofen in a continuous-flow reactor L Tamborini, D Romano, A Pinto, A Bertolani, F Molinari, P Conti Journal of Molecular Catalysis B: Enzymatic 84, 78-82, 2012 | 56 | 2012 |
| Synthesis, binding affinity at glutamic acid receptors, neuroprotective effects, and molecular modeling investigation of novel dihydroisoxazole amino acids P Conti, M De Amici, G Grazioso, G Roda, A Pinto, KB Hansen, B Nielsen, ... Journal of medicinal chemistry 48 (20), 6315-6325, 2005 | 55 | 2005 |
| Chemoenzymatic synthesis in flow reactors: A rapid and convenient preparation of Captopril V De Vitis, F Dall'Oglio, A Pinto, C De Micheli, F Molinari, P Conti, ... ChemistryOpen 6 (5), 668-673, 2017 | 50 | 2017 |
| An efficient continuous flow process for the synthesis of a non-conventional mixture of fructooligosaccharides P Zambelli, L Tamborini, S Cazzamalli, A Pinto, S Arioli, S Balzaretti, ... Food Chemistry 190, 607-613, 2016 | 49 | 2016 |
| Flow-based stereoselective reduction of ketones using an immobilized ketoreductase/glucose dehydrogenase mixed bed system F Dall'Oglio, ML Contente, P Conti, F Molinari, D Monfredi, A Pinto, ... Catalysis Communications 93, 29-32, 2017 | 47 | 2017 |
| Discovery of covalent inhibitors of glyceraldehyde-3-phosphate dehydrogenase, a target for the treatment of malaria S Bruno, A Pinto, G Paredi, L Tamborini, C De Micheli, V La Pietra, ... Journal of Medicinal Chemistry 57 (17), 7465-7471, 2014 | 47 | 2014 |
| Design and synthesis of novel isoxazole-based HDAC inhibitors P Conti, L Tamborini, A Pinto, L Sola, R Ettari, C Mercurio, C De Micheli European journal of medicinal chemistry 45 (9), 4331-4338, 2010 | 47 | 2010 |
| Development of rhodesain inhibitors with a 3‐bromoisoxazoline warhead R Ettari, L Tamborini, IC Angelo, S Grasso, T Schirmeister, L Lo Presti, ... ChemMedChem 8 (12), 2070-2076, 2013 | 44 | 2013 |
| Stilbenoids: A natural arsenal against bacterial pathogens LM Mattio, G Catinella, S Dallavalle, A Pinto Antibiotics 9 (6), 336, 2020 | 43 | 2020 |
| Biocatalytic N‐Acylation of Amines in Water Using an Acyltransferase from Mycobacterium smegmatis ML Contente, A Pinto, F Molinari, F Paradisi Advanced Synthesis & Catalysis 360 (24), 4814-4819, 2018 | 41 | 2018 |
| Biotransformation with whole microbial systems in a continuous flow reactor: resolution of (RS)-flurbiprofen using Aspergillus oryzae by direct esterification with ethanol in … L Tamborini, D Romano, A Pinto, M Contente, MC Iannuzzi, P Conti, ... Tetrahedron letters 54 (45), 6090-6093, 2013 | 41 | 2013 |
| Synthesis and in vitro/in vivo Evaluation of the Antitrypanosomal Activity of 3‐Bromoacivicin, a Potent CTP Synthetase Inhibitor P Conti, A Pinto, PE Wong, LL Major, L Tamborini, MC Iannuzzi, ... ChemMedChem 6 (2), 329-333, 2011 | 41 | 2011 |
| Synthesis and pharmacological characterization at glutamate receptors of the four enantiopure isomers of tricholomic acid A Pinto, P Conti, MD Amici, L Tamborini, U Madsen, B Nielsen, ... Journal of medicinal chemistry 51 (7), 2311-2315, 2008 | 40 | 2008 |
| Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow … S Castellano, L Tamborini, M Viviano, A Pinto, G Sbardella, P Conti The Journal of Organic Chemistry 75 (21), 7439-7442, 2010 | 38 | 2010 |
