Efficient Synthesis of 3H-Imidazo[4,5-b]pyridines from Malononitrile and 5-Amino-4-(cyanoformimidoyl)imidazoles

MEA Zaki, MF Proença, BL Booth - The Journal of Organic …, 2003 - ACS Publications
1-Aryl-5-amino-4-(cyanoformimidoyl) imidazoles 2 were reacted with malononitrile under
mild experimental conditions and led to 3-aryl-5, 7-diamino-6-cyano-3 H-imidazo [4, 5-b] …

Benzo [4, 5] imidazo [2, 1-b] quinazolin-12-ones and benzo [4, 5] imidazo [1, 2-a] pyrido [2, 3-d] pyrimidin-5-ones by a sequential N-acylation–SNAr reaction

KK Gnanasekaran, NP Muddala, RA Bunce - Tetrahedron letters, 2015 - Elsevier
An efficient synthesis of benzo [4.5] imidazo [2, 1-b] quinazolin-12-ones and benzo [4, 5]
imidazo [1, 2-a] pyrido [2, 3-d] pyrimidin-5-ones is reported from the reaction of 2 …

One-pot microwave-assisted protocol for the synthesis of substituted 2-amino-1H-imidazoles

DS Ermolat'ev, B Savaliya, A Shah… - Molecular diversity, 2011 - Springer
An efficient microwave-assisted one-pot two-step protocol was developed for the
construction of disubstituted 2-amino-1 H-imidazoles. This process involves the sequential …

The synthesis of 4H‐imidazo[5,1‐c][1,4]benzothiazine derivatives

RI Fryer, RF Lauer, EJ Trybulski… - Journal of …, 1983 - Wiley Online Library
A facile synthesis of the 4H‐imidazo [5, 1‐c][1, 4] benzothiazine ring system is described.
The synthesis utilized the annulation of an imidazole ring onto a 2H‐1, 4‐benzothiazin‐3 …

Synthesis and ring opening reactions of tetrahydroimidazo [1, 5-b][1, 2, 4] oxadiazol-2 (1 H)-thiones

N Coşkun, FT Tat - Phosphorus, Sulfur, and Silicon and the …, 2003 - Taylor & Francis
1, 3-Dipolar cycloaddition of imidazoline 3-oxides 1 with methylisothiocyanate proceeds
regio-and diastereoselectively to give tetrahydroimidazo [1, 5-b][1, 2, 4] oxadiazol-2 (1 H) …

Novel Regioselective Formation of S- and N-Hydroxyl-Alkyls of 5-(3-Chlorobenzo[b]Thien-2-yl)-3-Mercapto-4H-1,2,4-Triazole and A Facile Synthesis of Triazolo …

ESH El Ashry, AA Kassem, H Abdel-Hamid… - … , and Nucleic Acids, 2007 - Taylor & Francis
Regioselective alkylation of 5-(3-chlorobenzo [b] thien-2-yl)-4H-1, 2, 4-triazole (1) with
hydroxy alkylating agents 2, 3, 13, and the 2, 3-O-isopropylidene-1-O-(p-tolylsulfonyl) …

Synthesis of 5-arylmethylidene-3-(arylmethylideneamino)thiazolidine-2,4-diones via triazine ring cleavage of tetrahydroimidazothiazolotriazinediones and their …

AN Izmest'ev, GA Gazieva, NG Kolotyrkina… - Chemistry of …, 2020 - Springer
Cleavage of 1, 3-dimethyl-3, 3a, 9, 9a-tetrahydroimidazo [4, 5-e] thiazolo [3, 2-b][1, 2, 4]
triazine-2, 7 (1 H, 6 H)-diones upon treatment with aromatic aldehydes has been shown to …

DABCO catalyzed highly regioselective synthesis of fused imidazo-heterocycles in aqueous medium

VM Bangade, BC Reddy, PB Thakur, BM Babu… - Tetrahedron …, 2013 - Elsevier
An efficient regioselective synthesis of 3-aryl imidazo [1, 2-a] pyridines, 5-aryl imidazo [2, 1-
b] thiazoles, and 3-aryl benzo [d] imidazo [2, 1-b][1, 3] thiazoles is described by the reaction …

Microwave‐Assisted One‐Pot Synthesis of Substituted 3‐Bromoimidazo[1,2‐a]pyridines and Imidazoheterocycles

SM Patil, M Mascarenhas, R Sharma… - Journal of …, 2014 - Wiley Online Library
Herein, an efficient, one‐pot microwave‐assisted synthesis of a diverse set of 3‐
bromoimidazo [1, 2‐a] pyridines is being reported with good yields (40–85%). The method …

[HTML][HTML] Synthesis of functionalized imidazo [4, 5-e] thiazolo [3, 2-b] triazines by condensation of imidazo [4, 5-e] triazinethiones with DMAD or DEAD and …

AN Izmest'ev, DB Vinogradov… - Beilstein Journal of …, 2021 - beilstein-journals.org
Two series of functionalized imidazothiazolotriazine derivatives were synthesized via the
condensation of imidazo [4, 5-e]-1, 2, 4-triazine-3-thiones with acetylenedicarboxylic acid …