Potential of using low density lipoproteins (LDLs) as carriers of radioimaging agents for the early identification of atherosclerotic lesions and cervical cancer cells

W Xiao - 1999 - research.library.mun.ca
… transfer of a hydrophobic radiophannaceutical into acetylated … cholesteryl ester molecules
in its oily core, incorporation of … been widely employed in loading drugs into LDL, and in our …

Ellipticine derivatives with an affinity to the estrogen receptor. An approach to develop intercalating drugs with a specific effect on the hormone-dependent breast …

A Delbarre, R Oberlin, BP Roques… - Journal of medicinal …, 1985 - ACS Publications
RAC « 10™4) and their chloro derivatives 5Z and 5E (RAC = … Mixed compounds exhibit
RAC between 0.0005 and 0.0008. … ) spontaneously crystallized from the oily residue. The E …

Personalized pharmacological therapy for ARDS: a light at the end of the tunnel

PL Silva, P Pelosi, PRM Rocco - … Opinion on Investigational Drugs, 2020 - Taylor & Francis
… N-Acetylcysteine has been studied in ARDS due to its action increasing glutathione levels
… D3 (300,000 IU = 7.5 mg cholecalciferol in oily solution, administered 7 days preoperatively) …

Network pharmacology, molecular docking study, and in vivo validation of the wound healing activity of the Red Sea soft coral Paralemnalia thyrsoides (Ehrenberg …

RTM el-dien, SA Maher, M Hisham, EA Saber… - Beni-Suef University …, 2024 - Springer
… associated with wound healing, including AKT1(RAC-alpha serine/threonine–protein kinase),
… thyrsoides metabolites, very little has been discovered regarding the drug’s mechanism of …

β-Agonist and Hormone Immunoassays in Food

C Xu, H Kuang, L Xu, C Xu, H Kuang, L Xu - Food Immunoassay, 2019 - Springer
… Medically, these drugs have the effect of relaxing smooth … of RAC, one way is changing
the hydroxyl group of RAC to … The oily crude preparation was dissolved in ethyl acetate and …

N‐Substituted Nipecotic Acids as (S)‐SNAP‐5114 Analogues with Modified Lipophilic Domains

MC Böck, G Höfner, KT Wanner - ChemMedChem, 2020 - Wiley Online Library
… disorders is the application of drugs that inhibit the GABA … Serving as lead structure of this
study, rac-SNAP-5114 (rac-2… The oily or solid residue was solved in dry MeCN. Racemic, (…

Protective effect and mechanism of plant-based monoterpenoids in non-alcoholic fatty liver diseases

W Zhang, H Lin, W Cheng, Z Huang… - Journal of Agricultural …, 2022 - ACS Publications
drugs for NAFLD. This review provides a reference for the development of NAFLD drugs as
well … It is a colorless to pale yellow oily liquid with a sweet rose odor and has low solubility in …

Rational Design and Development of a Soluble Mesoporous Carrier for the Solidification of a Preconcentrated Self-Nanoemulsion Formulation

I Kuncahyo, A Indrayati, S Choiri - ACS omega, 2023 - ACS Publications
drug was used as a drugdrug release at 5 min due to the inflection point of the drug release
profile was selected. In addition, the multiple-point method was applied to compare the drug

Practical synthesis of the C-ring precursor of paclitaxel from 3-methoxytoluene

K Fukaya, Y Yamaguchi, A Watanabe… - The Journal of …, 2016 - nature.com
… been used as an anticancer drug. The challenging structure as … For the resolution of rac-9,
we chose lipase-catalyzed … % ee) as a mixture of oily product and crystalline residue, which …

Stereoselective Hydrolase‐Catalyzed Processes in Continuous‐Flow Mode

Z Boros, G Hornyánszky, J Nagy… - Cascade Biocatalysis …, 2014 - Wiley Online Library
… The search for more efficient drugs and agrochemicals … in the KRs of the three differently
flexible amines rac-19a,c,d as a … (1-phenylethanol rac-23i) by acetylation catalyzed by variously …