[PDF][PDF] An overview on the mechanisms of solubility and dissolution rate enhancement in solid dispersion
S Sapkal, M Babhulkar, A Rathi, G Mehetre… - Int J Pharm Tech …, 2013 - researchgate.net
… In this article more emphasis given to the mechanisms by which solubility & dissolution rate
occurs in solid dispersions. The possible mechanisms may be by particle size reduction and …
occurs in solid dispersions. The possible mechanisms may be by particle size reduction and …
Solid dispersions, part I: recent evolutions and future opportunities in manufacturing methods for dissolution rate enhancement of poorly water-soluble drugs
DN Bikiaris - Expert opinion on drug delivery, 2011 - Taylor & Francis
… dissolution enhancement of SDs is based on the fact that drugs in the nanoscale range, or in
amorphous phase, dissolve … the drug and the mechanism of dissolution rate enhancement. …
amorphous phase, dissolve … the drug and the mechanism of dissolution rate enhancement. …
Dissolution rate enhancement of loratadine in polyvinylpyrrolidone K-30 solid dispersions by solvent methods
F Frizon, J de Oliveira Eloy, CM Donaduzzi, ML Mitsui… - Powder technology, 2013 - Elsevier
… dissolution rate is most likely the limiting step in the intestinal absorption [14]. Thus, the
dissolution rate enhancement is of … the enhancement in the dissolution rate of loratadine in solid …
dissolution rate enhancement is of … the enhancement in the dissolution rate of loratadine in solid …
Solid dispersions, part II: new strategies in manufacturing methods for dissolution rate enhancement of poorly water-soluble drugs
DN Bikiaris - Expert opinion on drug delivery, 2011 - Taylor & Francis
… dissolution rate enhancement of such drugs. Among such techniques, nanosuspensions
and drug formulation in solid … been applied for the dissolution enhancement of poorly water-…
and drug formulation in solid … been applied for the dissolution enhancement of poorly water-…
[HTML][HTML] Formulation development and dissolution rate enhancement of efavirenz by solid dispersion systems
… dissolution rate of efavirenz using solid dispersion systems (binary and ternary). A comparison
between solvent and fusion method was also investigated. Solid … solid dispersion system. …
between solvent and fusion method was also investigated. Solid … solid dispersion system. …
Strongly enhanced dissolution rate of fenofibrate solid dispersion tablets by incorporation of superdisintegrants
P Srinarong, JH Faber, MR Visser, WLJ Hinrichs… - European Journal of …, 2009 - Elsevier
… was incorporated in the drug containing solid dispersions than when it was physically mixed
with the solid dispersions. The dissolution rate enhancement strongly depended on the type …
with the solid dispersions. The dissolution rate enhancement strongly depended on the type …
[PDF][PDF] Dissolution rate enhancement of alprazolam by solid dispersion
… When solubility and dissolution rate of solid dispersion of Alprazolam with PVP K30 were …
solid dispersion carrier seems more important for the initial enhancement of dissolution rate. …
solid dispersion carrier seems more important for the initial enhancement of dissolution rate. …
[PDF][PDF] Solubility and dissolution rate enhancement of curcumin using kollidon VA64 by solid dispersion technique
… and dissolution rate enhancement of curcumin by solid dispersion technique. For solid
dispersion preparation, Kollidon VA 64 polymer was selected as a hydrophilic carrier. Solid …
dispersion preparation, Kollidon VA 64 polymer was selected as a hydrophilic carrier. Solid …
Dissolution rate enhancement and physicochemical characterization of carbamazepine-poloxamer solid dispersions
DP Medarević, K Kachrimanis, M Mitrić… - Pharmaceutical …, 2016 - Taylor & Francis
… This study investigates the potential of poloxamers as solid dispersions (SDs) carriers in
improving the dissolution rate of a poorly soluble drug, carbamazepine (CBZ). Solid dispersions …
improving the dissolution rate of a poorly soluble drug, carbamazepine (CBZ). Solid dispersions …
[PDF][PDF] Dissolution rate enhancement of aceclofenac by solid dispersion technique
… rate of dissolution of drugs having limited watersolubility are frequently required [5]. Enhancement
in the dissolution rate … this characteristic such as solid dispersions, micronization, salt …
in the dissolution rate … this characteristic such as solid dispersions, micronization, salt …
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