Comparative clinical pharmacokinetics and pharmacodynamics of HIV-1 integrase strand transfer inhibitors: an updated review
… review summarizes and compares the pharmacokinetics and pharmacodynamics of the
integrase strand transfer inhibitor agents, and describes specific pharmacokinetic considerations …
integrase strand transfer inhibitor agents, and describes specific pharmacokinetic considerations …
Comparative clinical pharmacokinetics and pharmacodynamics of HIV-1 integrase strand transfer inhibitors
AT Podany, KK Scarsi, CV Fletcher - Clinical pharmacokinetics, 2017 - Springer
… This review summarizes the clinical pharmacokinetics of the three INSTIs currently
approved by the US Food and Drug Administration (FDA) for treatment of HIV in adult patients. …
approved by the US Food and Drug Administration (FDA) for treatment of HIV in adult patients. …
Pharmacokinetics and pharmacodynamics of cabotegravir, a long-acting HIV integrase strand transfer inhibitor
D Cattaneo, C Gervasoni - … of drug metabolism and pharmacokinetics, 2019 - Springer
… review, we aimed to summarize the pre-clinical and clinical … in the pharmacokinetics of
cabotegravir when comparing the two … inhibitor of HIV-1 integrase-catalyzed viral cDNA strand …
cabotegravir when comparing the two … inhibitor of HIV-1 integrase-catalyzed viral cDNA strand …
HIV-1 integrase strand transfer inhibitors: a review of current drugs, recent advances and drug resistance
N Mbhele, B Chimukangara, M Gordon - International journal of …, 2021 - Elsevier
… in INSTIs for HIV-1 treatment, we focus our review on the retroviral integrase, development
of … BIC also displays an improved resistance profile over RAL and EVG, comparable with that …
of … BIC also displays an improved resistance profile over RAL and EVG, comparable with that …
A clinical review of HIV integrase strand transfer inhibitors (INSTIs) for the prevention and treatment of HIV-1 infection
AV Zhao, RD Crutchley, RC Guduru, K Ton, T Lam… - Retrovirology, 2022 - Springer
… This article reviews current literature on the clinical pharmacology of INSTIs, … recent
comprehensive review for additional information related to the comparative clinical pharmacokinetics …
comprehensive review for additional information related to the comparative clinical pharmacokinetics …
The clinical pharmacology of integrase inhibitors
G Di Perri, A Calcagno, A Trentalange… - … Clinical Pharmacology, 2019 - Taylor & Francis
… non-inferiority designed comparative clinical trials, which led … HIV-1 RNA at day 8 and the
proportion of subjects with HIV-1 … Clinical pharmacology of the HIV integrase strand transfer …
proportion of subjects with HIV-1 … Clinical pharmacology of the HIV integrase strand transfer …
[HTML][HTML] Pharmacokinetic drug interactions of integrase strand transfer inhibitors
CH Lu, EM Bednarczyk, LM Catanzaro, A Shon… - … in Pharmacology and …, 2021 - Elsevier
… The integrase strand transfer inhibitor (INSTI)-containing regimens are currently considered
as … This review provides a summary of pharmacokinetic interactions with INSTIs and future …
as … This review provides a summary of pharmacokinetic interactions with INSTIs and future …
Clinical safety considerations of integrase strand transfer inhibitors in the older population living with HIV
E Vider, EM Gavioli - Drugs & Aging, 2021 - Springer
… review utilizing the keywords of “integrase strand transfer … DTG/RPV group in comparison to
the current ART regimen (CAR… with a high genetic barrier to HIV-1 resistance [38]. Bictegravir …
the current ART regimen (CAR… with a high genetic barrier to HIV-1 resistance [38]. Bictegravir …
HIV-1 integrase inhibitors: a comparative review of efficacy and safety
KK Scarsi, JP Havens, AT Podany, SN Avedissian… - Drugs, 2020 - Springer
… with HIV are the integrase strand transfer inhibitors (INSTIs). … favorable pharmacokinetic
and pharmacodynamic properties, … This review summarizes the current use of INSTIs in adults …
and pharmacodynamic properties, … This review summarizes the current use of INSTIs in adults …
Clinical pharmacology profile of raltegravir, an HIV‐1 integrase strand transfer inhibitor
DM Brainard, LA Wenning, JA Stone… - … Pharmacology, 2011 - Wiley Online Library
… Clinical efficacy comparing coadministration of … this review are overall not clinically meaningful
with respect to raltegravir's safety and efficacy profile. Raltegravir's clinical pharmacology …
with respect to raltegravir's safety and efficacy profile. Raltegravir's clinical pharmacology …