Recent progress in the development of β2 adrenergic receptor agonists: A patent review (2015-2020)
G Xing, C Yi, P Dou, Z Zhi, B Lin… - Expert Opinion on …, 2021 - Taylor & Francis
… The synthetic compounds, especially those compounds with muscarinic receptor antagonist
and β 2 AR agonist dual activities represent the future direction toward the development of …
and β 2 AR agonist dual activities represent the future direction toward the development of …
[HTML][HTML] Adrenoceptors—New roles for old players
… /or β 2 ‐adrenoceptors, more recent preclinical evidence supports a possible role of β 3 ‐…
existing uses as well as several potential future uses require further investigation, hopefully …
existing uses as well as several potential future uses require further investigation, hopefully …
An overview of the efficacy and safety of β2-Adrenoceptor antagonists for the treatment of chronic obstructive pulmonary disease
MG Matera, P Rogliani, L Calzetta… - Expert Opinion on Drug …, 2024 - Taylor & Francis
… minimal preference for β 2 -AR over β 1 -AR present a complex … randomized prospective
study assessing the effects of a β 2 -… careful consideration and personalised treatment plans. If β-…
study assessing the effects of a β 2 -… careful consideration and personalised treatment plans. If β-…
β2 Agonists
CK Billington, RB Penn, IP Hall - … and Therapeutics of Asthma and COPD, 2017 - Springer
… of β agonist use (pharmacogenetics). Finally we comment on what the future may hold for the
use of β agonists in … classes of β agonists available and consider their current clinical use. …
use of β agonists in … classes of β agonists available and consider their current clinical use. …
[PDF][PDF] Alpha adrenergic receptors in clinical practice–Present and future
P Lechsner, EG Ban - Acta Marisiensis-Seria Medica, 2022 - sciendo.com
… the adrenergic pathways for alpha 1 and alpha 2 receptors and the current as well as potential
future … Overall, there is ongoing research into a multitude of directions with a promising …
future … Overall, there is ongoing research into a multitude of directions with a promising …
Beta2-adrenoceptor agonists in Parkinson's disease and other synucleinopathies
L Magistrelli, C Comi - Journal of Neuroimmune Pharmacology, 2020 - Springer
… current knowledge in the field, opening with an outlook on the β adrenergic system and closing
with future directions… Most studies conclude that β2 adrenergic agonists exert a protective …
with future directions… Most studies conclude that β2 adrenergic agonists exert a protective …
[HTML][HTML] Detailed insight on β-adrenoceptors as therapeutic targets
BK Velmurugan, R Baskaran, CY Huang - Biomedicine & Pharmacotherapy, 2019 - Elsevier
… One recent study has found that β 2 -agonists regulate the transcription of α-synuclein gene
… [66], which has opened a new path toward identification of biased ligands and development …
… [66], which has opened a new path toward identification of biased ligands and development …
Adrenergic agonists and antagonists as antiglaucoma agents: a literature and patent review (2013–2019)
A Nocentini, CT Supuran - Expert Opinion on Therapeutic Patents, 2019 - Taylor & Francis
… current therapeutic arsenal for reducing IOP includes prostaglandin analogs, β-blockers,
carbonic anhydrase inhibitors, α-adrenergic agonist, … of art on adrenergic modulators for treating …
carbonic anhydrase inhibitors, α-adrenergic agonist, … of art on adrenergic modulators for treating …
State-of-the-art beta-adrenoreceptor agonists for the treatment of asthma
WT Garzon-Siatoya, I Carrillo-Martin… - Expert opinion on …, 2022 - Taylor & Francis
… β 2 -adrenoreceptor agonists with bronchodilating effects that last for more than 24 hours
(ultra-LABAs), and other more novel molecules are a primary focus of research in recent years …
(ultra-LABAs), and other more novel molecules are a primary focus of research in recent years …
β2-adrenoceptor function in asthma
Y Amrani, P Bradding - Advances in Immunology, 2017 - Elsevier
… More importantly, we present our latest research describing the role played by mast cells in
impairing β2-adrenoceptor … Future clinical trials are needed to determine whether TAS2R …
impairing β2-adrenoceptor … Future clinical trials are needed to determine whether TAS2R …