The β2-adrenergic receptor-ROS signaling axis: An overlooked component of β2AR function?
KM Rambacher, NH Moniri - Biochemical pharmacology, 2020 - Elsevier
… The β2-adrenergic receptor (β2AR), a prototype of the G protein-coupled receptor (GPCR) …
rapid bronchodilation and is therefore the current gold standard for therapeutic treatment of …
rapid bronchodilation and is therefore the current gold standard for therapeutic treatment of …
[PDF][PDF] Beta-adrenoceptors in obstetrics and gynecology
B Modzelewska - Dev Period Med, 2016 - researchgate.net
… to the future with both caution and hope, the potential metamorphosis of beta3adrenoceptor
agonists … e aim of this Commentary is to briefly review the current state of knowledge on beta-…
agonists … e aim of this Commentary is to briefly review the current state of knowledge on beta-…
[HTML][HTML] The Principles of Ligand Specificity on beta-2-adrenergic receptor
… fingerprint of the β 2 -adrenergic receptor (β 2 AR). β-adrenoceptors belong to rhodopsin-like …
& Matera, MG beta(2) -adrenoceptor agonists: current and future direction. British journal of …
& Matera, MG beta(2) -adrenoceptor agonists: current and future direction. British journal of …
Usage patterns of short-acting β2-agonists and inhaled corticosteroids in asthma: a targeted literature review
Despite the availability of effective asthma treatments, some patients are poorly controlled
because of overreliance on short-acting β 2 -agonists (SABAs) and underuse of inhaled …
because of overreliance on short-acting β 2 -agonists (SABAs) and underuse of inhaled …
Thyronamines and derivatives: physiological relevance, pharmacological actions, and future research directions
CS Hoefig, R Zucchi, J Köhrle - Thyroid, 2016 - liebertpub.com
… The present review will address the most … is also present in other tissues and if further amino
acid decarboxylases are also involved in this process need to be further tested in the future. …
acid decarboxylases are also involved in this process need to be further tested in the future. …
Pharmacological targeting of β2‐adrenoceptors is neuroprotective in the LPS inflammatory rat model of Parkinson's disease
E O'Neill, JD Yssel, C McNamara… - British journal of …, 2020 - Wiley Online Library
… high selectivity as a β 2 -adrenoceptor agonist, formoterol is … In the present investigation, the
immunomodulatory and … in both the forehand and backhand direction at 7 and 13 days post-…
immunomodulatory and … in both the forehand and backhand direction at 7 and 13 days post-…
[HTML][HTML] Allosteric modulation of cannabinoid receptor 1—Current challenges and future opportunities
S Hryhorowicz, M Kaczmarek-Ryś… - International Journal of …, 2019 - mdpi.com
… the complexity of the structure, function, and activity of cannabinoid receptors. In this
paper, we present the latest advances in research on the CB1R, its allosteric modulation and …
paper, we present the latest advances in research on the CB1R, its allosteric modulation and …
GS-5759, a bifunctional β2-adrenoceptor agonist and phosphodiesterase 4 inhibitor for chronic obstructive pulmonary disease with a unique mode of action: effects on …
T Joshi, D Yan, O Hamed, SL Tannheimer… - … of Pharmacology and …, 2017 - ASPET
… -containing pharmacophore responsible for β 2 -adrenoceptor agonism in several LABAs has
been … In the present study, we compared the pharmacology of GS-5759 with representative …
been … In the present study, we compared the pharmacology of GS-5759 with representative …
Membrane-facilitated receptor access and binding mechanisms of long-acting β2-adrenergic receptor agonists
… the aqueous path shared by other β2-AR agents. We observed a novel secondary path for
… action of long-acting β2-adrenergic receptor (β2-AR) agonists such as salmeterol has been …
… action of long-acting β2-adrenergic receptor (β2-AR) agonists such as salmeterol has been …
Long-Acting β2-Adrenoceptor Agonists Enhance Glucocorticoid Receptor (GR)–Mediated Transcription by Gene-Specific Mechanisms Rather Than Generic Effects …
In asthma, the clinical efficacy of inhaled corticosteroids (ICSs) is enhanced by long-acting β
2 -adrenoceptor agonists (LABAs). ICSs, or more accurately, glucocorticoids, promote …
2 -adrenoceptor agonists (LABAs). ICSs, or more accurately, glucocorticoids, promote …