… first antagonist was capsazepine, a synthetic form of capsaicin … activity against TRPV1 and
cannabinoid receptor 1. … has been used therapeutically for many years, there is little evidence …

… The TRPV1 antagonist capsazepine (10 μM) blocked the … is a selective and specific CB1
receptor antagonist/inverse … get direct evidence for the involvement of the CB1 receptor, …

… Capsazepine (CAPZ—a synthetic analog of capsaicin) derived by altering the chemical
backbone of capsaicin is the first antagonist … of capsaicin receptor and its location on peripheral …

… cells were blocked by the selective TRPA1 antagonists HC 030031 and A967079 and … with
AITC (1%) or capsaicin (0.5%) or injected with a CGRP receptor antagonist mice sensitized to …

… lacking capsaicin receptors (formerly known as VR1 receptors) [6] … Capsazepine, by an action
in the periaqueductal grey, also … capsaicin treatment and TRPV1 antagonists all result in a …

… receptor antagonist bicuculline (10 μM) and Glycine receptor … (91%) were tested with capsaicin
(0.1 μM) application at the … Increasing evidence indicates that spontaneous and evoked …

… Capsazepine, the antagonist of TRPV1 receptor, reduces the … Another piece of evidence
supporting mast cell involvement … of dorsal horn neurons in the spinal cord (134). Another …

… There is increasing evidence for a crosstalk between TRPV1 … acting as an opioid receptor
antagonist, naloxone may … we assessed the effect of capsaicin, capsazepine, DAMGO, …

… by the capsaicin receptor (transient receptor potential cation … Some evidence suggests
that capsaicin may inhibit signal … in these studies using appropriate antagonists (50). Future …

… antagonist capsazepine did not block the effect of capsaicin on glycinergic mIPSCs, we
conclude that a mechanism independent of TRPV1 receptor … brainstem/spinal cord preparation …