Novel [1,2,4]triazolo[3,4‐b][1,3,4]thiadiazine derivatives embedded with benzimidazole moiety as potent antioxidants
R Sathyanarayana, B Poojary… - Journal of the …, 2020 - Wiley Online Library
… Noticeably, triazolothiadiazines formed by the combination of … ,21 tubulin inhibitor,22
antimicrobial,23 acetyl- and butyryl-… scavenging activity was performed for the synthesized …
antimicrobial,23 acetyl- and butyryl-… scavenging activity was performed for the synthesized …
[HTML][HTML] Predictive quantitative structure–activity relationship modeling of the antifungal and antibiotic properties of triazolothiadiazine compounds
… series of triazolothiadiazine derivatives to … antifungal and antibiotic activities. The predictive
models developed demonstrate the method and serve as tools to develop new antimicrobial …
models developed demonstrate the method and serve as tools to develop new antimicrobial …
A Convenient One-Pot and Rapid Microwave-Assisted Synthesis of Biologically Active s-Triazolo [3, 4-b][1, 3, 4] Thiadiazine and s-Triazolo [3, 4-b][1, 3, 4] Thiadiazole …
AFM El-Mahdy, HAH El-Sherief… - … of Nanoscience and …, 2020 - ingentaconnect.com
… INTRODUCTION s-Triazole and its derivatives have been received an … Synthesis and
studies on some new fluorine containing triazolothiadiazines as possible antibacterial, antifungal …
studies on some new fluorine containing triazolothiadiazines as possible antibacterial, antifungal …
Synthesis and biological evaluation of 3, 6-dialkylsubstituted-[1, 2, 4] triazolo [3, 4-b][1, 3, 4] thiadiazoles
V Venepally, K Sirisha, CG Kumar, EV Krishna… - Journal of Chemical …, 2018 - Springer
… and lauryl (6f) derivatives exhibited promising antimicrobial activity against the tested strains…
antimicrobial activities in this study depend on the alkyl chain lengths of triazolothiadiazole …
antimicrobial activities in this study depend on the alkyl chain lengths of triazolothiadiazole …
… the alkaline phosphatase inhibition, anticancer, and antileishmanial potential of coumarin–triazolothiadiazine hybrids: design, synthesis, and molecular docking …
… The binding energies derived from docking indicated that almost all the synthesized
coumarin–triazolothiadiazine derivatives exhibited stronger binding affinity for ALP (Supporting …
coumarin–triazolothiadiazine derivatives exhibited stronger binding affinity for ALP (Supporting …
Green Synthesis of Novel Triazolothiadiazine‐Coumarins Catalyzed by Agro Waste Extract: An Approach towards In‐Silico and In‐Vitro Anti‐Fungal Activity
… confirmed that triazolothiadiazine derivatives possess anti-candidal activity (Figure 2). …
derivatives of coumarin substituted-1,2,4-triazolo[3,4-b]1,3,4-thiadiazines 9 i–w were synthesized …
derivatives of coumarin substituted-1,2,4-triazolo[3,4-b]1,3,4-thiadiazines 9 i–w were synthesized …
Monoamine oxidase A and B inhibitory activities of 3, 5-diphenyl-1, 2, 4-triazole substituted [1, 2, 4] triazolo [3, 4-b][1, 3, 4] thiadiazole derivatives
… synthesis and characterization of 3,5-diphenyl-1,2,4-triazole substituted [1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
derivatives … of pharmacological activities including antifungal, antimicrobial, …
derivatives … of pharmacological activities including antifungal, antimicrobial, …
[HTML][HTML] New benzimidazole-1, 2, 4-triazole hybrid compounds: Synthesis, anticandidal activity and cytotoxicity evaluation
… activity against Candida species by broth microdiluation methods. In vitro … antifungal profile.
Compounds 5w was the most active derivative and showed comparable antifungal activity to …
Compounds 5w was the most active derivative and showed comparable antifungal activity to …
[PDF][PDF] In Silico Design, Synthesis, Anti-Microbial and Anti-Tubercular Evaluation of New Series of Benzothiazinone Derivatives Containing Triazolo Thiadiazole Moiety
… antimicrobial activity, but some compounds BTZ4, BTZ7, BTZ8, BTZ9, BTZ15 showed best
Glide docking score as compared to other derivatives, … containing triazolothiadiazole moiety: …
Glide docking score as compared to other derivatives, … containing triazolothiadiazole moiety: …
[HTML][HTML] … ,2,4]triazolo[3,4-b][1,3,4]thiadiazine and [1,2,4]triazolo[3,4-b][1,3,4]thiadiazepine Derivatives: Synthesis, Anti-Viral In Vitro Study and Target Validation Activity
AV Khramchikhin, MA Skryl'nikova, IL Esaulkova… - Molecules, 2022 - mdpi.com
… We proposed a new synthesis route based on the interaction of 3-phenyl-2-… triazolothiadiazines
6, 8 and triazolothiadiazepines 7, 10 (Figure 4). A more detailed analysis of the synthesis …
6, 8 and triazolothiadiazepines 7, 10 (Figure 4). A more detailed analysis of the synthesis …