Design, Synthesis, and Biological Evaluation of Novel 7H-[1,2,4]Triazolo[3,4-b][1,3,4]thiadiazine Inhibitors as Antitumor Agents
… These derivatives were synthesized and biologically screened against full NCI-60 cancer …
–activity relationship (SAR) of triazolothiadiazine compounds with reported anticancer activity …
–activity relationship (SAR) of triazolothiadiazine compounds with reported anticancer activity …
A facile one-pot, three component synthesis of a new series of 1, 3, 4-thiadiazines: Anticancer evaluation and molecular docking studies
S Mamidala, V Vangala, SR Peddi… - Journal of Molecular …, 2021 - Elsevier
… The synthesized thiadiazin derivatives were sketched using maestro build panel and
prepared by using Ligprep application. Finally, the low energy conformers of the ligands were …
prepared by using Ligprep application. Finally, the low energy conformers of the ligands were …
[HTML][HTML] Synthesis, characterization and antimicrobial evaluation of some novel 1, 2, 4-triazolo [3, 4-b][1, 3, 4] thiadiazine bearing substituted phenylquinolin-2-one …
… twenty novel derivatives of phenylquinoline-1,2,4-triazolothiadiazines were synthesized, …
The starting material phenylquinoline-2-one derivatives (1a–1t) for the synthesis of desired …
The starting material phenylquinoline-2-one derivatives (1a–1t) for the synthesis of desired …
Synthesis and properties of some 3-(5-(4-methoxyphenyl) pyrazol-3-yl)-6-R-[1, 2, 4] triazolo [3, 4-b][1, 3, 4] thiadiazoles
SO Fedotov, AS Hotsulia, OI Panasenko - 2022 - dspace.zsmu.edu.ua
… Thus, the preliminary results of the study of biological properties in a number of derivatives
… antifungal activity in a number of synthesized substances. The high affinity of the synthesized …
… antifungal activity in a number of synthesized substances. The high affinity of the synthesized …
Indomethacin based new triazolothiadiazine derivatives: Synthesis, evaluation of their anticancer effects on T98 human glioma cell line related to COX-2 inhibition and …
… antifungal, antibacterial, antiviral and antitumor activities. Recent studies have reported that
new triazolothiadiazine derivatives, … to show significant anticancer activity against different …
new triazolothiadiazine derivatives, … to show significant anticancer activity against different …
[PDF][PDF] Synthesis and Evaluation of Antiphlogistic Activity of Some New 4-Fluorophenyltriazolothiadiazines
PD Bangre, NA Karande, LG Rathi… - Indian Journal of …, 2024 - researchgate.net
… to substantial differences in activity, driving the synthesis and testing of diazine derivatives
… synthesis of new derivatives of triazolothiadiazines (4a-l). The animal study has confirmed …
… synthesis of new derivatives of triazolothiadiazines (4a-l). The animal study has confirmed …
Synthesis of novel 6-(1H-pyrazol-4-yl)-[1, 2, 4] triazolo [3, 4-b][1, 3, 4] thiadiazoles as potential antimicrobial agents
R Pundeer, P Ranjan, R Prakash… - Letters in Organic …, 2018 - ingentaconnect.com
… The additional enhancement in the antifungal activity in the triazolothiadiazole 4f may be …
relies on an expeditious synthesis and biological evaluation of several new derivatives of 3-…
relies on an expeditious synthesis and biological evaluation of several new derivatives of 3-…
Design, Synthesis, Neuroprotective and Antibacterial Activities of 1, 2, 4‐Triazolo [3, 4‐b] 1, 3, 4‐thiadiazole Linked Thieno [2, 3‐d] pyrimidine Derivatives and In Silico …
T Settypalli, VR Chunduri, N Kerru… - …, 2019 - Wiley Online Library
… al33 synthesized some novel 4-amino thienopyrimidines (VI) and studied antimicrobial activity
… of thienopyrimdine-triazolothiadiazole hybrids were designed, synthesized, characterized …
… of thienopyrimdine-triazolothiadiazole hybrids were designed, synthesized, characterized …
In silico activity and target prediction analyses of three triazolothiadiazine derivatives
C Sucularlı, B Tozkoparan, SP Aytaç - Acta Medica, 2022 - actamedica.org
… of newly synthesized or known compounds and drugs. Previously, three novel triazolothiadiazine
derivatives; … growth factor antagonist, anti-inflammatory and antifungal activities. These …
derivatives; … growth factor antagonist, anti-inflammatory and antifungal activities. These …
[HTML][HTML] Synthetic Methods and Pharmacological Potentials of Triazolothiadiazines: A Review
… synthetic pathways for triazolothiadiazine derivatives, such as … wide range of therapeutic
activities such as antimicrobial [2,3]… , triazolothiadiazine derivatives 56 were synthesized through …
activities such as antimicrobial [2,3]… , triazolothiadiazine derivatives 56 were synthesized through …