Discovery, Synthesis and Activity Evaluation of Novel Compounds Bearing 1, 2, 4-triazolo [3, 4-b][1, 3, 4] thiadiazine Moiety: A Review

ED Dincel, NU Güzeldemirci - Sağlık Bilimlerinde İleri Araştırmalar …, 2019 - dergipark.org.tr
Son zamanlarda, geniş ölçekte çeşitlilik gösteren uygulamalardaki kullanımları nedeniyle
azot atomu taşıyan kaynaşmış heterosiklik bileşiklerin kimyası ve biyolojik aktivitesi üzerine …

[HTML][HTML] Synthetic Methods and Pharmacological Potentials of Triazolothiadiazines: A Review

MS Mostafa, IAM Radini, NMA El-Rahman, RE Khidre - Molecules, 2024 - mdpi.com
This review article examines the synthetic pathways for triazolothiadiazine derivatives, such
as triazolo [3, 4-b] thiadiazines, triazolo [5, 1-b] thiadiazines, and triazolo [4, 3-c] …

Synthesis, characterization and antibacterial evaluation of some new 1, 2, 4-triazolo [3, 4-b][1, 3, 4] thiadiazines as potential antibacterial agents

KM Sim, KC Teo - Letters in Drug Design & Discovery, 2018 - ingentaconnect.com
Background: Indole derivatives and 1, 2, 4-triazolo [3, 4-b][1, 3, 4] thiadiazines are important
heterocyclic compounds in medicinal chemistry. They have displayed broad spectrum of …

[PDF][PDF] Synthesis, characterization and biological evaluation of new fused triazine derivatives based on 6-methyl-3-thioxo-1, 2, 4-triazin-5-one

AS Abd El-All, AS Hassan, SA Osman, HAA Yosef… - Acta Pol. Pharm, 2016 - ptfarm.pl
A one-pot reaction of 6-methyl-3-thioxo-3, 4-dihydro-[1, 2, 4] triazin-5-one 1 with selected
aldehydes 2a-d and chloroacetic acid afforded the respective 2-arylidene-6-methyl-thiazolo …

New 6-amino-[1, 2, 4] triazolo [3, 4-b][1, 3, 4] thiadiazines and [1, 2, 4] triazolo [3, 4-b][1, 3, 4] thiadiazin-6-ones: Synthesis, characterization and antibacterial activity …

GL Almajan, SF Barbuceanu, I Saramet… - European journal of …, 2010 - Elsevier
(4-X-Phenylsulfonyl) phenyl] containing 6-amino-[1, 2, 4] triazolo [3, 4-b][1, 3, 4] thiadiazines
and [1, 2, 4] triazolo [3, 4-b][1, 3, 4] thiadiazin-6-ones were synthesized by intermolecular …

Synthesis and properties of 6-(2, 6-dichlorophenyl)-3-(3-methyl-1H-pyrazol-5-yl)-6, 7-dihydro-5H-[1, 2, 4] triazolo [3, 4-b][1, 3, 4] thiadiazine-7-carboxylic acid and its …

SO Fedotov, AS Hotsulia - 2023 - dspace.zsmu.edu.ua
Materials and methods. The synthetic part of the study involved the sequential synthesis of
the original compound 4-amino-5-(3-methyl-1H-pyrazol-5-yl)-1, 2, 4-triazole-3-thiol using a …

Synthesis, spectral characterization and biological evaluation of a novel series of 6-arylsubstituted-3-[2-(4-substitutedphenyl) propan-2-yl]-7H-[1, 2, 4] triazolo [3, 4-b][1 …

P Puthiyapurayil, B Poojary, C Chikkanna… - European journal of …, 2012 - Elsevier
On account of the reported anticancer activity of triazolothiadiazines, we have synthesized a
novel series of 6-arylsubstituted-3-[2-(4-substitutedphenyl) propan-2-yl]-7H-[1, 2, 4] triazolo …

[PDF][PDF] Synthesis of Some Novel Bis [1, 2, 4] triazolo [3, 4-b][1, 3, 4] thiadiazine Derivatives for Antimicrobial Evaluation

CS Reddy, DC Rao, V Yakub… - Acta Chimica …, 2011 - acta-arhiv.chem-soc.si
A new series of novel bis [1, 2, 4] triazolo [3, 4-b][1, 3, 4] thiadiazines 7a–j has been
synthesized by the reaction of [5, 5'-methylenebis (3-methylbenzofuran-7, 5-diyl)] bis [(4 …

Synthesis of some new biologically active bis-(thiadiazolotriazines) and bis-(thiadiazolotriazinyl) alkanes

BS Holla, R Gonsalves, BS Rao, S Shenoy… - Il farmaco, 2001 - Elsevier
4-Amino-3-mercapto-1, 2, 4-triazin-5 (4H)-ones (1) were condensed with dicarboxylic acids
2 to yield bis-(4-oxo-4H-1, 3, 4-thiadiazolo [2, 3-c]-1, 2, 4-triazin-7-yl) alkanes (3b–d, f–h, j–l …

[引用][C] Synthesis and antimicrobial activity of novel heterocycles containing thiazolidinone and 1, 3, 4-oxadiazole moieties

KR Raju, BS Kumar, A Prasad, LK Ravindranath - Journal of Clinical and Analytical …, 2016