Synthesis of some new pyrazoline-based thiazole derivatives and evaluation of their antimicrobial, antifungal, and anticancer activities
… Thiazolyl-pyrazoline derivatives have been used as cholinesterase inhibitors [34]. From
the above facts and our interest in designing new heterocyclic compounds that have the …
the above facts and our interest in designing new heterocyclic compounds that have the …
Synthesis of some novel pyrazoline‐thiazole hybrids and their antimicrobial activities
DM Masoud, RA Azzam, F Hamdy… - Journal of …, 2019 - Wiley Online Library
… series of novel thiazolyl pyrazolines 7a-h, 9a-f, and 11a-f have been synthesized by the reaction
of thioamide derivatives … The antifungal activities of pyrazole derivatives 7a-h, 9a-f, 11a-f…
of thioamide derivatives … The antifungal activities of pyrazole derivatives 7a-h, 9a-f, 11a-f…
A new series of thiazolyl pyrazoline derivatives linked to benzo [1, 3] dioxole moiety: Synthesis and evaluation of antimicrobial and anti-proliferative activities
E Mansour, A Aboelnaga, EM Nassar… - Synthetic …, 2020 - Taylor & Francis
… flavus with inhibition zones in the range of 1.5, 0.5, 1.0, 1.8, … racemosum with inhibition zones
in the range of 0.5–1.9 mm … antifungal action against Penicillium expansum in the range of …
in the range of 0.5–1.9 mm … antifungal action against Penicillium expansum in the range of …
A new approach for the synthesis and biological activities of novel thiazolyl‐pyrazole derivatives
GS Masaret - ChemistrySelect, 2021 - Wiley Online Library
… Moreover, the desired synthesized thiazolyl-pyrazole were screened as antifungal agents
alongside Candida albicans and Aspergillus fumigatus through using Cycloheximide as …
alongside Candida albicans and Aspergillus fumigatus through using Cycloheximide as …
Design, Synthesis, and Evaluation of Antifungal Bioactivity of Novel Pyrazole Carboxamide Thiazole Derivatives as SDH Inhibitors
M Li, W Wang, X Cheng, Y Wang, Y Chen… - Journal of Agricultural …, 2023 - ACS Publications
… In this study, a series of pyrazole carboxamide thiazole derivatives were designed,
synthesized, and evaluated for their antifungal activities against nine plant pathogens in vitro. …
synthesized, and evaluated for their antifungal activities against nine plant pathogens in vitro. …
Synthesis, anticancer evaluation, and molecular docking studies of thiazolyl-pyrazoline derivatives
… The molecular hybridization of thiazole and pyrazoline heterocyclic structures with diverse
… the synthesis of eleven new thiazolyl-pyrazoline derivatives (7a-k) and the evaluation of their …
… the synthesis of eleven new thiazolyl-pyrazoline derivatives (7a-k) and the evaluation of their …
Synthesis and biological evaluation of some novel thiazole-based heterocycles as potential anticancer and antimicrobial agents
… effectiveness of the newly synthesized thiazolyl pyrazoles 6a–h… On the contrary, all synthesized
compounds had no antifungal … carbonyl group and p-tolyl as substituents on the pyrazole …
compounds had no antifungal … carbonyl group and p-tolyl as substituents on the pyrazole …
New thiazolyl‐pyrazoline derivatives bearing nitrogen mustard as potential antimicrobial and antiprotozoal agents
… From these results, it is clear that cyclization of the chalcones–thiazole hybrids 5a–g into
their pyrazoline derivatives increases the antifungal effects of the compounds. …
their pyrazoline derivatives increases the antifungal effects of the compounds. …
Synthesis of new thiazolyl-pyrazolyl-1, 2, 3-triazole derivatives as potential antimicrobial agents
… Pyrazole clubbed with triazole were reported for antifungal [… The convincing antifungal
activity of synthesized compounds in our … newly synthesized thiazolyl-pyrazolyl-1,2,3-triazole,7a-y …
activity of synthesized compounds in our … newly synthesized thiazolyl-pyrazolyl-1,2,3-triazole,7a-y …
Synthesis of novel heterocyclic compounds containing thiazolyl-pyrazoline moiety from chalcone derivatives
ZM Nofal, AM Srour, NM Mansour… - Polycyclic Aromatic …, 2022 - Taylor & Francis
… A new set of thiazolyl-pyrazolines 3a–l was prepared by cyclization of carbothioamides 2a–g
with phenacyl bromide and/or 4-bromo phenacyl bromide. The new chemical entities were …
with phenacyl bromide and/or 4-bromo phenacyl bromide. The new chemical entities were …