Synthesis and biological evaluation of some novel thiazole-based heterocycles as potential anticancer and antimicrobial agents

S Abu-Melha, MM Edrees, HH Salem, NA Kheder… - Molecules, 2019 - mdpi.com
… developing new convenient approaches for the synthesis of … synthesis of some new series
of novel thiazole derivatives … of biological activities for the newly synthesized compounds …

Synthesis and biological evaluation of thiazole-based derivatives with potential against breast cancer and antimicrobial agents

E Pivovarova, A Climova, M Świątkowski… - International Journal of …, 2022 - mdpi.com
biologically-active coordination compounds that may be useful in the design of breast anticancer,
antifungal, and antimicrobialnew copper coordination compounds containing thiazole-…

Synthesis, X-ray analysis, biological evaluation and molecular docking study of new thiazoline derivatives

YN Mabkhot, H Algarni, A Alsayari, A Bin Muhsinah… - Molecules, 2019 - mdpi.com
… The data from the in vitro antitumor evaluation revealed that the thiazolines 5b and 2c were
… study supported anticancer results and showed binding affinities for thiazolines 5b and 2c …

Synthesis of some new pyrazoline-based thiazole derivatives and evaluation of their antimicrobial, antifungal, and anticancer activities

SI Elewa, E Mansour, IF Nassar… - Russian Journal of …, 2020 - Springer
… There are thiazole-based CNS drugs currently used as therapeutic agents for the treatment
… of thiazole derivatives are in clinical trials [22]. Diverse modifications of the thiazole ring at …

Synthesis and biological evaluation of thiazolyl-ethylidene hydrazino-thiazole derivatives: a novel heterocyclic system

LA Al-Mutabagani, FM Abdelrazek, SM Gomha… - Applied Sciences, 2021 - mdpi.com
synthesized a new series of bioactive thiazole derivatives, and … had good anticancer activity,
and that the thiazole derivative 10c … more powerful than the anticancer medication cisplatin. …

Synthesis and biological evaluation of new derivatives of thieno-thiazole and dihydrothiazolo-thiazole scaffolds integrated with a pyrazoline nucleus as anticancer and …

IMM Othman, ZM Alamshany, NY Tashkandi… - RSC …, 2022 - pubs.rsc.org
anticancer activity against A549 and MCF-7 human cancer cell lines as well as antimicrobial
activity of the derivatives bearing thiazole … Furthermore, the thiazoline-pyrazolines IV–VI …

Synthesis and Biological Evaluation of Some Novel Bis-Thiadiazoles as Antimicrobial and Antitumor Agents

WAMA El-Enany, SM Gomha, W Hussein… - Polycyclic Aromatic …, 2021 - Taylor & Francis
… for each of the new products. This research aimed at synthesizing a novel series of derivatives
of bis-thiadiazoles and investigating their antimicrobial and anticancer activity. The results …

[HTML][HTML] Design, synthesis and docking studies of new hydrazinyl-thiazole derivatives as anticancer and antimicrobial agents

AM El-Naggar, A Zidan, EB Elkaeed… - Journal of Saudi …, 2022 - Elsevier
anticancer and antimicrobial properties. The present study is concerned with synthesis and
screening for anticancer and antimicrobial … )hydrazinyl)thiazole derivatives. The structure …

[HTML][HTML] … study, and biological evaluation and of new thiadiazole and thiazole derivatives incorporating isoindoline-1, 3-dione moiety as anticancer and antimicrobial …

WA Mokbel, MA Hosny, SM Gomha, MEA Zaki… - Results in …, 2024 - Elsevier
… of thiadiazole and thiazole-containing drugs, we aim to develop new heterocyclic compounds
integrating these heterocycles, anticipating enhanced and superior biological activities. …

Synthesis, Characterization, and Biological Evaluation of Some Novel Pyrazolo[5,1-b]thiazole Derivatives as Potential Antimicrobial and Anticancer Agents

A Alsayari, AB Muhsinah, YI Asiri, FA Al-Aizari… - Molecules, 2021 - mdpi.com
… and anticancer agents have been thoroughly described in many literature reviews. In …
synthesis of novel pyrazolo[5,1-b]thiazole-based heterocycles was carried out. The synthesized