[HTML][HTML] Synthesis and biological evaluation of thiazolyl-ethylidene hydrazino-thiazole derivatives: a novel heterocyclic system
LA Al-Mutabagani, FM Abdelrazek, SM Gomha… - Applied Sciences, 2021 - mdpi.com
The reaction of 2-(1-(2-(2-(4-methoxybenzylidene) hydrazinyl)-4-methylthiazol-5-yl)
ethylidene) hydrazinecarbothioamide with a range of hydrazonoyl chlorides and α-halo …
ethylidene) hydrazinecarbothioamide with a range of hydrazonoyl chlorides and α-halo …
[HTML][HTML] Synthesis and in vitro evaluation of new nitro-substituted thiazolyl hydrazone derivatives as anticandidal and anticancer agents
Fourteen new thiazolyl hydrazone derivatives were synthesized and evaluated for their
anticandidal activity using a broth microdilution assay. Among the synthesized compounds …
anticandidal activity using a broth microdilution assay. Among the synthesized compounds …
[HTML][HTML] Synthesis, characterization and molecular docking of novel bioactive thiazolyl-thiazole derivatives as promising cytotoxic antitumor drug
SM Gomha, TA Salaheldin, HME Hassaneen… - Molecules, 2015 - mdpi.com
Reactions of ethylidenethiocarbohydrazide with hydrazonoyl halides gave 1, 3-thiazole or 1,
3, 4-thiadiazole derivatives according to the type of hydrazonoyl halides. Treatment of …
3, 4-thiadiazole derivatives according to the type of hydrazonoyl halides. Treatment of …
Synthesis and evaluation of new thiazolyl hydrazone derivatives as potential anticancer agents
Z Asım Kaplancıklı, B Sever… - Letters in Drug …, 2017 - ingentaconnect.com
Background: In recent years, thiazole derivatives incorporated with hydrazone moiety have
attracted a great deal of interest due to their pivotal role in the field of current cancer …
attracted a great deal of interest due to their pivotal role in the field of current cancer …
[HTML][HTML] The synthesis and antiproliferative activities of new arylidene-hydrazinyl-thiazole derivatives
New and known arylidene-hydrazinyl-thiazole derivatives have been synthesized by a
convenient Hantzsch condensation. All compounds were evaluated for their in vitro …
convenient Hantzsch condensation. All compounds were evaluated for their in vitro …
Synthesis and antitumor activity of 1, 3, 4-thiadiazole derivatives bearing coumarine ring
S Gomha, HM Abdel-aziz - Heterocycles, 2015 - ksascholar.dri.sa
In the present study, preparation of a novel series of N'-(3, 5-diphenyl-1, 3, 4-thiadiazol-2
(3H)-ylidene)-2-oxo-2H-chromene-3-carbohydrazide (8a-m) was prepared by two methods …
(3H)-ylidene)-2-oxo-2H-chromene-3-carbohydrazide (8a-m) was prepared by two methods …
Synthesis and SAR study of the novel thiadiazole–imidazole derivatives as a new anticancer agents
In the present study, a novel series of 2-(2-(3-aryl-5-substituted-1, 3, 4-thiadiazol-2 (3H)-
ylidene) hydrazinyl)-4, 4-diphenyl-1H-imidazol-5 (4H)-one derivatives were designed and …
ylidene) hydrazinyl)-4, 4-diphenyl-1H-imidazol-5 (4H)-one derivatives were designed and …
Synthesis of some p-toluenesulfonyl-hydrazinothiazoles and hydrazino-bis-thiazoles and their anticancer activity
V Zaharia, A Ignat, N Palibroda, B Ngameni… - European journal of …, 2010 - Elsevier
A series of novel p-toluenesulfonyl-hydrazinothiazoles and hydrazino-bis-thiazoles
derivatives (2a–f, 3a–f and 5–8) were synthesized by initial condensation of p …
derivatives (2a–f, 3a–f and 5–8) were synthesized by initial condensation of p …
Synthesis and Evaluation of Antimicrobial Activity of Some New Hetaryl‐Azoles Derivatives Obtained from 2‐Aryl‐4‐methylthiazol‐5‐carbohydrazides and Isonicotinic …
A series of new 1, 3, 4‐oxadiazole/thiadiazole and 1, 2, 4‐triazole derivatives have been
synthesized starting from 2‐aryl‐4‐methylthiazol‐5‐carbohydrazides and isonicotinic acid …
synthesized starting from 2‐aryl‐4‐methylthiazol‐5‐carbohydrazides and isonicotinic acid …
[HTML][HTML] Synthesis and biological evaluation of new 1, 3, 4-thiadiazole derivatives as potent antimicrobial agents
Abstract A series of 1, 3, 4-thiadiazole derivatives were designed and synthesized using N-
(4-nitrophenyl) acetohydrazonoyl bromide and 1-[3, 5-dimethyl-1-(4-nitrophenyl)-1 H …
(4-nitrophenyl) acetohydrazonoyl bromide and 1-[3, 5-dimethyl-1-(4-nitrophenyl)-1 H …