Synthesis and biological evaluation of some novel thiazole-based heterocycles as potential anticancer and antimicrobial agents
A novel series of thiazole-based heterocycles was synthesized using 1, 3-dipolar
cycloaddition reactions in the presence of chitosan-grafted-poly (vinylpyridine) as an eco …
cycloaddition reactions in the presence of chitosan-grafted-poly (vinylpyridine) as an eco …
Synthesis, characterization and in vitro anticancer activity of thiabendazole-derived 1, 2, 3-triazole derivatives
K El Bourakadi, MEM Mekhzoum, C Saby… - New Journal of …, 2020 - pubs.rsc.org
A series of thiabendazole-derived 1, 2, 3-triazole compounds were synthesized in good
yields via 1, 3-dipolar cycloaddition through click chemistry approach using different chain …
yields via 1, 3-dipolar cycloaddition through click chemistry approach using different chain …
Eco-friendly synthesis, characterization and biological evaluation of some novel pyrazolines containing thiazole moiety as potential anticancer and antimicrobial …
MM Edrees, SA Melha, AM Saad, NA Kheder… - Molecules, 2018 - mdpi.com
The one-pot synthesis of a series of pyrazoline derivatives containing the bioactive thiazole
ring has been performed through a 1, 3-dipolar cycloaddition reaction of N …
ring has been performed through a 1, 3-dipolar cycloaddition reaction of N …
One-pot synthesis of novel thiazoles as potential anti-cancer agents
Background Thiazole and thiosemicarbazone derivatives are known to have potential
anticancer activity with a mechanism of action related to inhibition of matrix metallo …
anticancer activity with a mechanism of action related to inhibition of matrix metallo …
Design, synthesis and anticancer evaluation of new substituted thiophene-quinoline derivatives
A series of new isoxazolyl, triazolyl and phenyl based 3-thiophen-2-yl-quinoline derivatives
were synthesized adopting click chemistry approach. In addition, the synthesis of new useful …
were synthesized adopting click chemistry approach. In addition, the synthesis of new useful …
Synthesis and Characterization of Some New Bis-Pyrazolyl-Thiazoles Incorporating the Thiophene Moiety as Potent Anti-Tumor Agents
SM Gomha, MM Edrees, FMA Altalbawy - International journal of …, 2016 - mdpi.com
A new series of 1, 4-bis (1-(5-(aryldiazenyl) thiazol-2-yl)-5-(thiophen-2-yl)-4, 5-dihydro-1 H-
pyrazol-3-yl) benzenes 3a–i were synthesized via reaction of 5, 5′-(1, 4-phenylene) bis (3 …
pyrazol-3-yl) benzenes 3a–i were synthesized via reaction of 5, 5′-(1, 4-phenylene) bis (3 …
Pharmacological evaluation of some novel synthesized compounds derived from spiro (cyclohexane-1, 2′-thiazolidines)
EM Flefel, HH Sayed, AI Hashem, EA Shalaby… - Medicinal Chemistry …, 2014 - Springer
A series of novel spiro (cyclohexane-1, 2′-thiazolidine) derivatives 1–5 and spiro
(cyclohexane1, 2′-thiazolo-pyridine) derivatives 6–14 were synthesized. Arylidene …
(cyclohexane1, 2′-thiazolo-pyridine) derivatives 6–14 were synthesized. Arylidene …
Synthesis, Characterization, and Biological Evaluation of Some Novel Pyrazolo[5,1-b]thiazole Derivatives as Potential Antimicrobial and Anticancer Agents
The pharmacological activities of thiazole and pyrazole moieties as antimicrobial and
anticancer agents have been thoroughly described in many literature reviews. In this study …
anticancer agents have been thoroughly described in many literature reviews. In this study …
Design, click synthesis, anticancer screening and docking studies of novel benzothiazole-1, 2, 3-triazoles appended with some bioactive benzofused heterocycles
Abstract New series of benzothiazole-1, 2, 3-triazoles; appended with benzothiazole, isatin
and/or benzimidazole moiety; were designed and synthesized through the click chemistry …
and/or benzimidazole moiety; were designed and synthesized through the click chemistry …
[PDF][PDF] Synthesis of some novel thiazole, thiadiazole and 1, 4-phenylene-bis-thiazole derivatives as potent antitumor agents
SM Gomha, FM Abdelrazek, AH Abdelrahman… - Heterocycles, 2016 - academia.edu
A novel series of 2-ethylidenehydrazono-5-arylazothiazoles 5a-h and 2-
ethylidenehydrazono-5-arylazothiazolones 9a-d were prepared by cyclocondensation of …
ethylidenehydrazono-5-arylazothiazolones 9a-d were prepared by cyclocondensation of …