[PDF][PDF] HAMSTER VAS DEFERENS CONTAINS 6-OPIOID RECEPTORS zyxwvutsrqponmlkjihgfedcbaZYXWVUTSRQPONMLKJIH

AT McKnight, AD Corbett, M Marcoli, HW Kosterlitz - academia.edu
… of the isolated vas deferens of the mouse were inhibited by morphine, … vas deferens of the
hamster for the possible presence of opioid receptors at which morphine has no agonist action

Effects of CA1 α2-adrenergic receptors on morphine-induced exploratory behaviors.

E Beirami… - Physiology & …, 2024 - search.ebscohost.com
… 1) To assess the potential role of morphine in anxiety-related … of mu-opioid receptors agonist,
morphine (6 mg/kg), induced … from sympathetic varicosities of the mouse vas deferens. Br J …

[PDF][PDF] Seyedhosseini Tamijani SM Effects of CA1 α2-adrenergic receptors on morphine-induced exploratory behaviors

E Beirami - Physiology and Pharma - ppj.phypha.ir
… 1) To assess the potential role of morphine in anxiety-related … of mu-opioid receptors agonist,
morphine (6 mg/kg), induced … from sympathetic varicosities of the mouse vas deferens. Br J …

[HTML][HTML] A systematic review of inverse agonism at adrenoceptor subtypes

MC Michel, MB Michel-Reher, P Hein - Cells, 2020 - mdpi.com
… opioid receptors by pre-treatment with morphine [20,53]. Of note, … behaved as a partial
agonist in rat vas deferens. … the receptor number, as assessed by radioligand binding in HepG2 …

[PDF][PDF] PREMATURE EJACULATION–POTENTIAL ROLE OF α2-ADRENOCEPTOR AGONISTS FOR SYMPTOMATIC TREATMENT

J Lehtimäki - utupub.fi
… by triggering contractions in the vas deferens, seminal vesicles, … agonist to prevent any effects
on presynaptic α2-adrenergic … To assess the agonistic effects of fadolmidine on the rodent …

[HTML][HTML] Comparison of the effects of fentanyls and other μ opioid receptor agonists on the electrical activity of respiratory muscles in the rat

D Cavallo, E Kelly, G Henderson… - Frontiers in …, 2023 - frontiersin.org
… the differential effects of the fentanyls and morphine on … rat vas deferens where high efficacy
μ opioid agonists inhibit … a full concentration-response analysis for each agonist in situ. …

[HTML][HTML] New Insights into the Opioid Analgesic Profile of cis-(−)-N-Normetazocine-derived Ligands

G Costanzo, R Turnaturi, C Parenti, S Spoto, S Piana… - Molecules, 2023 - mdpi.com
… In the mouse vas deferens (MVD) assay, compound 3 showed an antagonist effect
against … identical to that of (−)-morphine. Moreover, as different properties of its N-substituent …

[HTML][HTML] Biased opioid ligands

A Faouzi, BR Varga, S Majumdar - Molecules, 2020 - mdpi.com
agonist which produced a full antinociceptive effect in the … effect of Kurkinorin compared to
morphine (assessed … ) with 0.8 nM potency in mouse vas deferens, first isolated from the skin …

FBNTI, a DOR-selective antagonist that allosterically activates MOR within a MOR–DOR heteromer

E Akgün, MM Lunzer, D Tian, M Ansonoff, J Pintar… - Biochemistry, 2020 - ACS Publications
… The in vivo studies started with an assessment of the opioid agonist … the DOR-selective mouse
vas deferens (MVD) assay to … when morphine (10’ peak time) at its ED 50 dose of 50 pmol/…

[HTML][HTML] Fenfluramine acts as a positive modulator of sigma-1 receptors

P Martin, PAM de Witte, T Maurice, A Gammaitoni… - Epilepsy & Behavior, 2020 - Elsevier
… was assessed by the mouse vas deferens isometric … Agonist and antagonist activities were
assessed using human recombinant receptors expressed in HEK-293 cells (β 1 adrenergic