[PDF][PDF] HAMSTER VAS DEFERENS CONTAINS 6-OPIOID RECEPTORS zyxwvutsrqponmlkjihgfedcbaZYXWVUTSRQPONMLKJIH
AT McKnight, AD Corbett, M Marcoli, HW Kosterlitz - academia.edu
… of the isolated vas deferens of the mouse were inhibited by morphine, … vas deferens of the
hamster for the possible presence of opioid receptors at which morphine has no agonist action…
hamster for the possible presence of opioid receptors at which morphine has no agonist action…
Effects of CA1 α2-adrenergic receptors on morphine-induced exploratory behaviors.
E Beirami… - Physiology & …, 2024 - search.ebscohost.com
… 1) To assess the potential role of morphine in anxiety-related … of mu-opioid receptors agonist,
morphine (6 mg/kg), induced … from sympathetic varicosities of the mouse vas deferens. Br J …
morphine (6 mg/kg), induced … from sympathetic varicosities of the mouse vas deferens. Br J …
[PDF][PDF] Seyedhosseini Tamijani SM Effects of CA1 α2-adrenergic receptors on morphine-induced exploratory behaviors
E Beirami - Physiology and Pharma - ppj.phypha.ir
… 1) To assess the potential role of morphine in anxiety-related … of mu-opioid receptors agonist,
morphine (6 mg/kg), induced … from sympathetic varicosities of the mouse vas deferens. Br J …
morphine (6 mg/kg), induced … from sympathetic varicosities of the mouse vas deferens. Br J …
[HTML][HTML] A systematic review of inverse agonism at adrenoceptor subtypes
… opioid receptors by pre-treatment with morphine [20,53]. Of note, … behaved as a partial
agonist in rat vas deferens. … the receptor number, as assessed by radioligand binding in HepG2 …
agonist in rat vas deferens. … the receptor number, as assessed by radioligand binding in HepG2 …
[PDF][PDF] PREMATURE EJACULATION–POTENTIAL ROLE OF α2-ADRENOCEPTOR AGONISTS FOR SYMPTOMATIC TREATMENT
J Lehtimäki - utupub.fi
… by triggering contractions in the vas deferens, seminal vesicles, … agonist to prevent any effects
on presynaptic α2-adrenergic … To assess the agonistic effects of fadolmidine on the rodent …
on presynaptic α2-adrenergic … To assess the agonistic effects of fadolmidine on the rodent …
[HTML][HTML] Comparison of the effects of fentanyls and other μ opioid receptor agonists on the electrical activity of respiratory muscles in the rat
D Cavallo, E Kelly, G Henderson… - Frontiers in …, 2023 - frontiersin.org
… the differential effects of the fentanyls and morphine on … rat vas deferens where high efficacy
μ opioid agonists inhibit … a full concentration-response analysis for each agonist in situ. …
μ opioid agonists inhibit … a full concentration-response analysis for each agonist in situ. …
[HTML][HTML] New Insights into the Opioid Analgesic Profile of cis-(−)-N-Normetazocine-derived Ligands
G Costanzo, R Turnaturi, C Parenti, S Spoto, S Piana… - Molecules, 2023 - mdpi.com
… In the mouse vas deferens (MVD) assay, compound 3 showed an antagonist effect
against … identical to that of (−)-morphine. Moreover, as different properties of its N-substituent …
against … identical to that of (−)-morphine. Moreover, as different properties of its N-substituent …
[HTML][HTML] Biased opioid ligands
… agonist which produced a full antinociceptive effect in the … effect of Kurkinorin compared to
morphine (assessed … ) with 0.8 nM potency in mouse vas deferens, first isolated from the skin …
morphine (assessed … ) with 0.8 nM potency in mouse vas deferens, first isolated from the skin …
FBNTI, a DOR-selective antagonist that allosterically activates MOR within a MOR–DOR heteromer
E Akgün, MM Lunzer, D Tian, M Ansonoff, J Pintar… - Biochemistry, 2020 - ACS Publications
… The in vivo studies started with an assessment of the opioid agonist … the DOR-selective mouse
vas deferens (MVD) assay to … when morphine (10’ peak time) at its ED 50 dose of 50 pmol/…
vas deferens (MVD) assay to … when morphine (10’ peak time) at its ED 50 dose of 50 pmol/…
[HTML][HTML] Fenfluramine acts as a positive modulator of sigma-1 receptors
P Martin, PAM de Witte, T Maurice, A Gammaitoni… - Epilepsy & Behavior, 2020 - Elsevier
… was assessed by the mouse vas deferens isometric … Agonist and antagonist activities were
assessed using human recombinant receptors expressed in HEK-293 cells (β 1 adrenergic …
assessed using human recombinant receptors expressed in HEK-293 cells (β 1 adrenergic …