Synthesis of new pyrazolone and pyrazole-based adamantyl chalcones and antimicrobial activity
R Al-Saheb, S Makharza, F Al-Battah… - Bioscience …, 2020 - portlandpress.com
… were prepared by condensation of 1-adamantyl methyl ketone with pyridine-2-… adamantyl
chalcone compounds were prepared, wherein the chalcone moiety is an intermediate to new …
chalcone compounds were prepared, wherein the chalcone moiety is an intermediate to new …
Discovery of new chalone adamantyl arotinoids having RXRα-modulating and anticancer activities
M Ao, X Hu, Y Qian, B Li, J Zhang, Y Cao, Y Zhang… - Bioorganic …, 2021 - Elsevier
… , a new series of chalcone adamantly arotinoids (chalcone AdArs) derived from RAR antagonist
MX781, are synthesized, … , a new class of chalcone AdArs was synthesized as anticancer …
MX781, are synthesized, … , a new class of chalcone AdArs was synthesized as anticancer …
Synthesis and bioactivity of thiosemicarbazones containing adamantane skeletons
VH Pham, TPD Phan, DC Phan, BD Vu - Molecules, 2020 - mdpi.com
… In this study, 4-(1-adamantyl)-3-thiosemicarbazide (1) was synthesized by the reaction of
adamantan-1-yl isothiocyanate (Sigma Aldrich, MO, USA) with 80% hydrazine hydrate solution (…
adamantan-1-yl isothiocyanate (Sigma Aldrich, MO, USA) with 80% hydrazine hydrate solution (…
[PDF][PDF] Antiviral and antimicrobial applications of chalcones and their derivatives: From nature to greener synthesis
MH Nematollahi, M Mehrabani, Y Hozhabri… - Heliyon, 2023 - cell.com
… on the antibacterial and antiviral effects of chalcones and their … of greener techniques for
synthesizing these compounds are … , the antimicrobial activity of five pyrazole-based adamantyl …
synthesizing these compounds are … , the antimicrobial activity of five pyrazole-based adamantyl …
Synthesis and in vitro antibacterial, antifungal, anti-proliferative activities of novel adamantane-containing thiazole compounds
… retinoid CD437 was also reported as a promising anticancer … adamantane-based anticancer
drug for the treatment of advanced solid tumors 12 . Opaganib induces its anticancer activity …
drug for the treatment of advanced solid tumors 12 . Opaganib induces its anticancer activity …
Recent progresses in chalcone derivatives as potential anticancer agents
J Yang, J Lv, S Cheng, T Jing, T Meng… - Anti-Cancer Agents …, 2023 - ingentaconnect.com
… The antitumor activity of the coumarin-chalcone hybrid (11) was stronger than xanthohumol,
and it could induce apoptosis of cancer cells by stimulating intracellular reactive oxygen …
and it could induce apoptosis of cancer cells by stimulating intracellular reactive oxygen …
Chalcone derivatives: Role in anticancer therapy
Y Ouyang, J Li, X Chen, X Fu, S Sun, Q Wu - Biomolecules, 2021 - mdpi.com
… chalcones as potential anticancer agents has inspired many efforts directed to developing
novel synthetic chalcones with anticancer properties. … of the chalcone structure have promoted …
novel synthetic chalcones with anticancer properties. … of the chalcone structure have promoted …
Isatin-Schiff's base and chalcone hybrids as chemically apoptotic inducers and EGFR inhibitors; design, synthesis, anti-proliferative activities and in silico evaluation
EA Fayed, RRE Eldin, ABM Mehany… - Journal of Molecular …, 2021 - Elsevier
… base and chalcone were synthesized and screened for their anticancer activities against …
All the tested compounds exhibited moderate to high antitumor activity with IC 50 ranging from …
All the tested compounds exhibited moderate to high antitumor activity with IC 50 ranging from …
[PDF][PDF] Chalcone Derivatives: Role in Anticancer Therapy. Biomolecules 2021, 11, 894
Y Ouyang, J Li, X Chen, X Fu, S Sun, Q Wu - 2021 - researchgate.net
… Synthetic Chalcone Derivatives … occurring chalcones as potential anticancer agents has
inspired many efforts directed to developing novel synthetic chalcones with anticancer properties…
inspired many efforts directed to developing novel synthetic chalcones with anticancer properties…
Novel Adamantane-Linked Isothiourea Derivatives as Potential Chemotherapeutic Agents: Synthesis, Structural Insights, and Antimicrobial/Anti-Proliferative Profiles
FAM Al-Omary, N Alvarez, LS Al-Rasheed, N Veiga… - ACS …, 2023 - ACS Publications
… In this study, two adamantane-linked isothiourea derivatives containing a common 4-…
of the adamantane/isothiourea combination to render auspicious scaffolds for new potential …
of the adamantane/isothiourea combination to render auspicious scaffolds for new potential …