… studies of their biological activities have yet to be reported. … A solution of β-carbolin-1-one
thiohydantoin 5a (105 mg, 0.24 … , we studied their related structure–activity relationship by the …

… review summarizes the development in synthetic methods of THβCs and their comprehensive
biological activities over the … The SAR studies have demonstrated that the introduction of …

… pharmacological potentialities and their derivatives have attracted a great deal of interest due
to their wide range of biological activities. β-… The studies reveal that the synthetic strategies …

… to synthesize cis- and trans diastereomers to understand the effect of specific stereochemistry
on the biological activity. … Further SAR investigation on this lead compound to improve the …

… strategy, and their inhibitory activities … in the biological activities. Furthermore, the compounds
(11g–j, 12g–j and 13g–j) linked with alkanolamine presented more potent inhibitory activity …

… the structure activity relationship for this class of compounds. … Furthermore, the synthesis
and biological activity of TBHCs … tetrahydro-2-tosyl-9H-β-carbolin-4-ones 134, which could be …

… the progress on the synthesis and biological activities of this … investigate the possible
structure-activity relationship for this … )-H of the aryl ring of aryl(β-carbolin-1yl)methanones has also …

… to the structure-activity relationship studies performed in our … promising improved biological
activity. Unfortunately, neither … biology and strategies to delay emergence and spread. Int. J. …

… Interestingly, the above SAR of 8 for AChE is very similar to that of 2-aryl-β-carbolin-2-ium
salts … In fact, 8 can be considered as simple analogues of 2-aryl-β-carbolin-2-niums [24]. …

… DYRK1A is involved in multiple biological functions. For … Last but not least, new
strategies are being developed for in … Some investigators conducted SAR studies on …