Unexpected discovery of dichloroacetate derived adenosine triphosphate competitors targeting pyruvate dehydrogenase kinase to inhibit cancer proliferation

SL Zhang, X Hu, W Zhang, KY Tam - Journal of medicinal …, 2016 - ACS Publications
Pyruvate dehydrogenase kinases (PDKs) have recently emerged as an attractive target for
cancer therapy. Herein, we prepared a series of compounds derived from dichloroacetate …

Unexpected Discovery of Dichloroacetate Derived Adenosine Triphosphate Competitors Targeting Pyruvate Dehydrogenase Kinase To Inhibit Cancer Proliferation

SL Zhang, X Hu, W Zhang… - Journal of medicinal …, 2016 - pubmed.ncbi.nlm.nih.gov
Pyruvate dehydrogenase kinases (PDKs) have recently emerged as an attractive target for
cancer therapy. Herein, we prepared a series of compounds derived from dichloroacetate …

Unexpected Discovery of Dichloroacetate Derived Adenosine Triphosphate Competitors Targeting Pyruvate Dehydrogenase Kinase To Inhibit Cancer Proliferation.

SL Zhang, X Hu, W Zhang, KY Tam - Journal of Medicinal Chemistry, 2016 - europepmc.org
Pyruvate dehydrogenase kinases (PDKs) have recently emerged as an attractive target for
cancer therapy. Herein, we prepared a series of compounds derived from dichloroacetate …

Unexpected Discovery of Dichloroacetate Derived AdenosineTriphosphate Competitors Targeting Pyruvate DehydrogenaseKinase To Inhibit Cancer Proliferation

SL Zhang, X Hu, W Zhang, KY Tam - 2016 - repository.um.edu.mo
Pyruvate dehydrogenase kinases (PDKs) have recently emerged as an attractive target for
cancer therapy. Herein, we prepared a series of compounds derived from dichloroacetate …

Unexpected Discovery of Dichloroacetate Derived Adenosine Triphosphate Competitors Targeting Pyruvate Dehydrogenase Kinase to Inhibit Cancer Proliferation

SL Zhang, X Hu, W Zhang, KY Tam - 2016 - repository.um.edu.mo
Pyruvate dehydrogenase kinases (PDKs) have recently emerged as an attractive target for
cancer therapy. Herein, we prepared a series of compounds derived from dichloroacetate …