… with significant antinociceptive activity and reduced excitatory effects (93.94). Because the
antagonist capsazepine does not appear to be analgesic (95), capsaicin analogues that show …

… the emerging new evidence which demonstrate paradoxical, … the first competitive capsaicin
antagonist, capsazepine. The … specific TRPV1 antagonist inhibited capsaicin-induced release …

… receptor antagonist, capsazepine (10 nmol in 0.4 μl), into the dPAG blocked the capsaicin-induced …
, indicating that the VR1 receptor may contribute to this antinociception. In this report, …

… Our results provide evidence for the involvement of … not yield antinociceptive effects on
capsaicin-induced nociception, … and/or spinal level, thus binding mainly μ-opioid receptors, and …

… Dickenson AH, Dray A: Selective antagonism of capsaicin by capsazepine: evidence for
a spinal receptor site in capsaicin-induced antinociception. Br J Pharmacol 1991; 104(4):1045-…

… of capsazepine (CPZ) as a blocker of the ion channel TRPV1 (transient receptor potential …
(15,35)) have been identified with potent antagonism (IC5o<100nM) of capsaicin-induced …

… We used the vanilloid receptor antagonist capsazepine to establish the role of the vanilloid
… : Evidence for a spinal receptor site in capsaicin-induced antinociception. Br J Pharmacol …

… It has the unique property of selectively activating polymodal nociceptors following …
Capsazepine, a new competitive capsaicin receptor antagonist, could reverse the antinociceptive …

… Dickenson AH, Dray A (1991) Selective antagonism of capsaicin by capsazepine:
evidence for a spinal receptor site in capsaicin-induced antinociception. …

… ability of capsazepine to block capsaicin induced calcium uptake… There is evidence that
TRPV1 also play a role in bone … number of receptors and ion channels such as transient receptor …