… with [18F]fluoropropyl tosylate as the labelling reagent. Here we report the development
of a … the reagent was used without separate purification in the labelling of 2β-carbomethoxy-3β-(4…

… With both fluorescent reagents, DAT on the cell surface could be … , with 5 and 9 displaying
labeling that could be blocked with … The possibility of using this ligand for the direct labeling of …

… labelling with radionuclides such as 11C, 18F, 76Br, 1231, 1251 and 3H. Here we also report
the labelling … we have extended the labelling reactions to include 12SI-labelling of [l251]3, […

… from the same intermediate, the 2β-carbomethoxy-3β-(4‘-… Tropane 2 was then
converted to the 2β-carbomethoxy-3β-[4‘… corresponding desmethyl precursors 2β-carbomethoxy-3β-[4‘…

… ynylnortropane derivatives consisted of adding a Lipshutz reagent 22 (Bu 3 SnCuBuCNLi 2
) … In view of the promising in vitro results, we are currently labeling and testing compounds 3c,…

… Our aim in this work was to employ precursors for labelling of ['251]a-CIT and [1251]p-CIT
that were more easy to prepare than the trialkyltin precursor previously reported'. In addition, …

… In the present study, YP256 was labeled with 123 I by iododestannylation of the trimethylstannyl
precursor, and the time course of 123 I distribution in brain was assessed by SPECT …

… -vinyl halide group to the meta-position of the 3β-phenyl ring. We report here the … 2β-carbomethoxy-3β-(3‘-((Z)-2-iodoethenyl)phenyl)nortropane
(mZIENT, 1) 21 and 2β-carbomethoxy-3β…

… We found that the related reagents 1-hydoxybenzotriazole (HOBt) and 1-hydroxy-7-… The
product that was produced by both reagents, which eluted at 12.6 min under these conditions (…

… A chase study with the DAT ligand 2β-carbophenoxy-3β-(4-chlorophenyl)tropane (9, RTI-113)
failed to displace [ 18 F]1, indicating that [ 18 F]1 is specific to the SERT. The in vivo …