… , Natick, USA), a highly selective adenosine A 2A receptor agonist, to various parts of the rat
brain, … is a highly selective adenosine A 2A receptor agonist. Adenosine A 2A receptors are …

… Development of A2A receptor antagonists During the past 20 years, a … adenosine receptor
agonists and antagonists have been developed 4,", including selective A2A receptor agonists …

… A 1 /dopamine D 1 receptors in the ventral and dorsal striatum are at … of adenosine receptor
antagonists like caffeine and for the motor depressant actions of adenosine receptor agonists…

… and small molecules has been validated by the US Food and Drug Administration’s approval
of regadenoson (19, Figure 6), a selective A 2A adenosine receptor agonist that increases …

… (12, 13) A 2A −D 2 receptor heteromers were found to be constitutive because they were …
D 2 receptor agonist exposure. However, the stoichiometry of A 2A −D 2 receptor heteromers is …

… 2A and A 2B receptors stimulate this enzyme via a G s protein (Gao and Jacobson, 2007).
In this study, we focused on agonists for the human adenosine A 2A receptor (hA 2A receptor), …

… Since the order of potency of adenosine receptor agonist suggested that A2a receptors are
… effect of adenosine on IL-12 production, we tested the effect of adenosine in A2a receptor-…

… New, non-adenosine, high-potency agonists for the human adenosine A2B receptor with
an improved selectivity profile compared to the reference agonist N-…

… More recently, we found that CGS21680, a selective adenosine A 2A receptor agonist,
also promoted sleep when it was infused into or near the prostaglandin D 2 -sensitive zone, …

… cerebral cortex, where adenosine A 1 receptors are predominant, displays a mixed A 2A /A
1 receptor pharmacology. We now use adenosine A 1 and A 2A receptor knockout mice to …