… 2A and A 2B receptors stimulate this enzyme via a G s protein (Gao and Jacobson, 2007).
In this study, we focused on agonists for the human adenosine A 2A receptor (hA 2A receptor), …

… Development of A2A receptor antagonists During the past 20 years, a … adenosine receptor
agonists and antagonists have been developed 4,", including selective A2A receptor agonists …

… responsible for the motor stimulant effects of adenosine receptor antagonists like caffeine
and for the motor depressant actions of adenosine receptor agonists. A major mechanism for a …

… , Natick, USA), a highly selective adenosine A 2A receptor agonist, to various parts of the rat
brain, … is a highly selective adenosine A 2A receptor agonist. Adenosine A 2A receptors are …

… Synthetic A2A selective AR agonists are currently undergoing … A2A AR agonist treatment,
mechanisms of A2A AR agonist action and considerations for synthetic A2A AR agonist …

… Structures of adenosine receptor agonists in clinical trials for various conditions * . …
A2B receptor with an improved selectivity profile compared to the reference agonist N-…

… A2A receptor agonists developed in the period 2005-2017, their selectivity regarding other
adenosine receptors … Two important features of the adenosine A2A receptor are important for …

… and small molecules has been validated by the US Food and Drug Administration’s approval
of regadenoson (19, Figure 6), a selective A 2A adenosine receptor agonist that increases …

… Adenosine A2A receptors were cloned about ten years ago and are known to be well conserved
among mammals. Rather selective agonists … slices, adenosine A2A receptor agonists do …

… of agonist selectivity in defining the signalling pathways in cells with multiple adenosine
receptor … The events that are inhibited by adenosine A2A receptor agonist treatment are shown, …