… In the present study, a number of dopamine receptor agonists have been examined for their
… the dopamine receptor selectivity and affinities for a variety of dopamine receptor agonists. …

… dopamine receptor binding affinities of all currently approved dopamine receptor agonist …
Dihydroergocryptine and lisuride displayed higher comparative affinities (Ki ¼ 35.4 and …

… Dopamine D 2 receptors, similar to other G-protein-coupled receptors, exist in a high- and
low-affinity state for agonists… for detecting D 2 receptor agonist high-affinity states, we discuss …

… Overall, the series of dopamine receptor agonists in this study demonstrated a wider
range of affinities for in vitro binding to dopamine D 3 and DZL receptors, 372-fold and 557-fold …

… We postulate that haloperidol and dopamine respectively label the antagonist and agonist
states of dopamine receptors. This would explain the affinity of antagonists and agonists …

… 18,19 To find complete receptor-affinity data for DAs from experiments on cloned human
dopamine receptors when the receptors were in the "high-affinity state, ''2 a search of …

… The adaptation of receptors to agonist occupancy, as … of receptor molecules; the affinity
of the receptor for the agonist is … "receptor'-binding data, have been drawn eg for dopamine (…

… A subset of receptors existing in a high affinity state for agonists is detected in washed
membrane preparations, in which the coupling to intracellular G-proteins may have become …

… the D 2 dopamine receptor, the relation between the ability of agonists and inverse agonists
to … We have determined the affinities of a range of agonists and inverse agonists at the D 2 …

… affinities of agonists for G protein-coupled (higher affinity, K h ) and -uncoupled (lower affinity,
K l ) forms of the receptor… the K l /K h ratio for agonists and their relative efficacy (De Lean et …