The antiprotozoal activity of methylated flavonoids from Ageratum conyzoides L.

AMM Nour, SA Khalid, M Kaiser, R Brun… - Journal of …, 2010 - Elsevier
… ), we have recently reported on the antiprotozoal activity of Sudanese plants of the Asteraceae
… In the present communication we report on the isolation, identification and antiprotozoal

Evaluation of the in vitro trypanocidal activity of methylated flavonoid constituents of Vitex simplicifolia leaves

N Nwodo, F Okoye, D Lai, A Debbab, M Kaiser… - … and alternative medicine, 2015 - Springer
… similar flavonoids or its derivatives have been reported to possess trypanocidal activity against
… the trypanocidal activity of some methylated flavonoid derivatives from Vitex simplicifolia. …

Correlation study on methoxylation pattern of flavonoids and their heme-targeted antiplasmodial activity

S Ortiz, PG Vásquez-Ocmín, S Cojean, C Bouzidi… - Bioorganic …, 2020 - Elsevier
… No correlation was observed between the methoxylation pattern and the antiparasitic activity,
either for the 3D7 chloroquine-sensitive or for the W2 chloroquine-resistant P. falciparum …

Antitrypanosomal and antileishmanial activities of flavonoids and their analogues: in vitro, in vivo, structure-activity relationship, and quantitative structure-activity …

D Tasdemir, M Kaiser, R Brun, V Yardley… - Antimicrobial agents …, 2006 - Am Soc Microbiol
antiprotozoal activities of two flavonoid glycosides (17). This prompted us to screen a large
set of polyphenolic compounds mainly of a flavonoid … and leishmanicidal activities. As …

Antileishmanial and antitrypanosomal activities of flavonoids

F Nardella, JB Gallé, M Bourjot, B Weniger… - Natural Antimicrobial …, 2018 - Springer
… The selectivity index (SI) was calculated as the ratio of cytotoxic activity to antiparasitic
activity. We also recorded the in vivo data when they were available. We plotted the data …

Methylation of flavonoids: Chemical structures, bioactivities, progress and perspectives for biotechnological production

N Koirala, NH Thuan, GP Ghimire, D Van Thang… - Enzyme and microbial …, 2016 - Elsevier
… of methylated flavonoids using … methylated flavonoids focusing on their occurrence and
bioactivities is given in Table 1. Pharmaceutically significant flavonoids and their methylated

[PDF][PDF] Trypanocidal and leishmanicidal activities of flavonoids from Argentine medicinal plants

VP Sülsen, SI Cazorla, FM Frank… - American Journal of …, 2007 - researchgate.net
… As part of our ongoing search of antiparasitic compounds from natural sources, the
trypanocidal activity of selected Argentine medicinal plants has been reported by our group.Among …

Antiprotozoal activity of Melampyrum arvense and its metabolites

H Kirmizibekmez, I Atay, M Kaiser, R Brun… - Phytotherapy …, 2011 - Wiley Online Library
… the composition of 12 was identified by GC‐MS after methylation. Luteolin (7) appeared as
the most … arvense and the first report of the antiprotozoal effect of Melampyrum species and its …

Anti-African trypanocidal and antimalarial activity of natural flavonoids, dibenzoylmethanes and synthetic analogues

DAP dos Santos, PAC Braga… - Journal of Pharmacy …, 2009 - academic.oup.com
… to improve activity and selectivity, our results could help in directing the rational design of
flavonoid and dibenzoylmethane derivatives as potent and effective antiprotozoal agents. All …

[HTML][HTML] In vitro antileishmanial and antitrypanosomal activities of flavanones from Baccharis retusa DC.(Asteraceae)

SS Grecco, JQ Reimão, AG Tempone, P Sartorelli… - Experimental …, 2012 - Elsevier
… 1 did not show antiparasitic activity. Compound 2 was subjected to a methylation procedure
to … to one methoxyl group at C-7 in related flavonoids is important to the antiparasitic activity. …