[HTML][HTML] The biological activities of butyrylcholinesterase inhibitors
S Zhou, G Huang - Biomedicine & pharmacotherapy, 2022 - Elsevier
… Various studies have suggested that BuChE inhibition is a potential strategy for the treatment
… biological activity of selectivity butyrylcholinesterase inhibitors (BuChEI) in the past decade. …
… biological activity of selectivity butyrylcholinesterase inhibitors (BuChEI) in the past decade. …
2-Phenylbenzofuran derivatives as butyrylcholinesterase inhibitors: synthesis, biological activity and molecular modeling
… evaluated as cholinesterase inhibitors. The biological assay experiments showed that
most of the compounds displayed a clearly selective inhibition for butyrylcholinesterase (BChE), …
most of the compounds displayed a clearly selective inhibition for butyrylcholinesterase (BChE), …
Synthesis, molecular docking, and biological activity of 2-vinyl chromones: Toward selective butyrylcholinesterase inhibitors for potential Alzheimer's disease …
GF Makhaeva, NP Boltneva, SV Lushchekina… - Bioorganic & Medicinal …, 2018 - Elsevier
We investigated the biological activity of a series of substituted chromeno[3,2-c]pyridines,
including compounds previously synthesized by our group and novel compounds whose …
including compounds previously synthesized by our group and novel compounds whose …
In silico drug discovery of Acetylcholinesterase and Butyrylcholinesterase enzymes inhibitors based on Quantitative Structure-Activity Relationship (QSAR) and drug …
… The structures and their experimental values of the biological activity IC50 (ie, concentration
that is required for 50% inhibition of biological activity) were taken from the published …
that is required for 50% inhibition of biological activity) were taken from the published …
Discovery, biological evaluation, and crystal structure of a novel nanomolar selective butyrylcholinesterase inhibitor
B Brus, U Kosak, S Turk, A Pislar… - Journal of medicinal …, 2014 - ACS Publications
… Butyrylcholinesterase (BChE) is regarded as a promising drug target as its levels and
activity … To discover novel BChE inhibitors, we used a hierarchical virtual screening protocol …
activity … To discover novel BChE inhibitors, we used a hierarchical virtual screening protocol …
Acetylcholinesterase and butyrylcholinesterase inhibitory activity of Pinus species essential oils and their constituents
M Bonesi, F Menichini, R Tundis… - … of enzyme inhibition …, 2010 - Taylor & Francis
This study aimed to investigate the acetylcholinesterase (AChE) and butyrylcholinesterase (BChE)
inhibitory activity of the essential oils from Pinus nigra subsp. nigra, P. nigra var. …
inhibitory activity of the essential oils from Pinus nigra subsp. nigra, P. nigra var. …
[PDF][PDF] Butyrylcholinesterase: structure and physiological importance
AN Çokuğraş - Turk J Biochem, 2003 - scholar.archive.org
… is involved three different enzymatic activities in its structure like … activity of butyrylcholinesterase
becomes more important in scavenging of organophosphate and carbamate inhibitors …
becomes more important in scavenging of organophosphate and carbamate inhibitors …
Flavonols and 4-thioflavonols as potential acetylcholinesterase and butyrylcholinesterase inhibitors: Synthesis, structure-activity relationship and molecular docking …
… Moreover, sulfur containing compounds usually possess good biological activities, which
can be speculated by their ability to scavenge free radicals, high potential of chelating metal …
can be speculated by their ability to scavenge free radicals, high potential of chelating metal …
… alkaloids of norbelladine-type as inspiration for development of highly selective butyrylcholinesterase inhibitors: Synthesis, biological activity evaluation, and docking …
AA Mamun, F Pidaný, D Hulcová, J Maříková… - International Journal of …, 2021 - mdpi.com
… inhibitors and the N-methyl-d-aspartate receptor antagonist, memantine. Emerging evidence
strongly supports the relevance of targeting butyrylcholinesterase (… ) and BuChE inhibition …
strongly supports the relevance of targeting butyrylcholinesterase (… ) and BuChE inhibition …
Design, synthesis and biological evaluation of novel carbamates as potential inhibitors of acetylcholinesterase and butyrylcholinesterase
J Wu, M Pistolozzi, S Liu, W Tan - Bioorganic & Medicinal Chemistry, 2020 - Elsevier
… inhibitors of elAChE and eqBChE, respectively. Since ChEs activity and susceptibility to
inhibitors … of BMC-3 and BMC-16 to repress the activity of human ChEs (Table 1). By comparing …
inhibitors … of BMC-3 and BMC-16 to repress the activity of human ChEs (Table 1). By comparing …
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