The potent cocaine analog 2fl-carbomethoxy-3fl-(4-fluorophenyl)-tropane(CFT, also designated
WIN 35,428) was tritiated and evaluated as a molecular probe for cocaine receptors in …

Human and bovine dopamine transporters (DAT) demonstrate discrete functional differences
in dopamine (DA), 1-methyl-4-phenylpyridium (MPP + ) transport, and cocaine analog …

Using the MM2‐87 program and parameter set, conformational analyses have been performed
on cocaine (1), the potent analog 2β‐carbomethoxy‐3β‐(4‐fluorophenyl)tropane (CFT, 2)…

The present study reports the ion dependency of 2β‐carbomethoxy‐3β‐(4‐fluorophenyl)[ 3
H]tropane ([ 3 H]‐ CFT) binding to the dopamine transporter in the rat striaturn. The results …

A synthesis method has been developed for the labelling of N‐(3‐[ 18 F]fluoropropyl)‐2β‐carbomethoxy‐3β‐(4‐fluorophenyl)nortropane
([ 18 F]β‐CFT‐FP), a potential radioligand for …

… 2/3-Carbomethoxy-3/3-(4-chlorophenyl)tropane (2) was prepared in 55 … 4chlorophenyl)magnesium
bromide as previously reported by Carroll.23 The Michael addition of (4-chlorophenyl…

Purpose This study compares 2β-carbomethoxy-3β-(4-[ 18 F]fluorophenyl)tropane ([ 18 F]β-CFT)
and N-(3-[ 18 F]fluoropropyl)-2β-carbomethoxy-3β-(4-fluorophenyl)nortropane ([ 18 F]β-…

A dopamine transporter (DAT) ligand 2β‐carbomethoxy‐3β‐(4‐fluoro‐phenyl)‐8‐(2‐[ 18 F]fluoroethyl)nortropane
([ 18 F]β‐CFT‐FE) was synthesized and evaluated in comparison with [ …

… 18 F radioactivity accumulation of 2β-carbomethoxy-3β-(4-chlorophenyl)-8-(3… 4-chlorophenyl
group instead of the 4-fluorophenyl of [ 18 F]β-CFT-FP [34]. FPCT was reported to have four …

2β‐Carbomethoxy‐3β‐(4‐fluorophenyl)‐[N‐ 11 C‐methyl]tropane, a potent inhibitor of
dopamine transport, was prepared by N‐methylation of the appropriate nor‐methyl precursor in …