… inhibited intracellular hCES2A in living HepG2 cells. In summary, this study proposed an
integrated strategy to find hCES2A inhibitors … responsible for hCES2A inhibition, which would …

… hCES2A inhibitory assay The enzyme inhibitory assays were conducted according to the …
As for the inhibitory assay of hCES2A, it was evaluated by using FD as a fluorescent probe [25]. …

… 3-fold improvement inhibition in the intracellular hCES2A inhibition assays, suggesting that
the … Enzyme inhibition assays In this study, hCES2A inhibition assay was conducted using FD …

… was capable of inhibiting intracellular hCES2A in living cells … choices for the development
of hCES2A inhibitors, while B7 is a … , time-dependent inhibition assays of B7 on hCES2A were …

… inhibitory effects against hCES2A are assayed using a fluorescence-based biochemical
assay… are found with strong to moderate hCES2A inhibition activity. Primary structure–activity …

… real hCES2A activity in complex systems and find more efficacious hCES2A inhibitors with
… Next, a microplate-based high-throughput screening assay identified hCES2A inhibitors from …

… used to assay the inhibition of intracellular hCES2A by … hCES2A inhibitors. Some of them
can be used as leading compounds for development of more efficacious hCES2A inhibitors to …

… their inhibitory effects on hCES1A and hCES2A were assayed … –inhibition relationships of
ginsenosides as hCES inhibitors … were potent inhibitors against both hCES1A and hCES2A, …

… Meanwhile, the authors also assay the inhibition constants of these … hCES2A inhibitors
screening, respectively [83]. Among them, telmisartan and nitrendipine displayed strong inhibitory …

… Currently, the search for new hCES2A inhibitors is an … Prior to further experiments, we
performed an CCK-8 assay on 20w… 20w as a novel, potent hCES2A inhibitor, which could be used …