… Altogether it is suggested that ß-CFT-FP should have a higher … We report the labelling of
ß-CFT-FP with fluorine-18 or carbon-11 to … using V as the labelled reagent as described above. …

… the labelling reagent in the alkylation of nor-β-CFT. An equivalent molar ratio of nor-β-CFT to
1,3… ) incorporation of [18F]fluoropropyl tosylate into [18F]β-CFT-FP, see Figure 3. On a molar …

… C]β-CFT encouraged the further studies to labeled β-CFT with 18 F for PET imaging of dopamine
transporter. PET studies of [ 18 F]β-CFT showed that [ 18 F]β-CFT … reagent, β-CFT 5 was …

… synthesis of nor-β-CFT; and (c) labeling of [ 11 C]β-CFT at the O-… others have successfully
labeled the cocaine congener β-CIT … We note that the conjugate addition of Grignard reagent 4-…

… All other reagents that were purchased from commercial suppliers were either of synthesis
… and ED values for [ 18 F]CFT correspond well with those of other 18 F-labeled radioligands. …

… methyl triflate, i: that this labelling reagent is compatible with the base pentamethylpireridine
… temperatures employed when using the former reagent. A comparison of the product …

… The aim of this study was to develop the electrophilic labeling synthesis of [18F]FDOPA and
[18F]CFT for imaging different aspects of the presynaptic dopaminergic system in vivo with …

… All other reagents were commercially available. All reagents were used without further …
–water mixture) in a sealed reaction vessel containing nor-β-CFT (0.15 mg) and acetone (200 μl). …

… 18 F]β-CFT-FP was studied using two 18 Ffluoroalkylation reagents, [ 18 F]fluoropropyl …
Thus, it was concluded that [ 18 F]β-CFT-FP has potential as a radiotracer for imaging DAT …

… The purpose of this study was to prepare radiolabelled β-CFT-FP using two different [18F]…
In [11C]carboxylation the reaction of [11C]CO2 with a Grignard reagent yields the …