Synthesis and biological evaluation of novel phenylcarbazoles as potential anticancer agents

S Routier, JY Mérour, N Dias, A Lansiaux… - Journal of medicinal …, 2006 - ACS Publications
… We here report the synthesis and biological evaluation of new phenylcarbazole derivatives
designed as potential anticancer agents. Indole and hydroxyindole were used to generate …

Benzylidine pregnenolones and their oximes as potential anticancer agents: synthesis and biological evaluation

AH Banday, SMM Akram, SA Shameem - Steroids, 2014 - Elsevier
The present study reveals the anticancer activity of benzylidine pregnenolones and their
oxime derivatives. The synthesis of the analogs of both series is very simple and involves aldol …

[HTML][HTML] Novel hybrid pyrrolidinedione-thiazolidinones as potential anticancer agents: Synthesis and biological evaluation

N Finiuk, A Kryshchyshyn-Dylevych, S Holota… - European journal of …, 2022 - Elsevier
A series of novel pyrrolidinedione-thiazolidinones was synthesized and subjected to physico-chemical
characteristics. They were screened on a panel of cell lines representing different …

Synthesis and biological evaluation of novel naphthocarbazoles as potential anticancer agents

S Routier, P Peixoto, JY Mérour… - Journal of medicinal …, 2005 - ACS Publications
… We report the efficient synthesis involving palladium-catalyzed reactions and biological
evaluation of new naphthocarbazoles designed as potential anticancer agents. The use of 5- …

Development of potential antitumor agents. Synthesis and biological evaluation of a new set of sulfonamide derivatives as histone deacetylase inhibitors

G Bouchain, S Leit, S Frechette, EA Khalil… - Journal of Medicinal …, 2003 - ACS Publications
A series of sulfonamide hydroxamic acids and anilides have been synthesized and studied
as histone deacetylase (HDAC) inhibitors that can induce hyperacetylation of histones in …

Synthesis and biological evaluation of ursolic acid-triazolyl derivatives as potential anti-cancer agents

S Rashid, BA Dar, R Majeed, A Hamid… - European Journal of …, 2013 - Elsevier
… A library of ursolic acid-triazolyl derivatives modified at C-28 carboxylic position has been
synthesized by employing click chemistry protocol as potential anti-cancer compounds. Click …

Synthesis and biological evaluation of sophoridinol derivatives as a novel family of potential anticancer agents

C Bi, C Zhang, Y Li, S Tang, S Wang… - ACS Medicinal …, 2014 - ACS Publications
Synthesis, structure–activity relationship and biological evaluation of novel nitrogen
mustard sophoridinic acid derivatives as potential anticancer agents. Bioorganic & Medicinal …

Potential antitumor agents. Part 43. Synthesis and biological activity of dibasic 9-aminoacridine-4-carboxamides, a new class of antitumor agent

GJ Atwell, BF Cain, BC Baguley, GJ Finlay… - Journal of medicinal …, 1984 - ACS Publications
… side chain (Tables I and II) are potent antitumor agents both in vitro and in vivo,and this
paper describes the synthesis and biological evaluation of some examples of this new class. …

Design, synthesis, and biological evaluation of novel quinazolinyl-diaryl urea derivatives as potential anticancer agents

JN Chen, XF Wang, T Li, DW Wu, XB Fu… - European journal of …, 2016 - Elsevier
… site of the receptor c-Raf, which was consistent with the biological data. Therefore, compound
8g may be a potent antitumor agent, representing a promising lead for further optimization. …

Synthesis and biological evaluation of novel oxophenylarcyriaflavins as potential anticancer agents

A Bourderioux, V Bénéteau, JY Mérour… - Organic & …, 2008 - pubs.rsc.org
… We report the synthesis and biological evaluation of new oxophenylarcyriaflavins designed
as potential anticancer agents. An efficient synthesis involving palladium-catalyzed Suzuki …