[HTML][HTML] Androgen receptor antagonists for prostate cancer therapy
C Helsen, T Van den Broeck, A Voet… - … -related cancer, 2014 - erc.bioscientifica.com
Medullary thyroid carcinomas (MTC) arise from thyroid parafollicular, calcitonin-producing C-cells
and can occur either as sporadic or as hereditary diseases in the context of familial …
and can occur either as sporadic or as hereditary diseases in the context of familial …
Androgen receptors in endocrine‐therapy‐resistant human prostate cancer
TH van der Kwast, J Schalken… - … journal of cancer, 1991 - Wiley Online Library
… androgen ablation or anti-androgen therapy. In order to gain more insight into the role of the
androgen receptor (AR) in this process, AR and prostate-… in prostatic tumour tissues from pa…
androgen receptor (AR) in this process, AR and prostate-… in prostatic tumour tissues from pa…
Mechanisms of androgen receptor activation in castration-resistant prostate cancer
N Sharifi - Endocrinology, 2013 - academic.oup.com
… of advanced prostate cancer is initiated with androgen deprivation … prostate cancer (CRPC),
which is driven, at least in part, by a continued dependence on the androgen receptor (AR). …
which is driven, at least in part, by a continued dependence on the androgen receptor (AR). …
[HTML][HTML] Androgen receptor and prostate cancer
KE Livermore, J Munkley, DJ Elliott - AIMS Molecular Science, 2016 - aimspress.com
… Androgens drive prostate cancer cell growth via the androgen receptor (AR), which is a
transcription factor essential for prostate cancer cell viability, proliferation and invasion and has …
transcription factor essential for prostate cancer cell viability, proliferation and invasion and has …
Treatment-dependent androgen receptor mutations in prostate cancer exploit multiple mechanisms to evade therapy
MP Steinkamp, OA O'Mahony, M Brogley, H Rehman… - Cancer research, 2009 - AACR
… androgen receptor (AR) that enable activation by antiandrogens occur in hormone-refractory
prostate cancer… reflecting genetic heterogeneity of prostate cancer. Base changes recurring …
prostate cancer… reflecting genetic heterogeneity of prostate cancer. Base changes recurring …
Targeting the androgen receptor pathway in castration-resistant prostate cancer: progresses and prospects
… Androgen receptor (AR) signaling is a critical pathway for prostate cancer cells, and androgen-…
The view of castration-resistant prostate cancer (CRPC) has changed dramatically in the …
The view of castration-resistant prostate cancer (CRPC) has changed dramatically in the …
Amplification and overexpression of androgen receptor gene in hormone-refractory prostate cancer
MJ Linja, KJ Savinainen, OR Saramäki, TLJ Tammela… - Cancer research, 2001 - AACR
… of the androgen receptor (AR) gene in androgen-dependent and -independent prostate cancer
was … Eight benign prostate hyperplasias, 33 untreated and 13 hormone-refractory locally …
was … Eight benign prostate hyperplasias, 33 untreated and 13 hormone-refractory locally …
Splicing of a Novel Androgen Receptor Exon Generates a Constitutively Active Androgen Receptor that Mediates Prostate Cancer Therapy Resistance
SM Dehm, LJ Schmidt, HV Heemers, RL Vessella… - Cancer research, 2008 - AACR
… for prostate cancer (PCa) is androgen ablation, which causes tumor regression by
inhibiting activity of the androgen receptor (AR). Invariably, PCa recurs with a fatal androgen-…
inhibiting activity of the androgen receptor (AR). Invariably, PCa recurs with a fatal androgen-…
Androgen receptor and growth factor signaling cross-talk in prostate cancer cells
ML Zhu, N Kyprianou - Endocr Relat Cancer, 2008 - erc.bioscientifica.com
… Bonaccorsi L, Nosi D, Muratori M, Formigli L, Forti G & Baldi E 2007 Altered endocytosis
of epidermal growth factor receptor in androgen receptor positive prostate cancer cell lines. …
of epidermal growth factor receptor in androgen receptor positive prostate cancer cell lines. …
The androgen axis in recurrent prostate cancer
JL Mohler, CW Gregory, OH Ford III, D Kim… - Clinical cancer …, 2004 - AACR
… Androgen receptor activation in recurrent prostate cancer was suggested by the … The
persistence of androgen receptor protein in prostate cancer independent of circulating androgen …
persistence of androgen receptor protein in prostate cancer independent of circulating androgen …