Mechanisms of action of the 5-HT1B/1D receptor agonists

SJ Tepper, AM Rapoport, FD Sheftell - Archives of neurology, 2002 - jamanetwork.com
… 5-HT 1 receptors and the development of 5-HT receptor agonists with specific affinity for 5-HT
1 receptor subtypes provided evidence for substantial populations of 5-HT 1B receptors on …

Overview of the effects of β-adrenergic receptor agonists on animal growth including mechanisms of action

HJ Mersmann - Journal of animal science, 1998 - academic.oup.com
… β-Adrenergic Receptor Agonists The b-adrenergic receptor agonists are organic molecules
that bind to b-adrenergic receptors such that the agonist-receptor complex activates the Gs …

Receptors, agonists and antagonists

BJ Pleuvry - Anaesthesia & Intensive Care Medicine, 2004 - Elsevier
… The existence of G-proteins came to light when it was observed that stimulation of second
messenger systems such as adenylyl cyclase required not only the receptor agonist but also …

Possible antimigraine mechanisms of action of the 5HT1F receptor agonist LY334370

S Shepheard, L Edvinsson, M Cumberbatch… - …, 1999 - Wiley Online Library
… 5HT 1r receptor agonist LY334370 has other possible antimigraine mechanisms in addition
… to suggest that LY334370 has a central mechanism of action in blocking the transmission of …

Molecular mechanisms of glucocorticoid action and selective glucocorticoid receptor agonists

C Stahn, M Löwenberg, DW Hommes… - Molecular and cellular …, 2007 - Elsevier
… The classical, genomic mechanism of GC-action can be … , such as selective glucocorticoid
receptor agonists (SEGRAs). These … -mentioned mechanisms of glucocorticoid action and give …

User's guide to mechanism of action and clinical use of GLP-1 receptor agonists

CF Shaefer Jr, P Kushner, R Aguilar - Postgraduate Medicine, 2015 - Taylor & Francis
… Glucagon-like peptide-1 (GLP-1) receptor agonists (GLP-1RAs… These drugs provide levels
of GLP-1 receptor agonism many … is to review the mechanism of action and clinical profile of …

[HTML][HTML] Weight loss and maintenance related to the mechanism of action of glucagon-like peptide 1 receptor agonists

J Ard, A Fitch, S Fruh, L Herman - Advances in therapy, 2021 - Springer
… This article aims to inform primary care providers about the mechanism of action of one class
of AOMs, glucagon-like peptide 1 receptor agonists (GLP-1RAs), in weight loss and longer-…

Glucagon-like peptide 1 receptor agonists: cardiovascular benefits and mechanisms of action

JR Ussher, DJ Drucker - Nature Reviews Cardiology, 2023 - nature.com
… Accordingly, in the remainder of this Review, we focus on delineating the mechanisms of
action for GLP1R agonist-mediated cardioprotection (Fig. 3) and consider the major cell types …

A review of GLP‐1 receptor agonists in type 2 diabetes: a focus on the mechanism of action of once‐weekly agents

S Cornell - Journal of clinical pharmacy and therapeutics, 2020 - Wiley Online Library
… GLP-1 receptor agonists for individualized treatment of type 2 diabetes mellitus. Nat Rev …
-1 receptor agonist ameliorates renal injury through its anti-inflammatory action without lowering …

Dopamine receptor agonists: mechanisms underlying autoreceptor selectivity II. Theoretical considerations

D Clark, S Hjorth, A Carlsson - Journal of neural transmission, 1985 - Springer
… -PPP has no detectable agonist activity at normosensitive postsynaptic DA receptors but, in
… feedback mechanism is not responsible for the apparent DA autoreceptor agonist action of …