Synthesis of new chrysin derivatives with substantial antibiofilm activity
S Bhowmik, P Anand, R Das, T Sen, Y Akhter… - Molecular Diversity, 2021 - Springer
Multidrug resistance mechanism of microorganisms towards conventional antimicrobials
nowadays faces a common health problem. So, searching and development of new …
nowadays faces a common health problem. So, searching and development of new …
[PDF][PDF] Synthesis of Some New Chrysin Derivatives and Their Biological Assessment as Antibacterial, Antibiofilm and Antifungal Agent.
Some new derivatives of natural chrysin have been synthesized and evaluated for
antibacterial, antibiofilm and antifungal activities. Three compounds, namely 2a, 2e, 2i …
antibacterial, antibiofilm and antifungal activities. Three compounds, namely 2a, 2e, 2i …
Synthesis, characterization and molecular docking studies of novel 2-amino 3-cyano pyrano[2,3H]chrysin derivatives as potential antimicrobial agents
P Ramesh, CS Reddy, K Suresh Babu… - Medicinal Chemistry …, 2015 - Springer
A series of novel 2-amino 3-cyano 4-aryl pyrano [2, 3 H] chrysin derivatives (3a–m) were
efficiently synthesized by one-pot three-component reaction of aromatic aldehydes …
efficiently synthesized by one-pot three-component reaction of aromatic aldehydes …
Facile synthesis and biological evaluation of chrysin derivatives
N Omonga, Z Zia, H Ghanbour… - Journal of Chemical …, 2021 - journals.sagepub.com
In this paper, novel synthetic methods, including microwave O-alkylation, were used to
produce several chrysin derivatives. These compounds were purified, characterised and …
produce several chrysin derivatives. These compounds were purified, characterised and …
Xanthone synthetic derivatives with high anticandidal activity and positive mycostatic selectivity index values
With the current massive increases in drug-resistant microbial infection as well as the
significant role of fungal infections in the death toll of COVID-19, discovering new antifungals …
significant role of fungal infections in the death toll of COVID-19, discovering new antifungals …
Synthesis and biological evaluation of novel C (7) modified chrysin analogues as antibacterial agents
KS Babu, TH Babu, PV Srinivas, KH Kishore… - Bioorganic & medicinal …, 2006 - Elsevier
The natural product, chrysin (5, 7-dihydroxy flavone), obtained from Oroxylum indicum,
exhibits numerous biological activities including anticancer, anti-inflammatory, and …
exhibits numerous biological activities including anticancer, anti-inflammatory, and …
Click-based synthesis of bromotyrosine alkaloid analogs as potential anti-biofilm leads for SAR studies
S Andjouh, Y Blache - Bioorganic & Medicinal Chemistry Letters, 2015 - Elsevier
A library of triazole-based analogs of bromotyramine alkaloids such as verongamines,
hemibastadins, pseudoceramine D and clavatidine E was designed in order to identify …
hemibastadins, pseudoceramine D and clavatidine E was designed in order to identify …
Antimicrobial activity and docking study of synthesized xanthen-3-on derivatives
E Veljović, S Spirtovic-Halilovic… - Research Journal of …, 2018 - cer.ihtm.bg.ac.rs
Twelve previously synthesized biologically active 2, 6, 7-trihydroxy-9-aryl-3H-xanthen-3-one
derivatives (1-12) were evaluated in vitro for their antimicrobial activity against four bacteria …
derivatives (1-12) were evaluated in vitro for their antimicrobial activity against four bacteria …
In‐house chemical library repurposing: A case example for Pseudomonas aeruginosa antibiofilm activity and quorum sensing inhibition
Abstract Hit, Lead & Candidate Discovery Drug repurposing has become a recent trend in
drug development programs, where previously developed drugs are explored for hit and …
drug development programs, where previously developed drugs are explored for hit and …
Chromene-dihydropyrimidinone and xanthene-dihydropyrimidinone hybrids: design, synthesis, and antibacterial and antibiofilm activities
SJ Santos, FCP Rossatto, NS Jardim, DS Ávila… - New Journal of …, 2023 - pubs.rsc.org
A series of eleven chromene-dihydropyrimidinone and eleven xanthene-
dihydropyrimidinone hybrid compounds were easily synthesized through a sequential …
dihydropyrimidinone hybrid compounds were easily synthesized through a sequential …